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Peroxisome proliferator-activated receptor al.. [gi:3041727] - Target BioActivity Data
Also known as: Peroxisome proliferator-activated receptor alpha; PPAR-alpha; Nuclear receptor subfamily 1 group C member 1.
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BioActivity Outcomes:
Active(2337)
 
 
BioAssay Types:
Literature(2289)
 
 
Confirmatory(43)
 
 
BioActivity Types:
EC50(1618)
 
 
IC50(547)
 
 
Ki(51)
 
 
Potency(33)
 
 
Kd(10)
 
 
Substance Types:
Chemical(2337)
 
 
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Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 215    Data Row: 2337   Total Pages: 117   Display: Page     
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#StructureSubstanceCompoundActivityBioAssayLinks
OutcomeTypeValue [μM]
1
[SID134436215]
[CID56659348]
EC50 5e-08Transactivation of human PPARalpha expressed in human HepG2 cells co-transfected with PPRE3-TK-Luc by luciferase reporter gene assay [AID610309, Type: Literature]
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2
[SID134459372]
[CID56679849]
EC50 6e-08Transactivation of human PPARalpha expressed in human HepG2 cells co-transfected with PPRE3-TK-Luc by luciferase reporter gene assay [AID610309, Type: Literature]
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3
[SID134447814]
[CID56669690]
EC50 7e-08Transactivation of human PPARalpha expressed in human HepG2 cells co-transfected with PPRE3-TK-Luc by luciferase reporter gene assay [AID610309, Type: Literature]
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4
[SID134455510]
[CID53233135]
EC50 3.1e-07Transactivation of human PPARalpha expressed in human HepG2 cells co-transfected with PPRE3-TK-Luc by luciferase reporter gene assay [AID610309, Type: Literature]
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5
[SID103610257]
[CID44571517]
EC50 3.8e-06Agonist activity at human PPARalpha transactivation expressed in human HePG2 cells [AID371249, Type: Literature]
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6
[SID134436214]
[CID56659347]
EC50 2.6e-05Transactivation of human PPARalpha expressed in human HepG2 cells co-transfected with PPRE3-TK-Luc by luciferase reporter gene assay [AID610309, Type: Literature]
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7
[SID134447813]
[CID56669689]
EC50 0.0001Transactivation of human PPARalpha expressed in human HepG2 cells co-transfected with PPRE3-TK-Luc by luciferase reporter gene assay [AID610309, Type: Literature]
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8
[SID103559456]
[CID44446262]
EC50 0.0003Agonist activity at human PPARalpha assessed as receptor activation by cell based assay [AID313747, Type: Literature]
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9
[SID103326409]
[CID9825046]
EC50 0.000615Transcriptional activation activity on human Peroxisome proliferator activated receptor alpha expressed in CHO-K1 cells [AID156124, Type: Literature]
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10
[SID103281158]
[CID11178750]
EC50 0.001Transcriptional activation of reporter assay by human Peroxisome proliferator activated receptor alpha in CV-1 cells [AID156129, Type: Literature]
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11
[SID103187301]
[CID3392731]
Kd 0.001Binding affinity to human PPARalpha (unknown origin) by competitive TR-FRET assay [AID731521, Type: Literature]
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12
[SID103483181]
[CID44409279]
IC50 0.001Binding affinity to human PPAR alpha [AID261943, Type: Literature]
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13
[SID103483181]
[CID44409279]
EC50 0.001Transactivation by human PPAR alpha in COS1 cells [AID261946, Type: Literature]
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14
[SID103483119]
[CID44409249]
EC50 0.001Transactivation by human PPAR alpha in COS1 cells [AID261946, Type: Literature]
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15
[SID103549440]
[CID11397705]
EC50 0.001Agonist activity at human recombinant PPARalpha by GAL4 transactivation assay [AID308331, Type: Literature]
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16
[SID103549444]
[CID44440789]
EC50 0.001Agonist activity at human recombinant PPARalpha by GAL4 transactivation assay [AID308331, Type: Literature]
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17
[SID103549445]
[CID44440790]
EC50 0.001Agonist activity at human recombinant PPARalpha by GAL4 transactivation assay [AID308331, Type: Literature]
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18
[SID103549446]
[CID44440791]
EC50 0.001Agonist activity at human recombinant PPARalpha by GAL4 transactivation assay [AID308331, Type: Literature]
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19
[SID103549463]
[CID11526038]
EC50 0.001Agonist activity at human recombinant PPARalpha by GAL4 transactivation assay [AID308331, Type: Literature]
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20
[SID103610259]
[CID44571519]
EC50 0.001Agonist activity at human PPARalpha transactivation expressed in human HePG2 cells [AID371249, Type: Literature]
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