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SCN9A (geneid:6335) - Gene BioActivity Data
Also known as: ETHA, FEB3B, GEFSP7, NE-NA, NENA, Nav1.7, PN1, SFNP.
Filters: All Data » Active      
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BioActivity Outcomes:
Active(649)
 
 
BioAssay Types:
Literature(603)
 
 
BioActivity Types:
IC50(571)
 
 
Ki(30)
 
 
Substance Types:
Chemical(649)
 
 
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Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 51    Data Row: 649   Total Pages: 13   Display: Page     
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#StructureSubstanceCompoundActivityBioAssayTargetLinks
OutcomeTypeValue [μM]
1
[SID104245048]
[CID11231810]
Ki 1.8e-05Inhibition of human Nav 1.7 channel by electrophysiology [AID502582, Type: Literature] [gi:327478559]
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2
[SID104245047]
[CID49866005]
Ki 0.000111Inhibition of human Nav 1.7 channel by electrophysiology [AID502582, Type: Literature] [gi:327478559]
View
3
[SID103561514]
[CID25033155]
IC50 0.00154Inhibition of human Nav1.7 sodium channel expressed in HEK293 cells at a membrane potential of -70 mV by whole cell voltage clamp technique [AID314683, Type: Literature] [gi:327478559]
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4
[SID131275324]
[CID11998198]
IC50 0.003Inhibition of human NaV1.7 expressed in HEK293 cells by [14C]guanidinium influx assay [AID599097, Type: Literature] [gi:327478559]
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5
[SID103585628]
[CID11174599]
IC50 0.006Inhibition of human NaV1.7 expressed in HEK293 cells by [14C]guanidinium influx assay [AID599097, Type: Literature] [gi:327478559]
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6
[SID103552455]
[CID24874828]
IC50 0.009Blockade of human Nav1.7 by FRET assay [AID308661, Type: Literature] [gi:327478559]
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7
[SID124968015]
[CID53322584]
IC50 0.01Inhibition of human Nav1.7 by VIPR assay [AID549473, Type: Literature] [gi:327478559]
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8
[SID104244979]
[CID9927558]
Ki 0.013Inhibition of human Nav 1.7 channel by electrophysiology [AID502582, Type: Literature] [gi:327478559]
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9
[SID103552460]
[CID24874869]
IC50 0.014Blockade of human Nav1.7 by FRET assay [AID308661, Type: Literature] [gi:327478559]
View
10
[SID104244978]
[CID11740023]
Ki 0.015Inhibition of human Nav 1.7 channel by electrophysiology [AID502582, Type: Literature] [gi:327478559]
View
11
[SID104244978]
[CID11740023]
IC50 0.015Blockade of human Nav1.7 by electrophysiology assay [AID502846, Type: Literature] [gi:327478559]
View
12
[SID103708253]
[CID44555497]
IC50 0.02Inhibition of human Nav1.7 channel expressed in HEK293 cells by FRET assay [AID446725, Type: Literature] [gi:327478559]
View
13
[SID104245218]
[CID10021733]
Ki 0.02Binding affinity to human Nav1.7 [AID502843, Type: Literature] [gi:327478559]
View
14
[SID131287358]
[CID12004377]
IC50 0.02Inhibition of human NaV1.7 expressed in HEK293 cells by [14C]guanidinium influx assay [AID599097, Type: Literature] [gi:327478559]
View
15
[SID160666878]
[CID70681064]
IC50 0.02Antagonist activity at human NaV1.7 channel by patchXpress assay [AID655060, Type: Literature] [gi:327478559]
View
16
[SID160677519]
[CID70685264]
IC50 0.02Antagonist activity at human NaV1.7 channel by patchXpress assay [AID655060, Type: Literature] [gi:327478559]
View
17
[SID160704372]
[CID70695782]
IC50 0.02Antagonist activity at human NaV1.7 channel by patchXpress assay [AID655060, Type: Literature] [gi:327478559]
View
18
[SID103554616]
[CID24875058]
IC50 0.022Inhibition of human sodium channel Nav1.7 by FRET assay [AID310071, Type: Literature] [gi:327478559]
View
19
[SID103552459]
[CID24874870]
IC50 0.023Blockade of human Nav1.7 by FRET assay [AID308661, Type: Literature] [gi:327478559]
View
20
[SID103561511]
[CID25031205]
IC50 0.025Inhibition of human Nav1.7 sodium channel expressed in HEK293 cells by FRET assay [AID314674, Type: Literature] [gi:327478559]
View
21
[SID163312954]
[CID71449283]
IC50 0.02512Inhibition of human Nav1.7 expressed in HEK293 cells by whole cell voltage-clamp electrophysiology assay [AID688712, Type: Literature] [gi:327478559]
View
22
[SID163326645]
[CID71456401]
IC50 0.02512Inhibition of human Nav1.7 expressed in HEK293 cells by whole cell voltage-clamp electrophysiology assay [AID688712, Type: Literature] [gi:327478559]
View
23
[SID163326658]
[CID71456413]
