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RAC-gamma serine/threonine-protein kinase; Pr.. [gi:12643943] - Target BioActivity Data
Also known as: RAC-gamma serine/threonine-protein kinase; Protein kinase Akt-3; Protein kinase B gamma; PKB gamma; RAC-PK-gamma; STK-2.
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BioActivity Outcomes:
Active(150)
 
 
BioAssay Types:
Literature(150)
 
 
BioActivity Types:
IC50(132)
 
 
Kd(10)
 
 
Ki(3)
 
 
EC50(3)
 
 
Substance Types:
Chemical(150)
 
 
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Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 22    Data Row: 150   Total Pages: 8   Display: Page     
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#StructureSubstanceCompoundActivityBioAssayLinks
OutcomeTypeValue [μM]
1
[SID103718372]
[CID46226079]
IC50 0.001Inhibition of human AKT3 [AID455026, Type: Literature]
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2
[SID103718442]
[CID46226137]
IC50 0.001Inhibition of human AKT3 [AID455026, Type: Literature]
View
3
[SID103718472]
[CID46226156]
IC50 0.001Inhibition of human AKT3 [AID455026, Type: Literature]
View
4
[SID163331672]
[CID58458278]
IC50 0.001Competitive inhibition of wild-type full-length amino-terminal polyhistidine-tagged human Akt3 expressed in recombinant baculovirus system using fluorescence labeled Crosstide as substrate after 60 mins by fluorescence polarization assay in presence of ATP [AID708171, Type: Literature]
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5
[SID163335288]
[CID58191081]
IC50 0.002Competitive inhibition of wild-type full-length amino-terminal polyhistidine-tagged human Akt3 expressed in recombinant baculovirus system using fluorescence labeled Crosstide as substrate after 60 mins by fluorescence polarization assay in presence of ATP [AID708171, Type: Literature]
View
6
[SID103718441]
[CID46226136]
IC50 0.002Inhibition of human AKT3 [AID455026, Type: Literature]
View
7
[SID103718373]
[CID46226080]
IC50 0.002Inhibition of human AKT3 [AID455026, Type: Literature]
View
8
[SID103718374]
[CID25190977]
IC50 0.002Inhibition of human AKT3 [AID455026, Type: Literature]
View
9
[SID163321303]
[CID59671151]
IC50 0.002Competitive inhibition of wild-type full-length amino-terminal polyhistidine-tagged human Akt3 expressed in recombinant baculovirus system using fluorescence labeled Crosstide as substrate after 60 mins by fluorescence polarization assay in presence of ATP [AID708171, Type: Literature]
View
10
[SID103495052]
[CID16043304]
IC50 0.0026Inhibition of AKT3 in presence of 0.2 uM ATP [AID269858, Type: Literature]
View
11
[SID103495052]
[CID16043304]
IC50 0.003Inhibition of AKT3 [AID269861, Type: Literature]
View
12
[SID103718397]
[CID25222706]
IC50 0.003Inhibition of human AKT3 [AID455026, Type: Literature]
View
13
[SID103604655]
[CID16725726]
Kd 0.003Binding constant for AKT3 kinase domain [AID625019, Type: Literature]
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14
[SID163338532]
[CID58191080]
IC50 0.003Competitive inhibition of wild-type full-length amino-terminal polyhistidine-tagged human Akt3 expressed in recombinant baculovirus system using fluorescence labeled Crosstide as substrate after 60 mins by fluorescence polarization assay in presence of ATP [AID708171, Type: Literature]
View
15
[SID163338659]
[CID70676464]
IC50 0.003Competitive inhibition of wild-type full-length amino-terminal polyhistidine-tagged human Akt3 expressed in recombinant baculovirus system using fluorescence labeled Crosstide as substrate after 60 mins by fluorescence polarization assay in presence of ATP [AID708171, Type: Literature]
View
16
[SID164128907]
[CID42602264]
IC50 0.004Inhibition of recombinant Akt3 (unknown origin) using 5-FAM-labeled peptide as substrate after 1 hr by caliper off-chip incubation mobility shift assay [AID728521, Type: Literature]
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17
[SID163317839]
[CID59671148]
IC50 0.004Competitive inhibition of wild-type full-length amino-terminal polyhistidine-tagged human Akt3 expressed in recombinant baculovirus system using fluorescence labeled Crosstide as substrate after 60 mins by fluorescence polarization assay in presence of ATP [AID708171, Type: Literature]
View
18
[SID163314381]
[CID70676312]
IC50 0.004Competitive inhibition of wild-type full-length amino-terminal polyhistidine-tagged human Akt3 expressed in recombinant baculovirus system using fluorescence labeled Crosstide as substrate after 60 mins by fluorescence polarization assay in presence of ATP [AID708171, Type: Literature]
View
19
[SID103495241]
[CID44414579]
IC50 0.0048Inhibition of AKT3 in presence of 0.2 uM ATP [AID269858, Type: Literature]
View
20
[SID103243222]
[CID44299148]
IC50 0.005Inhibition of AKT3 [AID269861, Type: Literature]
View