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endothelial PAS domain-containing protein 1 [.. [gi:40254439] - Target BioActivity Data
Also known as: endothelial PAS domain-containing protein 1 [Homo sapiens].
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BioActivity Outcomes:
Active(3931)
 
 
BioAssay Types:
Screening(3608)
 
 
Confirmatory(323)
 
 
BioActivity Types:
IC50(323)
 
 
Substance Types:
Chemical(3931)
 
 
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Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 4    Data Row: 3931   Total Pages: 79   Display: Page     
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#StructureSubstanceCompoundActivityBioAssayLinks
OutcomeTypeValue [μM]
1
[SID4254515]
[CID972733]
IC50_HIF-2a_PANC_Mean 0.19Dose response confirmation of uHTS identification of HIF-2a Inhibitors in screening - selectivity counterscreen assays [AID651581_7, Type: confirmatory]
View
2
[SID103061877]
[CID666941]
IC50_Mean_HIF2a (PANC cells) 0.19SAR Analysis small molecule inhibitors of HIF-1a in a panel assay [AID652011, Type: confirmatory]
View
3
[SID103061905]
[CID1994282]
IC50_Mean_HIF2a (PANC cells) 0.19SAR Analysis small molecule inhibitors of HIF-1a in a panel assay [AID652011, Type: confirmatory]
View
4
[SID103061912]
[CID1943900]
IC50_Mean_HIF2a (PANC cells) 0.19SAR Analysis small molecule inhibitors of HIF-1a in a panel assay [AID652011, Type: confirmatory]
View
5
[SID103061963]
[CID2037423]
IC50_Mean_HIF2a (PANC cells) 0.19SAR Analysis small molecule inhibitors of HIF-1a in a panel assay [AID652011, Type: confirmatory]
View
6
[SID103061971]
[CID3159504]
IC50_Mean_HIF2a (PANC cells) 0.19SAR Analysis small molecule inhibitors of HIF-1a in a panel assay [AID652011, Type: confirmatory]
View
7
[SID110067542]
[CID50898039]
IC50_Mean_HIF2a (PANC cells) 0.19SAR Analysis small molecule inhibitors of HIF-1a in a panel assay [AID652011, Type: confirmatory]
View
8
[SID103061973]
[CID666941]
IC50_Mean_HIF2a (PANC cells) 0.19SAR Analysis small molecule inhibitors of HIF-1a in a panel assay [AID652011, Type: confirmatory]
View
9
[SID110067516]
[CID50898046]
IC50_Mean_HIF2a (PANC cells) 0.19SAR Analysis small molecule inhibitors of HIF-1a in a panel assay [AID652011, Type: confirmatory]
View
10
[SID110067538]
[CID50898044]
IC50_Mean_HIF2a (PANC cells) 0.19SAR Analysis small molecule inhibitors of HIF-1a in a panel assay [AID652011, Type: confirmatory]
View
11
[SID49675252]
[CID854968]
IC50_HIF-2a_PANC_Mean 0.247Dose response confirmation of uHTS identification of HIF-2a Inhibitors in screening - selectivity counterscreen assays [AID651581_7, Type: confirmatory]
View
12
[SID22411729]
[CID15945494]
IC50_HIF-2a_PANC_Mean 0.25Dose response confirmation of uHTS identification of HIF-2a Inhibitors in screening - selectivity counterscreen assays [AID651581_7, Type: confirmatory]
View
13
[SID49665726]
[CID2767825]
IC50_1_HIF-1a 0.274Dose response confirmation of uHTS identification of HIF-2a Inhibitors in screening - selectivity counterscreen assays [AID651581, Type: confirmatory]
View
14
[SID865680]
[CID666941]
IC50_HIF-2a_PANC_Mean 0.3Dose response confirmation of uHTS identification of HIF-2a Inhibitors in screening - selectivity counterscreen assays [AID651581_7, Type: confirmatory]
View
15
[SID17510599]
[CID9657888]
IC50_HIF-2a_PANC_Mean 0.3Dose response confirmation of uHTS identification of HIF-2a Inhibitors in screening - selectivity counterscreen assays [AID651581_7, Type: confirmatory]
View
16
[SID49725274]
[CID1991339]
IC50_HIF-2a_PANC_Mean 0.3Dose response confirmation of uHTS identification of HIF-2a Inhibitors in screening - selectivity counterscreen assays [AID651581_7, Type: confirmatory]