IC50 0.02512Inhibition of human Nav1.7 expressed in HEK293 cells by whole cell voltage-clamp electrophysiology assay [AID688712, Type: Literature] [gi:327478559]
View
24
[SID124968016]
[CID53322585]
IC50 0.029Inhibition of human Nav1.7 by VIPR assay [AID549473, Type: Literature] [gi:327478559]
View
25
[SID131277280]
[CID12004337]
IC50 0.03Inhibition of human NaV1.7 expressed in HEK293 cells by [14C]guanidinium influx assay [AID599097, Type: Literature] [gi:327478559]
View
26
[SID131273334]
[CID54580640]
IC50 0.03Inhibition of human NaV1.7 expressed in HEK293 cells by [14C]guanidinium influx assay [AID599097, Type: Literature] [gi:327478559]
View
27
[SID160672198]
[CID70683184]
IC50 0.03Antagonist activity at human NaV1.7 channel by patchXpress assay [AID655060, Type: Literature] [gi:327478559]
View
28
[SID160699035]
[CID70693674]
IC50 0.03Antagonist activity at human NaV1.7 channel by patchXpress assay [AID655060, Type: Literature] [gi:327478559]
View
29
[SID103561514]
[CID25033155]
IC50 0.03Inhibition of human Nav1.7 sodium channel expressed in HEK293 cells by FRET assay [AID314674, Type: Literature] [gi:327478559]
View
30
[SID103585628]
[CID11174599]
IC50 0.03Inhibition of voltage-gated Na channel 1.7 (unknown origin) [AID726285, Type: Literature] [gi:327478559]
View
31
[SID103554654]
[CID24896609]
IC50 0.03Inhibition of human sodium channel Nav1.7 by FRET assay [AID310071, Type: Literature] [gi:327478559]
View
32
[SID163316332]
[CID71451078]
IC50 0.03162Inhibition of human Nav1.7 expressed in HEK293 cells by whole cell voltage-clamp electrophysiology assay [AID688712, Type: Literature] [gi:327478559]
View
33
[SID163323259]
[CID71454670]
IC50 0.03162Inhibition of human Nav1.7 expressed in HEK293 cells by whole cell voltage-clamp electrophysiology assay [AID688712, Type: Literature] [gi:327478559]
View
34
[SID163326657]
[CID71456412]
IC50 0.03162Inhibition of human Nav1.7 expressed in HEK293 cells by whole cell voltage-clamp electrophysiology assay [AID688712, Type: Literature] [gi:327478559]
View
35
[SID103552466]
[CID24874959]
IC50 0.032Blockade of human Nav1.7 by FRET assay [AID308661, Type: Literature] [gi:327478559]
View
36
[SID103552469]
[CID44442675]
IC50 0.032Blockade of human Nav1.7 by FRET assay [AID308661, Type: Literature] [gi:327478559]
View
37
[SID103552468]
[CID23661730]
IC50 0.035Blockade of human Nav1.7 by FRET assay [AID308661, Type: Literature] [gi:327478559]
View
38
[SID103552468]
[CID23661730]
IC50 0.035Inhibition of human sodium channel Nav1.7 by FRET assay [AID310071, Type: Literature] [gi:327478559]
View
39
[SID103552468]
[CID23661730]
IC50 0.035Inhibition of human Nav1.7 sodium channel expressed in HEK293 cells by FRET assay [AID314674, Type: Literature] [gi:327478559]
View
40
[SID134459314]
[CID53361524]
Ki 0.035Binding affinity to inactivated human sodium channel Nav1.7 expressed in human HEK293 cells by patch-clamp electrophysiological assay [AID612078, Type: Literature] [gi:327478559]
View
41
[SID163323269]
[CID71454678]
IC50 0.03981Inhibition of human Nav1.7 expressed in HEK293 cells by whole cell voltage-clamp electrophysiology assay [AID688712, Type: Literature] [gi:327478559]
View
42
[SID163319807]
[CID71452899]
IC50 0.03981Inhibition of human Nav1.7 expressed in HEK293 cells by whole cell voltage-clamp electrophysiology assay [AID688712, Type: Literature] [gi:327478559]
View
43
[SID160704375]
[CID70695785]
IC50 0.04Antagonist activity at human NaV1.7 channel by patchXpress assay [AID655060, Type: Literature] [gi:327478559]
View
44
[SID160704370]
[CID70695780]
IC50 0.04Antagonist activity at human NaV1.7 channel by patchXpress assay [AID655060, Type: Literature] [gi:327478559]
View
45
[SID160699034]
[CID70693673]
IC50 0.04Antagonist activity at human NaV1.7 channel by patchXpress assay [AID655060, Type: Literature] [gi:327478559]
View
46
[SID160693646]
[CID70691577]
IC50 0.04Antagonist activity at human NaV1.7 channel by patchXpress assay [AID655060, Type: Literature] [gi:327478559]
View
47
[SID131275262]
[CID54581613]
IC50 0.04Inhibition of human NaV1.7 expressed in HEK293 cells by [14C]guanidinium influx assay [AID599097, Type: Literature] [gi:327478559]
View
48
[SID131281355]
[CID54584553]
IC50 0.04Inhibition of human NaV1.7 expressed in HEK293 cells by [14C]guanidinium influx assay [AID599097, Type: Literature] [gi:327478559]
View
49
[SID103552468]
[CID23661730]
Ki 0.04Binding affinity at human inactive state Nav1.7 by whole cell electrophysiology [AID308674, Type: Literature] [gi:327478559]
View
50
[SID104245212]
[CID49866117]
IC50 0.041Inhibition of human Nav 1.7 channel by voltage-ion-probe-reader [AID502584, Type: Literature] [gi:327478559]
View