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Mu-type opioid receptor; M-OR-1; MOR-1; Mu op.. [gi:2851402] - Target BioActivity Data
Also known as: Mu-type opioid receptor; M-OR-1; MOR-1; Mu opiate receptor; Mu opioid receptor; MOP; hMOP.
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BioActivity Outcomes:
Active(3007)
 
 
BioAssay Types:
Literature(2905)
 
 
BioActivity Types:
Ki(1751)
 
 
IC50(508)
 
 
EC50(366)
 
 
Kd(20)
 
 
Substance Types:
Chemical(3007)
 
 
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Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 310    Data Row: 3007   Total Pages: 61   Display: Page     
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#StructureSubstanceCompoundActivityBioAssayLinks
OutcomeTypeValue [μM]
1
[SID164129496]
[CID71605589]
EC50 4.2e-08Agonist activity at FLAG-tagged mu-type opioid receptor (unknown origin) expressed in HEK293 cells assessed as inhibition of forskolin-stimulated cAMP accumulation after 30 mins by liquid scintillation counting analysis [AID730862, Type: Literature]
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2
[SID164140762]
[CID71605588]
EC50 9.12e-08Agonist activity at FLAG-tagged mu-type opioid receptor (unknown origin) expressed in HEK293 cells assessed as inhibition of forskolin-stimulated cAMP accumulation after 30 mins by liquid scintillation counting analysis [AID730862, Type: Literature]
View
3
[SID164129460]
[CID71605755]
EC50 1.07e-07Agonist activity at FLAG-tagged mu-type opioid receptor (unknown origin) expressed in HEK293 cells assessed as inhibition of forskolin-stimulated cAMP accumulation after 30 mins by liquid scintillation counting analysis [AID730862, Type: Literature]
View
4
[SID164140761]
[CID71605756]
EC50 1.09e-07Agonist activity at FLAG-tagged mu-type opioid receptor (unknown origin) expressed in HEK293 cells assessed as inhibition of forskolin-stimulated cAMP accumulation after 30 mins by liquid scintillation counting analysis [AID730862, Type: Literature]
View
5
[SID164149159]
[CID71720682]
EC50 1.3e-07Agonist activity at FLAG-tagged mu-type opioid receptor (unknown origin) expressed in HEK293 cells assessed as inhibition of forskolin-stimulated cAMP accumulation after 30 mins by liquid scintillation counting analysis [AID730862, Type: Literature]
View
6
[SID164143536]
[CID71719454]
EC50 5.16e-07Agonist activity at FLAG-tagged mu-type opioid receptor (unknown origin) expressed in HEK293 cells assessed as inhibition of forskolin-stimulated cAMP accumulation after 30 mins by liquid scintillation counting analysis [AID730862, Type: Literature]
View
7
[SID103293205]
[CID5311080]
EC50 1e-06Activity at mu opioid receptor assessed as increase in calcium level in CHO cells by aequorin luminescence based calcium assay [AID277678, Type: Literature]
View
8
[SID163339747]
[CID58443234]
Ki 1.6e-06Displacement of [3H]DAMGO from human mu opioid receptor expressed in CHO cells after 60 mins by scintillation counting [AID719453, Type: Literature]
View
9
[SID163337288]
[CID54669894]
EC50 1.74e-06Agonist activity at human MOR expressed in HEK293 cell membrane assessed as inhibition of forskolin-induced cAMP accumulation by by liquid scintillation counting [AID690645, Type: Literature]
View
10
[SID134434099]
[CID6602241]
Ki 3e-06Displacement of [3H]DAMGO from human mu opioid receptor expressed in CHO cells [AID259394, Type: Literature]
View
11
[SID164129496]
[CID71605589]
Ki 3.72e-06Displacement of [3H]DAMGO from FLAG-tagged mu-type opioid receptor (unknown origin) expressed in HEK293 cells after 60 mins by liquid scintillation counting analysis [AID730870, Type: Literature]
View
12
[SID163322529]
[CID71454361]
