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apelin receptor [Homo sapiens] [gi:4885057] - Target BioActivity Data
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BioActivity Outcomes:
Probe(1)
 
 
Active(2761)
 
 
BioAssay Types:
Screening(2071)
 
 
Confirmatory(689)
 
 
Summary(2)
 
 
 
BioActivity Types:
IC50(640)
 
 
EC50(49)
 
 
Substance Types:
Chemical(2762)
 
 
 
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Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 20    Data Row: 2762   Total Pages: 56   Display: Page     
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#StructureSubstanceCompoundActivityBioAssayLinks
OutcomeTypeValue [μM]
1
[SID99361200]
[CID46905036]
Summary assay for small molecule agonists of the APJ receptor [AID2580, Type: summary]
View
2
[SID16953942]
[CID2055076]
IC50_Mean 0.694Dose Response confirmation of uHTS hits from a small molecule antagonists of the APJ receptor via a luminescent beta-arrestin assay [AID2784, Type: confirmatory]
View
3
[SID99213055]
[CID788619]
IC50_Mean 0.886SAR analysis of small molecule antagonists of the APJ receptor via a luminescent beta-arrestin assay [AID463109, Type: confirmatory]
View
4
[SID14729228]
[CID379337]
IC50_Mean 1.05Dose Response confirmation of uHTS hits from a small molecule antagonists of the APJ receptor via a luminescent beta-arrestin assay [AID2784, Type: confirmatory]
View
5
[SID49646648]
[CID917183]
IC50_Mean 1.08Dose Response confirmation of uHTS hits from a small molecule antagonists of the APJ receptor via a luminescent beta-arrestin assay [AID2784, Type: confirmatory]
View
6
[SID24812198]
[CID1511959]
IC50_Mean 1.27Dose Response confirmation of uHTS hits from a small molecule antagonists of the APJ receptor via a luminescent beta-arrestin assay [AID2784, Type: confirmatory]
View
7
[SID99213121]
[CID2345056]
IC50_Mean 1.42SAR analysis of small molecule antagonists of the APJ receptor via a luminescent beta-arrestin assay - Set 2 [AID488803, Type: confirmatory]
View
8
[SID99213049]
[CID326793]
IC50_Mean 1.46SAR analysis of small molecule antagonists of the APJ receptor via a luminescent beta-arrestin assay [AID463109, Type: confirmatory]
View
9
[SID26726443]
[CID2812498]
IC50_Mean 1.49Dose Response confirmation of uHTS hits from a small molecule antagonists of the APJ receptor via a luminescent beta-arrestin assay [AID2784, Type: confirmatory]
View
10
[SID49643505]
[CID788619]
IC50_Mean 1.59Dose Response confirmation of uHTS hits from a small molecule antagonists of the APJ receptor via a luminescent beta-arrestin assay [AID2784, Type: confirmatory]
View
11
[SID99213119]
[CID2360979]
IC50_Mean 1.7SAR analysis of small molecule antagonists of the APJ receptor via a luminescent beta-arrestin assay - Set 2 [AID488803, Type: confirmatory]
View
12
[SID99213130]
[CID12005992]
IC50_Mean 1.75SAR analysis of small molecule antagonists of the APJ receptor via a luminescent beta-arrestin assay - Set 2 [AID488803, Type: confirmatory]
View
13
[SID103061721]
[CID7217941]
IC50_Mean 1.75SAR analysis of small molecule antagonists of the APJ receptor via a luminescent beta-arrestin assay - Set 4 [AID492986, Type: confirmatory]
View
14
[SID7975750]
[CID2767330]
IC50_Mean 1.82Dose Response confirmation of uHTS hits from a small molecule antagonists of the APJ receptor via a luminescent beta-arrestin assay [AID2784, Type: confirmatory]
View
15
[SID14735144]
[CID5407397]
