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Peroxisome proliferator-activated receptor al.. [gi:3041727] - Target BioActivity Data
Also known as: Peroxisome proliferator-activated receptor alpha; PPAR-alpha; Nuclear receptor subfamily 1 group C member 1.
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BioActivity Outcomes:
Active(2305)
 
 
BioAssay Types:
Literature(2257)
 
 
Confirmatory(33)
 
 
BioActivity Types:
EC50(1595)
 
 
IC50(548)
 
 
Ki(51)
 
 
Potency(33)
 
 
Kd(10)
 
 
Substance Types:
Chemical(2305)
 
 
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Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 211    Data Row: 2305   Total Pages: 47   Display: Page     
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#StructureSubstanceCompoundActivityBioAssayLinks
OutcomeTypeValue [μM]
1
[SID134436215]
[CID56659348]
EC50 5e-08Transactivation of human PPARalpha expressed in human HepG2 cells co-transfected with PPRE3-TK-Luc by luciferase reporter gene assay [AID610309, Type: Literature]
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2
[SID134459372]
[CID56679849]
EC50 6e-08Transactivation of human PPARalpha expressed in human HepG2 cells co-transfected with PPRE3-TK-Luc by luciferase reporter gene assay [AID610309, Type: Literature]
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3
[SID134447814]
[CID56669690]
EC50 7e-08Transactivation of human PPARalpha expressed in human HepG2 cells co-transfected with PPRE3-TK-Luc by luciferase reporter gene assay [AID610309, Type: Literature]
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4
[SID134455510]
[CID53233135]
EC50 3.1e-07Transactivation of human PPARalpha expressed in human HepG2 cells co-transfected with PPRE3-TK-Luc by luciferase reporter gene assay [AID610309, Type: Literature]
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5
[SID103610257]
[CID44571517]
EC50 3.8e-06Agonist activity at human PPARalpha transactivation expressed in human HePG2 cells [AID371249, Type: Literature]
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6
[SID134436214]
[CID56659347]
EC50 2.6e-05Transactivation of human PPARalpha expressed in human HepG2 cells co-transfected with PPRE3-TK-Luc by luciferase reporter gene assay [AID610309, Type: Literature]
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7
[SID134447813]
[CID56669689]
EC50 0.0001Transactivation of human PPARalpha expressed in human HepG2 cells co-transfected with PPRE3-TK-Luc by luciferase reporter gene assay [AID610309, Type: Literature]
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8
[SID103559456]
[CID44446262]
EC50 0.0003Agonist activity at human PPARalpha assessed as receptor activation by cell based assay [AID313747, Type: Literature]
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9
[SID103326409]
[CID9825046]
EC50 0.000615Transcriptional activation activity on human Peroxisome proliferator activated receptor alpha expressed in CHO-K1 cells [AID156124, Type: Literature]
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10
[SID103281158]
[CID11178750]
EC50 0.001Transcriptional activation of reporter assay by human Peroxisome proliferator activated receptor alpha in CV-1 cells [AID156129, Type: Literature]
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11
[SID103187301]
[CID3392731]
Kd 0.001Binding affinity to human PPARalpha (unknown origin) by competitive TR-FRET assay [AID731521, Type: Literature]
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12
[SID103483119]
[CID44409249]
EC50 0.001Transactivation by human PPAR alpha in COS1 cells [AID261946, Type: Literature]
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13
[SID103483181]
[CID44409279]
IC50 0.001Binding affinity to human PPAR alpha [AID261943, Type: Literature]
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14
[SID103483181]
[CID44409279]
EC50 0.001Transactivation by human PPAR alpha in COS1 cells [AID261946, Type: Literature]
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15
[SID103549463]
[CID11526038]
EC50 0.001Agonist activity at human recombinant PPARalpha by GAL4 transactivation assay [AID308331, Type: Literature]
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16
[SID103549440]
[CID11397705]
EC50 0.001Agonist activity at human recombinant PPARalpha by GAL4 transactivation assay [AID308331, Type: Literature]
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17
[SID103549444]
[CID44440789]
EC50 0.001Agonist activity at human recombinant PPARalpha by GAL4 transactivation assay [AID308331, Type: Literature]
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18
[SID103549445]
[CID44440790]
EC50 0.001Agonist activity at human recombinant PPARalpha by GAL4 transactivation assay [AID308331, Type: Literature]
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19
[SID103549446]
[CID44440791]
EC50 0.001Agonist activity at human recombinant PPARalpha by GAL4 transactivation assay [AID308331, Type: Literature]
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20
[SID103610259]
[CID44571519]
EC50 0.001Agonist activity at human PPARalpha transactivation expressed in human HePG2 cells [AID371249, Type: Literature]
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21
[SID103630554]
[CID25149125]
EC50 0.001Agonist activity at human PPARalpha in U2OS cells by transactivation assay [AID396052, Type: Literature]
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22
[SID103521626]
[CID25263404]
EC50 0.0013Agonist activity at human PPARalpha in HepG2 cells by PPAR-GAL4 transactivation assay [AID289934, Type: Literature]
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23
[SID134459373]
[CID56679850]