View
17
[SID26660824]
[CID6902747]
IC50_HIF-2a_PANC_Mean 0.378Dose response confirmation of uHTS identification of HIF-2a Inhibitors in screening - selectivity counterscreen assays [AID651581_7, Type: confirmatory]
View
18
[SID24824544]
[CID2767852]
IC50_1_HIF-1a 0.397Dose response confirmation of uHTS identification of HIF-2a Inhibitors in screening - selectivity counterscreen assays [AID651581, Type: confirmatory]
View
19
[SID22414953]
[CID4592654]
IC50_HIF-2a_PANC_Mean 0.417Dose response confirmation of uHTS identification of HIF-2a Inhibitors in screening - selectivity counterscreen assays [AID651581_7, Type: confirmatory]
View
20
[SID4249581]
[CID3243514]
IC50_HIF-2a_PANC_Mean 0.447Dose response confirmation of uHTS identification of HIF-2a Inhibitors in screening - selectivity counterscreen assays [AID651581_7, Type: confirmatory]
View
21
[SID22411729]
[CID15945494]
IC50_1_HIF-1a 0.486Dose response confirmation of uHTS identification of HIF-2a Inhibitors in screening - selectivity counterscreen assays [AID651581, Type: confirmatory]
View
22
[SID858142]
[CID659499]
IC50_HIF-2a_PANC_Mean 0.506Dose response confirmation of uHTS identification of HIF-2a Inhibitors in screening - selectivity counterscreen assays [AID651581_7, Type: confirmatory]
View
23
[SID103061910]
[CID1994219]
IC50_Mean_HIF2a (PANC cells) 0.573SAR Analysis small molecule inhibitors of HIF-1a in a panel assay [AID652011, Type: confirmatory]
View
24
[SID85198232]
[CID24896921]
IC50_HIF-2a_PANC_Mean 0.7Dose response confirmation of uHTS identification of HIF-2a Inhibitors in screening - selectivity counterscreen assays [AID651581_7, Type: confirmatory]
View
25
[SID24792303]
[CID907197]
IC50_HIF-2a_PANC_Mean 0.708Dose response confirmation of uHTS identification of HIF-2a Inhibitors in screening - selectivity counterscreen assays [AID651581_7, Type: confirmatory]
View
26
[SID17416347]
[CID5710160]
IC50_HIF-2a_PANC_Mean 0.711Dose response confirmation of uHTS identification of HIF-2a Inhibitors in screening - selectivity counterscreen assays [AID651581_7, Type: confirmatory]
View
27
[SID14735515]
[CID9550743]
IC50_HIF-2a_PANC_Mean 0.787Dose response confirmation of uHTS identification of HIF-2a Inhibitors in screening - selectivity counterscreen assays [AID651581_7, Type: confirmatory]
View
28
[SID14722386]
[CID774798]
IC50_HIF-2a_PANC_Mean 0.796Dose response confirmation of uHTS identification of HIF-2a Inhibitors in screening - selectivity counterscreen assays [AID651581_7, Type: confirmatory]
View
29
[SID49829119]
[CID6351343]
IC50_1_HIF-1a 0.824Dose response confirmation of uHTS identification of HIF-2a Inhibitors in screening - selectivity counterscreen assays [AID651581, Type: confirmatory]
View
30
[SID24797240]
[CID900837]
IC50_HIF-2a_PANC_Mean 0.92Dose response confirmation of uHTS identification of HIF-2a Inhibitors in screening - selectivity counterscreen assays [AID651581_7, Type: confirmatory]
View
31
[SID49735234]
[CID23605826]
IC50_HIF-2a_PANC_Mean 0.975Dose response confirmation of uHTS identification of HIF-2a Inhibitors in screening - selectivity counterscreen assays [AID651581_7, Type: confirmatory]
View
32
[SID17505190]
[CID9633427]
IC50_HIF-2a_PANC_Mean 1Dose response confirmation of uHTS identification of HIF-2a Inhibitors in screening - selectivity counterscreen assays [AID651581_7, Type: confirmatory]
View
33
[SID49829119]
[CID6351343]
IC50_HIF-2a_PANC_Mean 1.12Dose response confirmation of uHTS identification of HIF-2a Inhibitors in screening - selectivity counterscreen assays [AID651581_7, Type: confirmatory]
