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epidermal growth factor receptor isoform a pr.. [gi:29725609] - Target BioActivity Data
Also known as: epidermal growth factor receptor isoform a precursor [Homo sapiens].
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BioActivity Outcomes:
Probe(1)
 
 
Active(90)
 
 
BioAssay Types:
Confirmatory(81)
 
 
Summary(10)
 
 
 
BioActivity Types:
Potency(23)
 
 
IC50(10)
 
 
 
Substance Types:
Chemical(91)
 
 
 
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Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 6    Data Row: 91   Total Pages: 2   Display: Page     
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#StructureSubstanceCompoundActivityBioAssayLinks
OutcomeTypeValue [μM]
1
[SID22409543]
[CID2303746]
EGFR IC50 0.7079Quantitative High-Throughput Screen for Inhibitors of the ERK Signaling Pathway using a Homogeneous Screening Assay: Summary [AID1742, Type: summary]
View
2
[SID26757996]
[CID176870]
Potency 0.0008Assay for Inhibitors of the ERK Signaling Pathway using a Homogeneous Screening Assay: EGFR Kinase Inhibition [AID1731, Type: confirmatory]
View
3
[SID26757996]
[CID176870]
Potency 0.0009Assay for Inhibitors of the ERK Signaling Pathway using a Homogeneous Screening Assay: EGFR L858R Kinase Inhibition [AID1727, Type: confirmatory]
View
4
[SID26757996]
[CID176870]
EGFR IC50 0.001Quantitative High-Throughput Screen for Inhibitors of the ERK Signaling Pathway using a Homogeneous Screening Assay: Summary [AID1742, Type: summary]
View
5
[SID29215403]
[CID123631]
Potency 0.0032Assay for Inhibitors of the ERK Signaling Pathway using a Homogeneous Screening Assay: EGFR L858R Kinase Inhibition [AID1727, Type: confirmatory]
View
6
[SID29215403]
[CID123631]
Potency 0.0032Assay for Inhibitors of the ERK Signaling Pathway using a Homogeneous Screening Assay: EGFR Kinase Inhibition [AID1731, Type: confirmatory]
View
7
[SID29215403]
[CID123631]
EGFR IC50 0.004Quantitative High-Throughput Screen for Inhibitors of the ERK Signaling Pathway using a Homogeneous Screening Assay: Summary [AID1742, Type: summary]
View
8
[SID26755744]
[CID44259]
Potency 0.0056Assay for Inhibitors of the ERK Signaling Pathway using a Homogeneous Screening Assay: EGFR T790M Kinase Inhibition [AID1729, Type: confirmatory]
View
9
[SID26753250]
[CID16219404]
Potency 0.0089Assay for Inhibitors of the ERK Signaling Pathway using a Homogeneous Screening Assay: EGFR Kinase Inhibition [AID1731, Type: confirmatory]
View
10
[SID26753250]
[CID16219404]
EGFR IC50 0.01Quantitative High-Throughput Screen for Inhibitors of the ERK Signaling Pathway using a Homogeneous Screening Assay: Summary [AID1742, Type: summary]
View
11
[SID26755744]
[CID44259]
Potency 0.0398Assay for Inhibitors of the ERK Signaling Pathway using a Homogeneous Screening Assay: EGFR T790M/L858R Kinase Inhibition [AID1726, Type: confirmatory]
View
12
[SID22406015]
[CID5211059]
Potency 0.0447Assay for Inhibitors of the ERK Signaling Pathway using a Homogeneous Screening Assay: EGFR L858R Kinase Inhibition [AID1727, Type: confirmatory]
View
13
[SID26753250]
[CID16219404]
Potency 0.0501Assay for Inhibitors of the ERK Signaling Pathway using a Homogeneous Screening Assay: EGFR L858R Kinase Inhibition [AID1727, Type: confirmatory]
View
14
[SID22406015]
[CID5211059]
Potency 0.0708Assay for Inhibitors of the ERK Signaling Pathway using a Homogeneous Screening Assay: EGFR Kinase Inhibition [AID1731, Type: confirmatory]
View
15
[SID22406015]
[CID5211059]
EGFR IC50 0.0708Quantitative High-Throughput Screen for Inhibitors of the ERK Signaling Pathway using a Homogeneous Screening Assay: Summary [AID1742, Type: summary]
View
16
[SID50100094]
[CID156414]
0.13Kinase Inhibitor Selectivity Profiling Assay [AID1433_19, Type: confirmatory]
View
17
[SID50100094]
[CID156414]
0.17Kinase Inhibitor Selectivity Profiling Assay [AID1433_80, Type: confirmatory]
View
18
[SID50100094]
[CID156414]
0.19Kinase Inhibitor Selectivity Profiling Assay [AID1433_78, Type: confirmatory]
View
19
[SID50100094]
[CID156414]
0.19Kinase Inhibitor Selectivity Profiling Assay [AID1433_79, Type: confirmatory]