EC50 0.0019Transactivation of human PPARalpha expressed in human HepG2 cells co-transfected with PPRE3-TK-Luc by luciferase reporter gene assay [AID610309, Type: Literature]
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24
[SID103652551]
[CID44591724]
EC50 0.002Agonist activity at human PPARalpha by luciferase reporter transactivation assay [AID354042, Type: Literature]
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25
[SID103687418]
[CID44190861]
EC50 0.002Agonist activity at human PPARalpha receptor expressed in african green monkey COS1 cells co-transfected with fused yeast Gal4-DBD by transactivation assay [AID421050, Type: Literature]
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26
[SID103724537]
[CID46229871]
EC50 0.002Agonist activity at human full length PPARalpha expressed in human HepG2 cells co-transfected with PPRE3-TK-luc assessed as induction of beta-galactosidase activity by firefly luciferase assay [AID457059, Type: Literature]
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27
[SID103610258]
[CID44571518]
EC50 0.002Agonist activity at human PPARalpha transactivation expressed in human HePG2 cells [AID371249, Type: Literature]
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28
[SID103588451]
[CID11225048]
EC50 0.002Agonist activity at human PPARalpha receptor by cell based transient transfection assay [AID410081, Type: Literature]
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29
[SID103549432]
[CID44440779]
EC50 0.002Agonist activity at human recombinant PPARalpha by GAL4 transactivation assay [AID308331, Type: Literature]
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30
[SID103550097]
[CID16747684]
EC50 0.002Agonist activity at human PPARalpha by transactivation assay [AID307130, Type: Literature]
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31
[SID103549450]
[CID44440795]
EC50 0.002Agonist activity at human recombinant PPARalpha by GAL4 transactivation assay [AID308331, Type: Literature]
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32
[SID103549455]
[CID44440800]
EC50 0.002Agonist activity at human recombinant PPARalpha by GAL4 transactivation assay [AID308331, Type: Literature]
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33
[SID103483119]
[CID44409249]
IC50 0.002Binding affinity to human PPAR alpha [AID261943, Type: Literature]
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34
[SID103393729]
[CID10162008]
EC50 0.002Cotransfection activity against human Peroxisome proliferator activated receptor alpha [AID156131, Type: Literature]
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35
[SID103442382]
[CID10182946]
EC50 0.002Agonist activity against human PPARalpha in COS-1 cell Gal4 assay [AID246052, Type: Literature]
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36
[SID103453949]
[CID446642]
Ki 0.002Binding affinity for human peroxisome proliferator activated receptor alpha [AID238856, Type: Literature]
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37
[SID103453949]
[CID446642]
EC50 0.002Effective concentration against human peroxisome proliferator activated receptor alpha in Gal4 transactivation assay [AID240312, Type: Literature]
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38
[SID103460463]
[CID9981617]
EC50 0.002Effective concentration against human PPAR-alpha in Gal4 transactivation assay [AID246706, Type: Literature]
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39
[SID103460779]
[CID10367018]
EC50 0.002Effective concentration against human PPAR-alpha in Gal4 transactivation assay [AID246706, Type: Literature]
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40
[SID103460814]
[CID11248512]
EC50 0.002Effective concentration against human PPAR-alpha in Gal4 transactivation assay [AID246706, Type: Literature]
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41
[SID103460838]
[CID11386220]
EC50 0.002Effective concentration against human PPAR-alpha in Gal4 transactivation assay [AID246706, Type: Literature]
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42
[SID103472786]
[CID11620018]
EC50 0.002Functional activity at human PPAR alpha in Huh7 cells by transactivation assay [AID256777, Type: Literature]
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43
[SID103482764]
[CID44409098]
EC50 0.0021Transactivation by human PPAR alpha in COS1 cells [AID261946, Type: Literature]
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44
[SID103521625]
[CID25263403]
EC50 0.0022Agonist activity at human PPARalpha in HepG2 cells by PPAR-GAL4 transactivation assay [AID289934, Type: Literature]
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45
[SID103569797]
[CID446642]
EC50 0.0023Agonist activity at human PPARalpha [AID330491, Type: Literature]
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46
[SID103483470]
[CID44409427]
EC50 0.0025Transactivation by human PPAR alpha in COS1 cells [AID261946, Type: Literature]
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47
[SID103483476]
[CID44409429]
EC50 0.0027Transactivation by human PPAR alpha in COS1 cells [AID261946, Type: Literature]
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48
[SID103483174]
[CID44409274]
EC50 0.0029Transactivation by human PPAR alpha in COS1 cells [AID261946, Type: Literature]
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49
[SID103482824]
[CID44409126]
EC50 0.003Transactivation by human PPAR alpha in COS1 cells [AID261946, Type: Literature]
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50
[SID103482764]
[CID44409098]
IC50 0.003Binding affinity to human PPAR alpha [AID261943, Type: Literature]
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