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Serine/threonine-protein kinase mTOR; FK506-b.. [gi:1169735] - Target BioActivity Data
Also known as: Serine/threonine-protein kinase mTOR; FK506-binding protein 12-rapamycin complex-associated protein 1; FKBP12-rapamycin complex-associated protein; Mammalian target of rapamycin; mTOR; Mechanistic target of rapamycin; Rapamycin and FKBP12 target 1; Rapamycin target protein 1.
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BioActivity Outcomes:
Active(607)
 
 
BioAssay Types:
Literature(578)
 
 
BioActivity Types:
IC50(435)
 
 
Ki(141)
 
 
Kd(4)
 
 
Substance Types:
Chemical(607)
 
 
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Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 69    Data Row: 607   Total Pages: 13   Display: Page     
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#StructureSubstanceCompoundActivityBioAssayLinks
OutcomeTypeValue [μM]
1
[SID103691165]
[CID24936050]
IC50 8e-05Inhibition of flag-tagged truncated human mTOR (1360-2549) expressed in HEK293 cells by DELFIA assay [AID422366, Type: Literature]
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2
[SID103164548]
[CID5284616]
IC50 0.0001Inhibition of mTOR kinase expressed in human HEK293 cells by western blot analysis [AID360764, Type: Literature]
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3
[SID103709118]
[CID25262783]
IC50 0.0001Inhibition of human FLAG-tagged mTOR expressed in HEK293 cells after 2 hrs by DELFIA [AID444218, Type: Literature]
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4
[SID103709137]
[CID45488052]
IC50 0.0001Inhibition of human FLAG-tagged mTOR expressed in HEK293 cells after 2 hrs by DELFIA [AID444218, Type: Literature]
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5
[SID103709147]
[CID45488058]
IC50 0.0001Inhibition of human FLAG-tagged mTOR expressed in HEK293 cells after 2 hrs by DELFIA [AID444218, Type: Literature]
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6
[SID103749989]
[CID44605039]
IC50 0.0001Inhibition of human mTOR (1360-2549 amino acids) expressed in HEK293 cells [AID477628, Type: Literature]
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7
[SID103697308]
[CID25261555]
IC50 0.00011Inhibition of FLAG-tagged human mTOR by DELFIA method [AID442311, Type: Literature]
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8
[SID134448064]
[CID25262965]
IC50 0.00013Inhibition of recombinant FLAG-tagged mTOR (1362 to 2549) (unknown origin) expressed in HEK293 cells [AID735578, Type: Literature]
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9
[SID103697309]
[CID45482923]
IC50 0.00016Inhibition of FLAG-tagged human mTOR by DELFIA method [AID442311, Type: Literature]
View
10
[SID103697342]
[CID45482935]
IC50 0.00017Inhibition of FLAG-tagged human mTOR by DELFIA method [AID442311, Type: Literature]
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11
[SID103697542]
[CID25261230]
IC50 0.00019Inhibition of FLAG-tagged human mTOR by DELFIA method [AID442311, Type: Literature]
View
12
[SID103697567]
[CID45482982]
IC50 0.0002Inhibition of FLAG-tagged human mTOR by DELFIA method [AID442311, Type: Literature]
View
13
[SID103697517]
[CID44606133]
IC50 0.0002Inhibition of mTOR in HEK293 cells by DELFIA assay [AID453451, Type: Literature]
View
14
[SID103697409]
[CID45482947]
IC50 0.0002Inhibition of FLAG-tagged human mTOR by DELFIA method [AID442311, Type: Literature]
View
15
[SID103682456]
[CID44233639]
IC50 0.0002Inhibition of flag-tagged truncated human mTOR (1360-2549) expressed in HEK293 cells by DELFIA assay [AID422366, Type: Literature]
View
16
[SID103682456]
[CID44233639]
IC50 0.0002Inhibition of FLAG-tagged human mTOR by DELFIA method [AID442311, Type: Literature]
View
17
[SID103749951]
[CID44605249]
IC50 0.0002Inhibition of human mTOR (1360-2549 amino acids) expressed in HEK293 cells [AID477628, Type: Literature]
View
18
[SID103709149]
[CID45488060]
IC50 0.0002Inhibition of human FLAG-tagged mTOR expressed in HEK293 cells after 2 hrs by DELFIA [AID444218, Type: Literature]
View
19
[SID103709150]
[CID45488061]
IC50 0.0002Inhibition of human FLAG-tagged mTOR expressed in HEK293 cells after 2 hrs by DELFIA [AID444218, Type: Literature]
View
20
[SID103709179]
[CID45488080]
IC50 0.0002Inhibition of human FLAG-tagged mTOR expressed in HEK293 cells after 2 hrs by DELFIA [AID444218, Type: Literature]
View
21
[SID103709097]
[CID45488032]
IC50 0.0002Inhibition of human FLAG-tagged mTOR expressed in HEK293 cells after 2 hrs by DELFIA [AID444218, Type: Literature]
View
22
[SID103697316]