IC50_Mean 1.882Dose Response confirmation of uHTS hits from a small molecule antagonists of the APJ receptor via a luminescent beta-arrestin assay [AID2784, Type: confirmatory]
View
16
[SID47195243]
[CID5416363]
IC50_Mean 1.9Dose Response confirmation of uHTS hits from a small molecule antagonists of the APJ receptor via a luminescent beta-arrestin assay [AID2784, Type: confirmatory]
View
17
[SID110167709]
[CID50898261]
EC50_Mean 1.94SAR analysis of a small molecule agonists of the APJ receptor via a luminescent beta-arrestin assay - Set 5 [AID504524, Type: confirmatory]
View
18
[SID110167726]
[CID50898257]
EC50_Mean 1.96SAR analysis of a small molecule agonists of the APJ receptor via a luminescent beta-arrestin assay - Set 5 [AID504524, Type: confirmatory]
View
19
[SID17409048]
[CID788410]
IC50_Mean 2.01Dose Response confirmation of uHTS hits from a small molecule antagonists of the APJ receptor via a luminescent beta-arrestin assay [AID2784, Type: confirmatory]
View
20
[SID49673869]
[CID2360979]
IC50_Mean 2.048Dose Response confirmation of uHTS hits from a small molecule antagonists of the APJ receptor via a luminescent beta-arrestin assay [AID2784, Type: confirmatory]
View
21
[SID24804410]
[CID800048]
IC50_Mean 2.06Dose Response confirmation of uHTS hits from a small molecule antagonists of the APJ receptor via a luminescent beta-arrestin assay [AID2784, Type: confirmatory]
View
22
[SID47197979]
[CID877472]
IC50_Mean 2.12Dose Response confirmation of uHTS hits from a small molecule antagonists of the APJ receptor via a luminescent beta-arrestin assay [AID2784, Type: confirmatory]
View
23
[SID85199439]
[CID2539399]
IC50_Mean 2.14Dose Response confirmation of uHTS hits from a small molecule antagonists of the APJ receptor via a luminescent beta-arrestin assay [AID2784, Type: confirmatory]
View
24
[SID47201524]
[CID9590741]
IC50_Mean 2.15Dose Response confirmation of uHTS hits from a small molecule antagonists of the APJ receptor via a luminescent beta-arrestin assay [AID2784, Type: confirmatory]
View
25
[SID99213078]
[CID7217941]
IC50_Mean 2.16SAR analysis of small molecule antagonists of the APJ receptor via a luminescent beta-arrestin assay - Set 2 [AID488803, Type: confirmatory]
View
26
[SID99213025]
[CID804442]
IC50_Mean 2.26SAR analysis of small molecule antagonists of the APJ receptor via a luminescent beta-arrestin assay [AID463109, Type: confirmatory]
View
27
[SID49679699]
[CID689509]
IC50_Mean 2.26Dose Response confirmation of uHTS hits from a small molecule antagonists of the APJ receptor via a luminescent beta-arrestin assay [AID2784, Type: confirmatory]
View
28
[SID49667626]
[CID5720743]
IC50_Mean 2.28Dose Response confirmation of uHTS hits from a small molecule antagonists of the APJ receptor via a luminescent beta-arrestin assay [AID2784, Type: confirmatory]
View
29
[SID99213046]
[CID618081]
IC50_Mean 2.3SAR analysis of small molecule antagonists of the APJ receptor via a luminescent beta-arrestin assay [AID463109, Type: confirmatory]
View
30
[SID99213052]
[CID788618]
IC50_Mean 2.31SAR analysis of small molecule antagonists of the APJ receptor via a luminescent beta-arrestin assay [AID463109, Type: confirmatory]
View
31
[SID24804310]
[CID2905495]
IC50_Mean 2.46Dose Response confirmation of uHTS hits from a small molecule antagonists of the APJ receptor via a luminescent beta-arrestin assay [AID2784, Type: confirmatory]
View
32
[SID99361256]
[CID2906074]
EC50_Mean 2.5SAR analysis of a small molecule agonists of the APJ receptor via a luminescent beta-arrestin assay [AID488811, Type: confirmatory]
View
33
[SID99361258]
