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MAP kinase-activated protein kinase 2; MAPK-a.. [gi:1346538] - Target BioActivity Data
Also known as: MAP kinase-activated protein kinase 2; MAPK-activated protein kinase 2; MAPKAP kinase 2; MAPKAP-K2; MAPKAPK-2; MK-2; MK2.
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BioActivity Outcomes:
Active(578)
 
 
BioAssay Types:
Literature(578)
 
 
BioActivity Types:
IC50(477)
 
 
EC50(79)
 
 
Kd(7)
 
 
Ki(5)
 
 
Substance Types:
Chemical(578)
 
 
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Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 56    Data Row: 578   Total Pages: 29   Display: Page     
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#StructureSubstanceCompoundActivityBioAssayLinks
OutcomeTypeValue [μM]
1
[SID134436469]
[CID56659490]
IC50 0.001Inhibition of human MK2 using hsp27 peptide biotinyl-AYSRALSRQLSSGVSEIRCOOH as substrate after 45 mins by FRET assay [AID604988, Type: Literature]
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2
[SID174516734]
[CID53235497]
IC50 0.0019Inhibition of MK2 (unknown origin) phosphorylation using TAMRA labeled peptide as substrate incubated 30 mins before substrate addition measured after 30 mins [AID749353, Type: Literature]
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3
[SID174516735]
[CID71625683]
IC50 0.003Inhibition of MK2 (unknown origin) phosphorylation using TAMRA labeled peptide as substrate incubated 30 mins before substrate addition measured after 30 mins [AID749353, Type: Literature]
View
4
[SID134444187]
[CID56666415]
IC50 0.003Inhibition of human MK2 using biotinyl-AYSRALSRQLSSGVSEIRCOOH as substrate after 45 mins by FRET analysis [AID604890, Type: Literature]
View
5
[SID134444188]
[CID56666416]
IC50 0.003Inhibition of human MK2 using biotinyl-AYSRALSRQLSSGVSEIRCOOH as substrate after 45 mins by FRET analysis [AID604890, Type: Literature]
View
6
[SID134448078]
[CID56669831]
IC50 0.003Inhibition of human MK2 using biotinyl-AYSRALSRQLSSGVSEIRCOOH as substrate after 45 mins by FRET analysis [AID604890, Type: Literature]
View
7
[SID134448079]
[CID56669832]
IC50 0.003Inhibition of human MK2 using biotinyl-AYSRALSRQLSSGVSEIRCOOH as substrate after 45 mins by FRET analysis [AID604890, Type: Literature]
View
8
[SID134451969]
[CID56673316]
IC50 0.003Inhibition of human MK2 using biotinyl-AYSRALSRQLSSGVSEIRCOOH as substrate after 45 mins by FRET analysis [AID604890, Type: Literature]
View
9
[SID134455766]
[CID56676654]
IC50 0.003Inhibition of human MK2 using biotinyl-AYSRALSRQLSSGVSEIRCOOH as substrate after 45 mins by FRET analysis [AID604890, Type: Literature]
View
10
[SID134455767]
[CID56676655]
IC50 0.003Inhibition of human MK2 using biotinyl-AYSRALSRQLSSGVSEIRCOOH as substrate after 45 mins by FRET analysis [AID604890, Type: Literature]
View
11
[SID134455768]
[CID56676656]
IC50 0.003Inhibition of human MK2 using biotinyl-AYSRALSRQLSSGVSEIRCOOH as substrate after 45 mins by FRET analysis [AID604890, Type: Literature]
View
12
[SID134455771]
[CID42646706]
IC50 0.003Inhibition of human MK2 using biotinyl-AYSRALSRQLSSGVSEIRCOOH as substrate after 45 mins by FRET analysis [AID604890, Type: Literature]
View
13
[SID104250105]
[CID42646698]
IC50 0.003Inhibition of human MK2 using biotinyl-AYSRALSRQLSSGVSEIRCOOH as substrate after 45 mins by FRET analysis [AID604890, Type: Literature]
View
14
[SID134440359]
[CID56662943]
IC50 0.004Inhibition of human MK2 using biotinyl-AYSRALSRQLSSGVSEIRCOOH as substrate after 45 mins by FRET analysis [AID604890, Type: Literature]
View
15
[SID103746415]
[CID25052767]
IC50 0.0043Inhibition of LPS-induced MK2 phosphorylation in human whole blood treated 30 mins before LPS challenge measured after 45 mins by FACS analysis [AID476158, Type: Literature]
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16
[SID174521920]
[CID71625566]
IC50 0.0049Inhibition of MK2 (unknown origin) phosphorylation using TAMRA labeled peptide as substrate incubated 30 mins before substrate addition measured after 30 mins [AID749353, Type: Literature]
View
17
[SID134440369]
[CID25066415]
IC50 0.005Inhibition of human MK2 using hsp27 peptide biotinyl-AYSRALSRQLSSGVSEIRCOOH as substrate after 45 mins by FRET assay [AID604988, Type: Literature]
View
18
[SID134444194]
[CID25066206]
IC50 0.005Inhibition of human MK2 using hsp27 peptide biotinyl-AYSRALSRQLSSGVSEIRCOOH as substrate after 45 mins by FRET assay [AID604988, Type: Literature]
View
19
[SID134436470]
[CID25065561]
IC50 0.005Inhibition of human MK2 using hsp27 peptide biotinyl-AYSRALSRQLSSGVSEIRCOOH as substrate after 45 mins by FRET assay [AID604988, Type: Literature]
View
20
[SID174491027]
[CID53251322]
IC50 0.0057Inhibition of MK2 (unknown origin) phosphorylation using TAMRA labeled peptide as substrate incubated 30 mins before substrate addition measured after 30 mins [AID749353, Type: Literature]
View