[CID45482926]
IC50 0.00022Inhibition of FLAG-tagged human mTOR by DELFIA method [AID442311, Type: Literature]
View
23
[SID103697306]
[CID25261389]
IC50 0.00022Inhibition of FLAG-tagged human mTOR by DELFIA method [AID442311, Type: Literature]
View
24
[SID103697275]
[CID25261388]
IC50 0.00023Inhibition of FLAG-tagged human mTOR by DELFIA method [AID442311, Type: Literature]
View
25
[SID103697517]
[CID44606133]
IC50 0.00023Inhibition of FLAG-tagged human mTOR by DELFIA method [AID442311, Type: Literature]
View
26
[SID164148752]
[CID58379501]
Ki 0.000243Inhibition of mTOR (unknown origin) [AID732390, Type: other]
View
27
[SID103697412]
[CID44606644]
IC50 0.00028Inhibition of FLAG-tagged human mTOR by DELFIA method [AID442311, Type: Literature]
View
28
[SID123085155]
[CID49836027]
IC50 0.00029Inhibition of human mTOR complex 1 after 30 mins by FRET assay [AID517847, Type: Literature]
View
29
[SID103749988]
[CID44605038]
IC50 0.0003Inhibition of human mTOR (1360-2549 amino acids) expressed in HEK293 cells [AID477628, Type: Literature]
View
30
[SID103749984]
[CID44605426]
IC50 0.0003Inhibition of human mTOR (1360-2549 amino acids) expressed in HEK293 cells [AID477628, Type: Literature]
View
31
[SID103749923]
[CID25195788]
IC50 0.0003Inhibition of human mTOR (1360-2549 amino acids) expressed in HEK293 cells [AID477628, Type: Literature]
View
32
[SID103709175]
[CID25262782]
IC50 0.0003Inhibition of human FLAG-tagged mTOR expressed in HEK293 cells after 2 hrs by DELFIA [AID444218, Type: Literature]
View
33
[SID103709176]
[CID45488077]
IC50 0.0003Inhibition of human FLAG-tagged mTOR expressed in HEK293 cells after 2 hrs by DELFIA [AID444218, Type: Literature]
View
34
[SID103709148]
[CID45488059]
IC50 0.0003Inhibition of human FLAG-tagged mTOR expressed in HEK293 cells after 2 hrs by DELFIA [AID444218, Type: Literature]
View
35
[SID103709168]
[CID45488070]
IC50 0.0003Inhibition of human FLAG-tagged mTOR expressed in HEK293 cells after 2 hrs by DELFIA [AID444218, Type: Literature]
View
36
[SID103692964]
[CID44233641]
IC50 0.0003Inhibition of human mTOR (1360-2549 amino acids) expressed in HEK293 cells [AID477628, Type: Literature]
View
37
[SID103687722]
[CID44233640]
IC50 0.0003Inhibition of flag-tagged truncated human mTOR (1360-2549) expressed in HEK293 cells by DELFIA assay [AID422366, Type: Literature]
View
38
[SID103692958]
[CID44233389]
IC50 0.00032Inhibition of flag-tagged truncated human mTOR (1360-2549) expressed in HEK293 cells by DELFIA assay [AID422366, Type: Literature]
View
39
[SID103692958]
[CID44233389]
IC50 0.00032Inhibition of FLAG-tagged human mTOR by DELFIA method [AID442311, Type: Literature]
View
40
[SID103692964]
[CID44233641]
IC50 0.00034Inhibition of flag-tagged truncated human mTOR (1360-2549) expressed in HEK293 cells by DELFIA assay [AID422366, Type: Literature]
View
41
[SID131276844]
[CID53237048]
Ki 0.00034Inhibition of human recombinant mTOR expressed in insect cells using 4E-BP1 substrate after 30 mins by fluorescence resonance energy transfer assay [AID597427, Type: Literature]
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42
[SID164131895]
[CID58379663]
Ki 0.000377Inhibition of mTOR (unknown origin) [AID732390, Type: other]
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43
[SID103687704]
[CID25260915]
IC50 0.00038Inhibition of flag-tagged truncated human mTOR (1360-2549) expressed in HEK293 cells by DELFIA assay [AID422366, Type: Literature]
View
44
[SID103687704]
[CID25260915]
IC50 0.00038Inhibition of FLAG-tagged human mTOR by DELFIA method [AID442311, Type: Literature]
View
45
[SID103687704]
[CID25260915]
IC50 0.0004Inhibition of human mTOR (1360-2549 amino acids) expressed in HEK293 cells [AID477628, Type: Literature]
View
46
[SID103750031]
[CID44605037]
IC50 0.0004Inhibition of human mTOR (1360-2549 amino acids) expressed in HEK293 cells [AID477628, Type: Literature]
View
47
[SID164131898]
[CID59239300]
Ki 0.0004Inhibition of recombinant mTOR (1360 to 2549)+GBL (unknown origin) using GFP-4E-BP1 as substrate after 30 mins by FRET assay [AID732418, Type: other]
View
48
[SID103685903]
[CID44233391]
IC50 0.00045Inhibition of flag-tagged truncated human mTOR (1360-2549) expressed in HEK293 cells by DELFIA assay [AID422366, Type: Literature]
View
49
[SID103682447]
[CID25261231]
IC50 0.00046Inhibition of flag-tagged truncated human mTOR (1360-2549) expressed in HEK293 cells by DELFIA assay [AID422366, Type: Literature]
View
50
[SID103682447]
[CID25261231]
IC50 0.00046Inhibition of FLAG-tagged human mTOR by DELFIA method [AID442311, Type: Literature]
View