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Acetylcholine (CID 187) - Compound BioActivity Data
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Filters: All Data » Ki      
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BioActivity Outcomes:
Active(39)
 
 
Inconclusive(2)
 
 
Unspecified(2)
 
 
Top Targets:
Neur chan LBD(34)
 
 
 
 
7TM GPCR Srsx(1)
 
 
BioAssay Types:
Literature(43)
 
 
 
 
BioActivity Types:
Ki(43)
 
 
 
 
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Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 27    Data Row: 43   Total Pages: 3   Display: Page     
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#SubstanceActivityBioAssayTargetLinks
OutcomeTypeValue [μM]
1
[SID104234160]
Ki 0.0076Displacement of [3H]-cytisine from Alpha4-beta2 Nicotinic acetylcholine receptor of rat brain homogenates [AID239589, Type: Literature]Neuronal acetylcholine receptor subunit beta-2 [gi:6226548]
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2
[SID104234160]
Ki 0.0076Displacement of [3H]-cytisine from Alpha4-beta2 Nicotinic acetylcholine receptor of rat brain homogenates [AID239589, Type: Literature]Neuronal acetylcholine receptor subunit alpha-4 [gi:8469182]
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3
[SID104234160]
Ki 0.011Binding affinity towards rat nicotinic acetylcholine receptor alpha2-beta2 expressed in HEK293 cells using [3H]EB as radioligand [AID145983, Type: Literature]Neuronal acetylcholine receptor subunit beta-2 [gi:6226548]
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4
[SID104234160]
Ki 0.011Binding affinity towards rat nicotinic acetylcholine receptor alpha2-beta2 expressed in HEK293 cells using [3H]EB as radioligand [AID145983, Type: Literature]Neuronal acetylcholine receptor subunit alpha-2 [gi:2851491]
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5
[SID104234160]
Ki 0.03311Displacement of [3H]epibatidine from rat recombinant alpha4beta2 nAChR expressed in HEK293 cells after 4 hrs by scintillation counting analysis [AID724038, Type: Literature]Neuronal acetylcholine receptor subunit alpha-4 [gi:8469182]
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6
[SID104234160]
Ki 0.03311Displacement of [3H]epibatidine from rat recombinant alpha4beta2 nAChR expressed in HEK293 cells after 4 hrs by scintillation counting analysis [AID724038, Type: Literature]Neuronal acetylcholine receptor subunit beta-2 [gi:6226548]
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7
[SID104234160]
Ki 0.0377Displacement of [3H]epibatidine from rat alpha4beta2 nAChR expressed in HEK292 cells after 3 hrs [AID536863, Type: Literature]Neuronal acetylcholine receptor subunit alpha-4 [gi:8469182]
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8
[SID104234160]
Ki 0.0377Displacement of [3H]epibatidine from rat alpha4beta2 nAChR expressed in HEK292 cells after 3 hrs [AID536863, Type: Literature]Neuronal acetylcholine receptor subunit beta-2 [gi:6226548]
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9
[SID104234160]
Ki 0.039Displacement of [3H]cystisine from nicotinic alpha-4-beta-2 receptor in rat brain [AID320061, Type: Literature]Neuronal acetylcholine receptor subunit beta-2 [gi:6226548]
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10
[SID104234160]
Ki 0.039Displacement of [3H]cystisine from nicotinic alpha-4-beta-2 receptor in rat brain [AID320061, Type: Literature]Neuronal acetylcholine receptor subunit alpha-4 [gi:8469182]
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11
[SID104234160]
Ki 0.041Binding affinity towards rat Nicotinic acetylcholine receptor alpha3-beta2 expressed in HEK293 cells using [3H]EB as radioligand [AID146006, Type: Literature]Neuronal acetylcholine receptor subunit alpha-3 [gi:113061]
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12
[SID104234160]
Ki 0.041Binding affinity towards rat Nicotinic acetylcholine receptor alpha3-beta2 expressed in HEK293 cells using [3H]EB as radioligand [AID146006, Type: Literature]Neuronal acetylcholine receptor subunit beta-2 [gi:6226548]
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13
[SID104234160]
Ki 0.043Binding affinity towards rat forebrain nicotinic acetylcholine receptor using [3H]EB as radioligand [AID145685, Type: Literature]
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14
[SID104234160]
Ki 0.045Binding affinity towards rat Nicotinic acetylcholine receptor alpha4-beta2 expressed in HEK293 cells using [3H]EB as radioligand [AID146486, Type: Literature]Neuronal acetylcholine receptor subunit beta-2 [gi:6226548]
View
15
[SID104234160]
Ki 0.045Binding affinity towards rat Nicotinic acetylcholine receptor alpha4-beta2 expressed in HEK293 cells using [3H]EB as radioligand [AID146486, Type: Literature]Neuronal acetylcholine receptor subunit alpha-4 [gi:8469182]
View
16
[SID104234160]
Ki 0.05754Displacement of [3H]epibatidine from rat recombinant alpha4beta4 nAChR expressed in HEK293 cells after 4 hrs by scintillation counting analysis [AID724035, Type: Literature]Neuronal acetylcholine receptor subunit alpha-4 [gi:8469182]
View
17
[SID104234160]
Ki 0.05754Displacement of [3H]epibatidine from rat recombinant alpha4beta4 nAChR expressed in HEK293 cells after 4 hrs by scintillation counting analysis [AID724035, Type: Literature]Neuronal acetylcholine receptor subunit beta-4 [gi:113111]
View
18
[SID104234160]
Ki 0.083Binding affinity towards rat Nicotinic acetylcholine receptor alpha4-beta4 expressed in HEK293 cells using [3H]EB as radioligand [AID146772, Type: Literature]Neuronal acetylcholine receptor subunit beta-4 [gi:113111]
View
19
[SID104234160]
Ki 0.083Binding affinity towards rat Nicotinic acetylcholine receptor alpha4-beta4 expressed in HEK293 cells using [3H]EB as radioligand [AID146772, Type: Literature]Neuronal acetylcholine receptor subunit alpha-4 [gi:8469182]
View
20
[SID104234160]
Ki 0.085Displacement of [3H]oxotremorine from muscarinic receptor in rat brain [AID320063, Type: Literature]
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