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apelin receptor [Homo sapiens] [gi:4885057] - Target BioActivity Data
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BioActivity Outcomes:
Probe(1)
 
 
Active(2761)
 
 
BioAssay Types:
Screening(2071)
 
 
Confirmatory(689)
 
 
Summary(2)
 
 
 
BioActivity Types:
IC50(640)
 
 
EC50(49)
 
 
Substance Types:
Chemical(2762)
 
 
 
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Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 20    Data Row: 2762   Total Pages: 139   Display: Page     
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#StructureSubstanceCompoundActivityBioAssayLinks
OutcomeTypeValue [μM]
1
[SID99361200]
[CID46905036]
Summary assay for small molecule agonists of the APJ receptor [AID2580, Type: summary]
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2
[SID16953942]
[CID2055076]
IC50_Mean 0.694Dose Response confirmation of uHTS hits from a small molecule antagonists of the APJ receptor via a luminescent beta-arrestin assay [AID2784, Type: confirmatory]
View
3
[SID99213055]
[CID788619]
IC50_Mean 0.886SAR analysis of small molecule antagonists of the APJ receptor via a luminescent beta-arrestin assay [AID463109, Type: confirmatory]
View
4
[SID14729228]
[CID379337]
IC50_Mean 1.05Dose Response confirmation of uHTS hits from a small molecule antagonists of the APJ receptor via a luminescent beta-arrestin assay [AID2784, Type: confirmatory]
View
5
[SID49646648]
[CID917183]
IC50_Mean 1.08Dose Response confirmation of uHTS hits from a small molecule antagonists of the APJ receptor via a luminescent beta-arrestin assay [AID2784, Type: confirmatory]
View
6
[SID24812198]
[CID1511959]
IC50_Mean 1.27Dose Response confirmation of uHTS hits from a small molecule antagonists of the APJ receptor via a luminescent beta-arrestin assay [AID2784, Type: confirmatory]
View
7
[SID99213121]
[CID2345056]
IC50_Mean 1.42SAR analysis of small molecule antagonists of the APJ receptor via a luminescent beta-arrestin assay - Set 2 [AID488803, Type: confirmatory]
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8
[SID99213049]
[CID326793]
IC50_Mean 1.46SAR analysis of small molecule antagonists of the APJ receptor via a luminescent beta-arrestin assay [AID463109, Type: confirmatory]
View
9
[SID26726443]
[CID2812498]
IC50_Mean 1.49Dose Response confirmation of uHTS hits from a small molecule antagonists of the APJ receptor via a luminescent beta-arrestin assay [AID2784, Type: confirmatory]
View
10
[SID49643505]
[CID788619]
IC50_Mean 1.59Dose Response confirmation of uHTS hits from a small molecule antagonists of the APJ receptor via a luminescent beta-arrestin assay [AID2784, Type: confirmatory]
View
11
[SID99213119]
[CID2360979]
IC50_Mean 1.7SAR analysis of small molecule antagonists of the APJ receptor via a luminescent beta-arrestin assay - Set 2 [AID488803, Type: confirmatory]
View
12
[SID99213130]
[CID12005992]
IC50_Mean 1.75SAR analysis of small molecule antagonists of the APJ receptor via a luminescent beta-arrestin assay - Set 2 [AID488803, Type: confirmatory]
View
13
[SID103061721]
[CID7217941]
IC50_Mean 1.75SAR analysis of small molecule antagonists of the APJ receptor via a luminescent beta-arrestin assay - Set 4 [AID492986, Type: confirmatory]
View
14
[SID7975750]
[CID2767330]
IC50_Mean 1.82Dose Response confirmation of uHTS hits from a small molecule antagonists of the APJ receptor via a luminescent beta-arrestin assay [AID2784, Type: confirmatory]
View
15
[SID14735144]
[CID5407397]
IC50_Mean 1.882Dose Response confirmation of uHTS hits from a small molecule antagonists of the APJ receptor via a luminescent beta-arrestin assay [AID2784, Type: confirmatory]
View
16
[SID47195243]
[CID5416363]
IC50_Mean 1.9Dose Response confirmation of uHTS hits from a small molecule antagonists of the APJ receptor via a luminescent beta-arrestin assay [AID2784, Type: confirmatory]
View
17
[SID110167709]
[CID50898261]
EC50_Mean 1.94SAR analysis of a small molecule agonists of the APJ receptor via a luminescent beta-arrestin assay - Set 5 [AID504524, Type: confirmatory]
View
18
[SID110167726]
[CID50898257]
EC50_Mean 1.96SAR analysis of a small molecule agonists of the APJ receptor via a luminescent beta-arrestin assay - Set 5 [AID504524, Type: confirmatory]
View
19
[SID17409048]
[CID788410]
IC50_Mean 2.01Dose Response confirmation of uHTS hits from a small molecule antagonists of the APJ receptor via a luminescent beta-arrestin assay [AID2784, Type: confirmatory]
View
20
[SID49673869]
[CID2360979]
IC50_Mean 2.048Dose Response confirmation of uHTS hits from a small molecule antagonists of the APJ receptor via a luminescent beta-arrestin assay [AID2784, Type: confirmatory]
View