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BioActivity Data for Target Mu-type opioid receptor [gi:2851402]

Filters: All Data » Active      
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BioActivity Outcomes:
Active(3375)
 
 
BioAssay Types:
Literature(3311)
 
 
Confirmatory(42)
 
 
BioAssay Categories:
Biochemical(3146)
 
 
Cell-based(2720)
 
 
ADME(4)
 
 
In vitro(119)
 
 
BioActivity Types:
Ki(1942)
 
 
IC50(484)
 
 
EC50(479)
 
 
Kd(20)
 
 
Substance Types:
Chemical(3375)
 
 
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Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 363    Data Row: 3375   Total Pages: 169   Display: Page     
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#StructureSubstanceCompoundActivityBioAssayLinks
OutcomeTypeValue [μM]
1
[SID163339747]
[CID58443234]
Ki 1.6e-06Displacement of [3H]DAMGO from human mu opioid receptor expressed in CHO cells after 60 mins by scintillation counting [AID719453, Type: Literature]
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2
[SID163337288]
[CID54669894]
EC50 1.74e-06Agonist activity at human MOR expressed in HEK293 cell membrane assessed as inhibition of forskolin-induced cAMP accumulation by by liquid scintillation counting [AID690645, Type: Literature]
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3
[SID134434099]
[CID6602241]
Ki 3e-06Displacement of [3H]DAMGO from human mu opioid receptor expressed in CHO cells [AID259394, Type: Literature]
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4
[SID164129496]
[CID71605589]
Ki 3.72e-06Displacement of [3H]DAMGO from FLAG-tagged mu-type opioid receptor (unknown origin) expressed in HEK293 cells after 60 mins by liquid scintillation counting analysis [AID730870, Type: Literature]
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5
[SID163322529]
[CID71454361]
Ki 4.9e-06Displacement of [3H]DAMGO from human mu opioid receptor expressed in CHO cells after 60 mins by scintillation counting [AID719453, Type: Literature]
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6
[SID163322528]
[CID58443225]
Ki 5.6e-06Displacement of [3H]DAMGO from human mu opioid receptor expressed in CHO cells after 60 mins by scintillation counting [AID719453, Type: Literature]
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7
[SID163325912]
[CID71456106]
Ki 5.6e-06Displacement of [3H]DAMGO from human mu opioid receptor expressed in CHO cells after 60 mins by scintillation counting [AID719453, Type: Literature]
View
8
[SID163322530]
[CID71454362]
Ki 7.1e-06Displacement of [3H]DAMGO from human mu opioid receptor expressed in CHO cells after 60 mins by scintillation counting [AID719453, Type: Literature]
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9
[SID164140762]
[CID71605588]
Ki 9.86e-06Displacement of [3H]DAMGO from FLAG-tagged mu-type opioid receptor (unknown origin) expressed in HEK293 cells after 60 mins by liquid scintillation counting analysis [AID730870, Type: Literature]
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10
[SID103248656]
[CID44301701]
Ki 1e-05Binding affinity to mu opioid receptor (unknown origin) [AID754478, Type: Literature]
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11
[SID103476378]
[CID44406663]
Ki 1e-05Displacement of [3H]DAMGO from human mu opioid receptor expressed in CHO cells [AID259394, Type: Literature]
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12
[SID103500785]
[CID16087283]
IC50 1.25e-05Activity at human recombinant mu opioid receptor expressed in CHO cells assessed as stimulation of [35S]GTP-gamma-S binding [AID273141, Type: Literature]
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13
[SID164140761]
[CID71605756]
Ki 1.28e-05Displacement of [3H]DAMGO from FLAG-tagged mu-type opioid receptor (unknown origin) expressed in HEK293 cells after 60 mins by liquid scintillation counting analysis [AID730870, Type: Literature]
View
14
[SID164129460]
[CID71605755]
Ki 1.37e-05Displacement of [3H]DAMGO from FLAG-tagged mu-type opioid receptor (unknown origin) expressed in HEK293 cells after 60 mins by liquid scintillation counting analysis [AID730870, Type: Literature]
View
15
[SID103607911]
[CID25181466]
Ki 1.5e-05Displacement of [3H]DAMGO form human mu opioid receptor expressed in CHO cells [AID410718, Type: Literature]
View
16
[SID163329343]
[CID24873473]
Ki 1.8e-05Displacement of [3H]DAMGO from human mu opioid receptor expressed in CHO cells after 60 mins by scintillation counting [AID719453, Type: Literature]
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17
[SID131283791]
[CID5360515]
Ki 2e-05Ratio of mu/delta-opioid receptors Binding affinity [AID228132, Type: Literature]
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18
[SID163332933]
[CID71459821]
Ki 2.1e-05Displacement of [3H]DAMGO from human mu opioid receptor expressed in CHO cells after 60 mins by scintillation counting [AID719453, Type: Literature]
View
19
[SID103705684]
[CID44627899]
Ki 2.6e-05Displacement of [3H]DAMGO from human mu opioid receptor expressed in CHO cells [AID445095, Type: Literature]
View
20
[SID103500899]
[CID16087270]
IC50 2.8e-05Activity at human recombinant mu opioid receptor expressed in CHO cells assessed as stimulation of [35S]GTP-gamma-S binding [AID273141, Type: Literature]
View