[CID2906244]
EC50_Mean 2.52SAR analysis of a small molecule agonists of the APJ receptor via a luminescent beta-arrestin assay [AID488811, Type: confirmatory]
View
34
[SID99213117]
[CID4230722]
IC50_Mean 2.53SAR analysis of small molecule antagonists of the APJ receptor via a luminescent beta-arrestin assay - Set 2 [AID488803, Type: confirmatory]
View
35
[SID26660282]
[CID9653239]
IC50_Mean 2.53Dose Response confirmation of uHTS hits from a small molecule antagonists of the APJ receptor via a luminescent beta-arrestin assay [AID2784, Type: confirmatory]
View
36
[SID99361257]
[CID2221149]
EC50_Mean 2.56SAR analysis of a small molecule agonists of the APJ receptor via a luminescent beta-arrestin assay [AID488811, Type: confirmatory]
View
37
[SID104222787]
[CID49852493]
EC50_Mean 2.61SAR analysis of a small molecule agonists of the APJ receptor via a luminescent beta-arrestin assay - Set 5 [AID504524, Type: confirmatory]
View
38
[SID99213043]
[CID8480343]
IC50_Mean 2.62SAR analysis of small molecule antagonists of the APJ receptor via a luminescent beta-arrestin assay [AID463109, Type: confirmatory]
View
39
[SID49721505]
[CID16012896]
IC50_Mean 2.63Dose Response confirmation of uHTS hits from a small molecule antagonists of the APJ receptor via a luminescent beta-arrestin assay [AID2784, Type: confirmatory]
View
40
[SID56422197]
[CID3117]
IC50_Mean 2.63Dose Response confirmation of uHTS hits from a small molecule antagonists of the APJ receptor via a luminescent beta-arrestin assay [AID2784, Type: confirmatory]
View
41
[SID49817228]
[CID1593681]
IC50_Mean 2.65Dose Response confirmation of uHTS hits from a small molecule antagonists of the APJ receptor via a luminescent beta-arrestin assay [AID2784, Type: confirmatory]
View
42
[SID24783706]
[CID16188229]
IC50_Mean 2.75Dose Response confirmation of uHTS hits from a small molecule antagonists of the APJ receptor via a luminescent beta-arrestin assay [AID2784, Type: confirmatory]
View
43
[SID99213040]
[CID2564786]
IC50_Mean 2.81SAR analysis of small molecule antagonists of the APJ receptor via a luminescent beta-arrestin assay [AID463109, Type: confirmatory]
View
44
[SID26724400]
[CID9660957]
IC50_Mean 2.81Dose Response confirmation of uHTS hits from a small molecule antagonists of the APJ receptor via a luminescent beta-arrestin assay [AID2784, Type: confirmatory]
View
45
[SID26725274]
[CID330973]
IC50_Mean 2.85Dose Response confirmation of uHTS hits from a small molecule antagonists of the APJ receptor via a luminescent beta-arrestin assay [AID2784, Type: confirmatory]
View
46
[SID99213017]
[CID2796987]
IC50_Mean 2.89SAR analysis of small molecule antagonists of the APJ receptor via a luminescent beta-arrestin assay [AID463109, Type: confirmatory]
View
47
[SID99213039]
[CID2539399]
IC50_Mean 2.9SAR analysis of small molecule antagonists of the APJ receptor via a luminescent beta-arrestin assay [AID463109, Type: confirmatory]
View
48
[SID99361252]
[CID2217688]
EC50_Mean 2.9SAR analysis of a small molecule agonists of the APJ receptor via a luminescent beta-arrestin assay [AID488811, Type: confirmatory]
View
49
[SID99213016]
[CID583493]
IC50_Mean 2.92SAR analysis of small molecule antagonists of the APJ receptor via a luminescent beta-arrestin assay [AID463109, Type: confirmatory]
View
50
[SID24813820]
[CID5295671]
IC50_Mean 2.936Dose Response confirmation of uHTS hits from a small molecule antagonists of the APJ receptor via a luminescent beta-arrestin assay [AID2784, Type: confirmatory]
View