Ki 4.9e-06Displacement of [3H]DAMGO from human mu opioid receptor expressed in CHO cells after 60 mins by scintillation counting [AID719453, Type: Literature]
View
13
[SID163322528]
[CID58443225]
Ki 5.6e-06Displacement of [3H]DAMGO from human mu opioid receptor expressed in CHO cells after 60 mins by scintillation counting [AID719453, Type: Literature]
View
14
[SID163325912]
[CID71456106]
Ki 5.6e-06Displacement of [3H]DAMGO from human mu opioid receptor expressed in CHO cells after 60 mins by scintillation counting [AID719453, Type: Literature]
View
15
[SID163322530]
[CID71454362]
Ki 7.1e-06Displacement of [3H]DAMGO from human mu opioid receptor expressed in CHO cells after 60 mins by scintillation counting [AID719453, Type: Literature]
View
16
[SID164137991]
[CID71605419]
EC50 8.53e-06Agonist activity at FLAG-tagged mu-type opioid receptor (unknown origin) expressed in HEK293 cells assessed as inhibition of forskolin-stimulated cAMP accumulation after 30 mins by liquid scintillation counting analysis [AID730862, Type: Literature]
View
17
[SID164140762]
[CID71605588]
Ki 9.86e-06Displacement of [3H]DAMGO from FLAG-tagged mu-type opioid receptor (unknown origin) expressed in HEK293 cells after 60 mins by liquid scintillation counting analysis [AID730870, Type: Literature]
View
18
[SID103476378]
[CID44406663]
Ki 1e-05Displacement of [3H]DAMGO from human mu opioid receptor expressed in CHO cells [AID259394, Type: Literature]
View
19
[SID103500785]
[CID16087283]
IC50 1.25e-05Activity at human recombinant mu opioid receptor expressed in CHO cells assessed as stimulation of [35S]GTP-gamma-S binding [AID273141, Type: Literature]
View
20
[SID164140761]
[CID71605756]
Ki 1.28e-05Displacement of [3H]DAMGO from FLAG-tagged mu-type opioid receptor (unknown origin) expressed in HEK293 cells after 60 mins by liquid scintillation counting analysis [AID730870, Type: Literature]
View
21
[SID164129460]
[CID71605755]
Ki 1.37e-05Displacement of [3H]DAMGO from FLAG-tagged mu-type opioid receptor (unknown origin) expressed in HEK293 cells after 60 mins by liquid scintillation counting analysis [AID730870, Type: Literature]
View
22
[SID103607911]
[CID25181466]
Ki 1.5e-05Displacement of [3H]DAMGO form human mu opioid receptor expressed in CHO cells [AID410718, Type: Literature]
View
23
[SID163329343]
[CID24873473]
Ki 1.8e-05Displacement of [3H]DAMGO from human mu opioid receptor expressed in CHO cells after 60 mins by scintillation counting [AID719453, Type: Literature]
View
24
[SID131283791]
[CID5360515]
Ki 2e-05Ratio of mu/delta-opioid receptors Binding affinity [AID228132, Type: Literature]
View
25
[SID163332933]
[CID71459821]
Ki 2.1e-05Displacement of [3H]DAMGO from human mu opioid receptor expressed in CHO cells after 60 mins by scintillation counting [AID719453, Type: Literature]
View
26
[SID103705684]
[CID44627899]
Ki 2.6e-05Displacement of [3H]DAMGO from human mu opioid receptor expressed in CHO cells [AID445095, Type: Literature]
View
27
[SID103500899]
[CID16087270]
IC50 2.8e-05Activity at human recombinant mu opioid receptor expressed in CHO cells assessed as stimulation of [35S]GTP-gamma-S binding [AID273141, Type: Literature]
View
28
[SID103500794]
[CID16087275]
IC50 3e-05Activity at human recombinant mu opioid receptor expressed in CHO cells assessed as stimulation of [35S]GTP-gamma-S binding [AID273141, Type: Literature]
View
29
[SID164149159]
[CID71720682]
Ki 3.22e-05Displacement of [3H]DAMGO from FLAG-tagged mu-type opioid receptor (unknown origin) expressed in HEK293 cells after 60 mins by liquid scintillation counting analysis [AID730870, Type: Literature]
View
30
[SID164132274]
[CID71605418]
