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Adenosine Diphosphate (CID 6022) - Compound BioActivity Data
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Filters: All Data » EC50      
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BioActivity Outcomes:
Active(11)
 
 
Unspecified(9)
 
 
Top Targets:
HSP90(4)
 
 
 
HprK C(1)
 
 
BioAssay Types:
Literature(20)
 
 
 
BioActivity Types:
EC50(20)
 
 
 
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Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 19    Data Row: 20   Total Pages: 1   
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#SubstanceActivityBioAssayTargetLinks
OutcomeTypeValue [μM]
1
[SID103176960]
EC50 0.014Agonist activity at G-protein coupled P2Y1 receptor expressed in human 1321N1 cells assessed as increase in calcium by Fura2 assay [AID462811, Type: Literature]
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2
[SID103176960]
EC50 0.024Agonist activity at human GFP-tagged P2Y1R transfected in human 1321N1 cells assessed as induction of intracellular calcium mobilization by fluorescence assay [AID751213, Type: Literature]P2Y purinoceptor 1 [gi:1352692]
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3
[SID103176960]
EC50 0.069Antagonist activity against phospholipase C coupled rat P2Y purinoceptor 12 (P2Y12) [AID150495, Type: Literature]
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4
[SID103176960]
EC50 0.1Agonist activity at turkey P2Y1 receptor expressed in human 1321N1 cells assessed as increase in intracellular calcium concentration by dual-excitation spectrofluorimetric analysis [AID373705, Type: Literature]P2Y purinoceptor 1 [gi:1352693]
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5
[SID103176960]
EC50 1.7Agonist activity at human GFP-tagged P2Y11R transfected in human 1321N1 cells assessed as induction of intracellular calcium mobilization by fluorescence assay [AID751212, Type: Literature]P2Y purinoceptor 11 [gi:21263830]
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6
[SID103176960]
EC50 8Evaluated for agonist activity against phospholipase C coupled P2Y purinoceptor 1 (P2Y1) of turkey erythrocytes [AID150470, Type: Literature]P2Y purinoceptor 1 [gi:1352693]
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7
[SID103176960]
EC50 10Antagonist activity against recombinant human P2X purinoceptor 1 (P2X1 ) [AID152476, Type: Literature]
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8
[SID103176960]
EC50 11Antagonist activity against recombinant rat P2X purinoceptor 6 (P2X6 ) [AID150172, Type: Literature]
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9
[SID103176960]
EC50 18Antagonist activity against recombinant rat P2X purinoceptor 5 (P2X5) [AID150170, Type: Literature]
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10
[SID103176960]
EC50 21Inhibition of BODIPY-AG binding to dog Grp94 [AID266547, Type: Literature]Endoplasmin [gi:729425]
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11
[SID103176960]
EC50 28Antagonist activity against recombinant rat P2X purinoceptor 4 (P2X4) at 30 uM, expressed in Xenopus oocytes [AID150166, Type: Literature]
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12
[SID103176960]
EC50 65Agonist activity at human recombinant P2Y6 receptor expressed in 1321N1 cells assessed as PLC-mediated [3H]IP production [AID271163, Type: Literature]P2Y purinoceptor 6 [gi:2495018]
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13
[SID103176960]
EC50 87Inhibition of BODIPY-AG binding to human HSP90 [AID266546, Type: Literature]Heat shock protein HSP 90-alpha [gi:92090606]
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14
[SID103176960]
EC50 87Inhibition of BODIPY-AG binding to human HSP90 [AID266546, Type: Literature]Heat shock protein HSP 90-beta [gi:17865718]
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15
[SID103176960]
EC50 100The compound was evaluated for antagonist activity against recombinant human receptor P2X purinoceptor 2 (P2X2 ) [AID152489, Type: Literature]
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16
[SID103176960]
EC50 100Antagonist activity against recombinant human P2X purinoceptor 3 (P2X3 ) [AID150151, Type: Literature]
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17
[SID103176960]
EC50 100Evaluated for agonist activity against phospholipase C coupled recombinant human P2Y purinoceptor 2 (P2Y2) [AID150321, Type: Literature]
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18
[SID103176960]
EC50 120Displacement of cy3B-GM from Hsp90alpha [AID270492, Type: Literature]Heat shock protein HSP 90-alpha [gi:92090606]
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19
[SID103176960]
EC50 4300Inhibition of histidine containing protein in kinase assay [AID90064, Type: Literature]HPr kinase/phosphorylase [gi:3122218]
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20
[SID103176960]
EC50 7400Effective concentration for inhibition of Corticotropin-releasing hormone (CRH) in kinase assay [AID54140, Type: Literature]
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