View
20
[SID50100094]
[CID156414]
0.19Kinase Inhibitor Selectivity Profiling Assay [AID1433_175, Type: confirmatory]
View
21
[SID50100094]
[CID156414]
0.22Kinase Inhibitor Selectivity Profiling Assay [AID1433_83, Type: confirmatory]
View
22
[SID50100098]
[CID6445562]
0.23Kinase Inhibitor Selectivity Profiling Assay [AID1433_82, Type: confirmatory]
View
23
[SID50100098]
[CID6445562]
0.24Kinase Inhibitor Selectivity Profiling Assay [AID1433_80, Type: confirmatory]
View
24
[SID50100094]
[CID156414]
0.24Kinase Inhibitor Selectivity Profiling Assay [AID1433_119, Type: confirmatory]
View
25
[SID50100098]
[CID6445562]
0.24Kinase Inhibitor Selectivity Profiling Assay [AID1433_19, Type: confirmatory]
View
26
[SID50100094]
[CID156414]
0.26Kinase Inhibitor Selectivity Profiling Assay [AID1433_118, Type: confirmatory]
View
27
[SID50100094]
[CID156414]
0.26Kinase Inhibitor Selectivity Profiling Assay [AID1433_81, Type: confirmatory]
View
28
[SID50100094]
[CID156414]
0.26Kinase Inhibitor Selectivity Profiling Assay [AID1433_82, Type: confirmatory]
View
29
[SID50100098]
[CID6445562]
0.27Kinase Inhibitor Selectivity Profiling Assay [AID1433_81, Type: confirmatory]
View
30
[SID22409543]
[CID2303746]
Potency 0.3162Assay for Inhibitors of the ERK Signaling Pathway using a Homogeneous Screening Assay: EGFR T790M Kinase Inhibition [AID1729, Type: confirmatory]
View
31
[SID50100098]
[CID6445562]
0.33Kinase Inhibitor Selectivity Profiling Assay [AID1433_175, Type: confirmatory]
View
32
[SID50100099]
[CID176870]
0.35Kinase Inhibitor Selectivity Profiling Assay [AID1433_82, Type: confirmatory]
View
33
[SID22409885]
[CID2322338]
Potency 0.3548Assay for Inhibitors of the ERK Signaling Pathway using a Homogeneous Screening Assay: EGFR T790M Kinase Inhibition [AID1729, Type: confirmatory]
View
34
[SID26755744]
[CID44259]
Potency 0.3548Assay for Inhibitors of the ERK Signaling Pathway using a Homogeneous Screening Assay: EGFR L858R Kinase Inhibition [AID1727, Type: confirmatory]
View
35
[SID50100098]
[CID6445562]
0.38Kinase Inhibitor Selectivity Profiling Assay [AID1433_118, Type: confirmatory]
View
36
[SID26755744]
[CID44259]
Potency 0.3981Assay for Inhibitors of the ERK Signaling Pathway using a Homogeneous Screening Assay: EGFR Kinase Inhibition [AID1731, Type: confirmatory]
View
37
[SID50100098]
[CID6445562]
0.41Kinase Inhibitor Selectivity Profiling Assay [AID1433_119, Type: confirmatory]
View
38
[SID50100098]
[CID6445562]
0.42Kinase Inhibitor Selectivity Profiling Assay [AID1433_79, Type: confirmatory]
View
39
[SID50100098]
[CID6445562]
0.44Kinase Inhibitor Selectivity Profiling Assay [AID1433_83, Type: confirmatory]
View
40
[SID50100098]
[CID6445562]
0.44Kinase Inhibitor Selectivity Profiling Assay [AID1433_78, Type: confirmatory]
View
41
[SID26755744]
[CID44259]
EGFR IC50 0.4467Quantitative High-Throughput Screen for Inhibitors of the ERK Signaling Pathway using a Homogeneous Screening Assay: Summary [AID1742, Type: summary]
View
42
[SID50100099]
[CID176870]
0.47Kinase Inhibitor Selectivity Profiling Assay [AID1433_81, Type: confirmatory]
View
43
[SID50100099]
[CID176870]
0.48Kinase Inhibitor Selectivity Profiling Assay [AID1433_118, Type: confirmatory]
View
44
[SID50100099]
[CID176870]
0.52Kinase Inhibitor Selectivity Profiling Assay [AID1433_79, Type: confirmatory]
View
45
[SID50100099]
[CID176870]
0.52Kinase Inhibitor Selectivity Profiling Assay [AID1433_80, Type: confirmatory]
View
46
[SID50100103]
[CID123631]
0.52Kinase Inhibitor Selectivity Profiling Assay [AID1433_82, Type: confirmatory]
View
47
[SID50100103]
[CID123631]
0.54Kinase Inhibitor Selectivity Profiling Assay [AID1433_118, Type: confirmatory]
View
48
[SID50100103]
[CID123631]
0.57Kinase Inhibitor Selectivity Profiling Assay [AID1433_80, Type: confirmatory]
View
49
[SID50100103]
[CID123631]
0.57Kinase Inhibitor Selectivity Profiling Assay [AID1433_81, Type: confirmatory]
View
50
[SID22409885]
[CID2322338]
Potency 0.631Assay for Inhibitors of the ERK Signaling Pathway using a Homogeneous Screening Assay: EGFR L858R Kinase Inhibition [AID1727, Type: confirmatory]
View