EC50 3.97e-05Agonist activity at FLAG-tagged mu-type opioid receptor (unknown origin) expressed in HEK293 cells assessed as inhibition of forskolin-stimulated cAMP accumulation after 30 mins by liquid scintillation counting analysis [AID730862, Type: Literature]
View
31
[SID163326400]
[CID71456262]
EC50 4e-05Stimulation of [35S]GTPgammaS binding to human recombinant MOR [AID269575, Type: Literature]
View
32
[SID103347472]
[CID5311081]
EC50 4e-05Activity at mu opioid receptor assessed as increase in calcium level in CHO cells by aequorin luminescence based calcium assay [AID277678, Type: Literature]
View
33
[SID103735540]
[CID11849285]
EC50 4e-05Stimulation of [35S]GTPgammaS binding to human recombinant MOR [AID269575, Type: Literature]
View
34
[SID164143536]
[CID71719454]
Ki 4.05e-05Displacement of [3H]DAMGO from FLAG-tagged mu-type opioid receptor (unknown origin) expressed in HEK293 cells after 60 mins by liquid scintillation counting analysis [AID730870, Type: Literature]
View
35
[SID103234501]
[CID9906198]
Ki 4.3e-05Antagonist activity at human mu opioid receptor expressed in CHO cells by [35S]GTP-gamma-S binding assay [AID301031, Type: Literature]
View
36
[SID103577221]
[CID24824635]
Ki 5e-05Displacement of [3H]DAMGO from human mu opioid receptor expressed in CHO cells [AID317853, Type: Literature]
View
37
[SID131283791]
[CID5360515]
Kd 5.01e-05Activity at human mu opioid receptor by [35S]GTPgammaS binding assay [AID317858, Type: Literature]
View
38
[SID103653141]
[CID44592018]
Ki 5.2e-05Displacement of [3H]DAMGO from human mu opioid receptor expressed in CHO cells after 60 mins by scintillation counting [AID416813, Type: Literature]
View
39
[SID103465875]
[CID11667832]
Ki 5.2e-05Binding affinity against Opioid receptor mu 1 expressed in CHO cells using [3H]DAMGO as radioligand [AID238974, Type: Literature]
View
40
[SID164140760]
[CID71605420]
EC50 5.7e-05Agonist activity at FLAG-tagged mu-type opioid receptor (unknown origin) expressed in HEK293 cells assessed as inhibition of forskolin-stimulated cAMP accumulation after 30 mins by liquid scintillation counting analysis [AID730862, Type: Literature]
View
41
[SID163315590]
[CID58443217]
Ki 5.9e-05Displacement of [3H]DAMGO from human mu opioid receptor expressed in CHO cells after 60 mins by scintillation counting [AID719453, Type: Literature]
View
42
[SID103531554]
[CID11983337]
Ki 5.9e-05Displacement of [3H]DAMGO from mu opioid receptor in human SHSY5Y cells [AID408420, Type: Literature]
View
43
[SID103576500]
[CID44456785]
Ki 6e-05Displacement of [3H]DAMGO from human mu opioid receptor expressed in CHO cells [AID317853, Type: Literature]
View
44
[SID103642833]
[CID44586917]
Ki 6.1e-05Displacement of [3H]DAMGO from human mu opioid receptor expressed in CHO cell membrane [AID362196, Type: Literature]
View
45
[SID103230838]
[CID5359966]
Ki 6.2e-05Displacement of [3H]DAMGO from human mu opioid receptor expressed in CHO membrane [AID296053, Type: Literature]
View
46
[SID103230838]
[CID5359966]
Ki 6.2e-05Displacement of [3H]DAMGO from human mu opioid receptors expressed in CHO cell membrane [AID290256, Type: Literature]
View
47
[SID103230838]
[CID5359966]
Ki 6.2e-05Displacement of [3H]DAMGO from human mu opioid receptor expressed in CHO cells [AID445095, Type: Literature]
View
48
[SID103230838]
[CID5359966]
Ki 6.2e-05Displacement of [3H]DAMGO from human mu opioid receptor expressed in CHO cells after 60 mins by scintillation counting [AID592435, Type: Literature]
View
49
[SID103230838]
[CID5359966]
Ki 6.2e-05Displacement of [3H]-DAMGO from human mu opioid receptor expressed in CHO cells after 60 mins by scintillation counting [AID670110, Type: Literature]
View
50
[SID103242977]
[CID44299063]
Ki 6.2e-05Displacement of [3H]DAMGO from human mu opioid receptor expressed in CHO cells [AID259394, Type: Literature]
View