View
34
[SID24824544]
[CID2767852]
IC50_HIF-2a_PANC_Mean 1.14Dose response confirmation of uHTS identification of HIF-2a Inhibitors in screening - selectivity counterscreen assays [AID651581_7, Type: confirmatory]
View
35
[SID49647507]
[CID1757603]
IC50_1_HIF-1a 1.228Dose response confirmation of uHTS identification of HIF-2a Inhibitors in screening - selectivity counterscreen assays [AID651581, Type: confirmatory]
View
36
[SID49735234]
[CID23605826]
IC50_1_HIF-1a 1.263Dose response confirmation of uHTS identification of HIF-2a Inhibitors in screening - selectivity counterscreen assays [AID651581, Type: confirmatory]
View
37
[SID22406405]
[CID2426240]
IC50_HIF-2a_PANC_Mean 1.29Dose response confirmation of uHTS identification of HIF-2a Inhibitors in screening - selectivity counterscreen assays [AID651581_7, Type: confirmatory]
View
38
[SID47202097]
[CID2193280]
IC50_1_HIF-1a 1.48Dose response confirmation of uHTS identification of HIF-2a Inhibitors in screening - selectivity counterscreen assays [AID651581, Type: confirmatory]
View
39
[SID103163054]
[CID1089417]
IC50_HIF-2a_PANC_Mean 1.51Dose response confirmation of uHTS identification of HIF-2a Inhibitors in screening - selectivity counterscreen assays [AID651581_7, Type: confirmatory]
View
40
[SID14735522]
[CID9550750]
IC50_HIF-2a_PANC_Mean 1.59Dose response confirmation of uHTS identification of HIF-2a Inhibitors in screening - selectivity counterscreen assays [AID651581_7, Type: confirmatory]
View
41
[SID49820116]
[CID6351467]
IC50_HIF-2a_PANC_Mean 1.72Dose response confirmation of uHTS identification of HIF-2a Inhibitors in screening - selectivity counterscreen assays [AID651581_7, Type: confirmatory]
View
42
[SID103073926]
[CID49789464]
IC50_HIF-2a_PANC_Mean 1.85Dose response confirmation of uHTS identification of HIF-2a Inhibitors in screening - selectivity counterscreen assays [AID651581_7, Type: confirmatory]
View
43
[SID24822404]
[CID1157635]
IC50_HIF-2a_PANC_Mean 1.93Dose response confirmation of uHTS identification of HIF-2a Inhibitors in screening - selectivity counterscreen assays [AID651581_7, Type: confirmatory]
View
44
[SID22401701]
[CID2420694]
IC50_HIF-2a_PANC_Mean 2.01Dose response confirmation of uHTS identification of HIF-2a Inhibitors in screening - selectivity counterscreen assays [AID651581_7, Type: confirmatory]
View
45
[SID4252437]
[CID3245990]
IC50_HIF-2a_PANC_Mean 2.03Dose response confirmation of uHTS identification of HIF-2a Inhibitors in screening - selectivity counterscreen assays [AID651581_7, Type: confirmatory]
View
46
[SID14735523]
[CID9550751]
IC50_HIF-2a_PANC_Mean 2.16Dose response confirmation of uHTS identification of HIF-2a Inhibitors in screening - selectivity counterscreen assays [AID651581_7, Type: confirmatory]
View
47
[SID103159290]
[CID721101]
IC50_HIF-2a_PANC_Mean 2.26Dose response confirmation of uHTS identification of HIF-2a Inhibitors in screening - selectivity counterscreen assays [AID651581_7, Type: confirmatory]
View
48
[SID17412124]
[CID707664]
IC50_1_HIF-1a 2.297Dose response confirmation of uHTS identification of HIF-2a Inhibitors in screening - selectivity counterscreen assays [AID651581, Type: confirmatory]
View
49
[SID103159036]
[CID2426236]
IC50_HIF-2a_PANC_Mean 2.3Dose response confirmation of uHTS identification of HIF-2a Inhibitors in screening - selectivity counterscreen assays [AID651581_7, Type: confirmatory]
View
50
[SID49679251]
[CID1490583]
IC50_HIF-2a_PANC_Mean 2.37Dose response confirmation of uHTS identification of HIF-2a Inhibitors in screening - selectivity counterscreen assays [AID651581_7, Type: confirmatory]
View