Bookmark and Share
GABRA1 (geneid:2554) - Gene BioActivity Data
Also known as: ECA4, EIEE19, EJM, EJM5.
Filters: All Data » Active      
Filter selected
BioActivity Outcomes:
Active(734)
 
 
BioAssay Types:
Literature(708)
 
 
Confirmatory(15)
 
 
BioActivity Types:
Ki(480)
 
 
IC50(46)
 
 
EC50(29)
 
 
Substance Types:
Chemical(734)
 
 
Data download

Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 75    Data Row: 734   Total Pages: 37   Display: Page     
Sort: [Click the result table header to sort]
#StructureSubstanceCompoundActivityBioAssayTargetLinks
OutcomeTypeValue [μM]
1
[SID103484726]
[CID11646612]
Ki 0.0001Displacement of [3H]Ro-151788 from recombinant human GABA-Aalpha1 receptor plus beta3gamma2 [AID262644, Type: Literature] [gi:27808653]
View
2
[SID124968046]
[CID44466078]
Ki 0.00014Displacement of [3H]flumazenil human recombinant alpha1beta3gamma2 GABA(A) receptor expressed in HEK293 cells after 30 mins by glass fiber filtration assay [AID552801, Type: Literature] [gi:27808653]
View
3
[SID103479487]
[CID11524362]
Ki 0.00015Displacement of [3H]Ro 15-1788 from recombinant human GABAA alpha-1 receptor plus beta3gamma2 expressed in L(tk-) cells [AID260334, Type: Literature] [gi:27808653]
View
4
[SID103482895]
[CID44409159]
Ki 0.00016Displacement of [3H]Ro-151788 from human recombinant GABA-Aalpha1 receptor plus beta3gamma2 [AID262295, Type: Literature] [gi:27808653]
View
5
[SID103482437]
[CID10000391]
Ki 0.0002Displacement of [3H]Ro 15-1788 from human GABA-Aalpha1 receptor plus beta-3-gamma-2 expressed in mouse L(tk-) cells [AID262219, Type: Literature] [gi:27808653]
View
6
[SID103226602]
[CID44291154]
Ki 0.0002Displacement of [3H]Ro-151788 from human GABA-A receptor alpha-1-beta-3-gamma-2 subunits expressed in L(tk) cells [AID72914, Type: Literature] [gi:27808653]
View
7
[SID103513034]
[CID9799023]
Ki 0.00023Displacement of [3H]Ro 15-1788 from human recombinant GABAA alpha-1-beta-3-gamma-2 receptor expressed in L(tk-) cells [AID282665, Type: Literature] [gi:27808653]
View
8
[SID103479915]
[CID11611050]
Ki 0.00025Displacement of [3H]Ro 15-1788 from recombinant human GABAA alpha-1 receptor plus beta3gamma2 expressed in L(tk-) cells [AID260334, Type: Literature] [gi:27808653]
View
9
[SID103476287]
[CID9908684]
Ki 0.00026Displacement of [3H]-Ro15-1788 from human recombinant GABAA alpha1 in combination with beta-3-gamma-2 expressed in L(tk-) cells [AID259129, Type: Literature] [gi:27808653]
View
10
[SID103476287]
[CID9908684]
Ki 0.00027Displacement of [3H]Ro 15-1788 from human recombinant GABAA alpha-1-beta-3-gamma-2 receptor expressed in L(tk-) cells [AID282665, Type: Literature] [gi:27808653]
View
11
[SID103483578]
[CID11529633]
Ki 0.00027Displacement of [3H]Flumazenil from human GABA-Aalpha1 receptor plus beta-2-gamma-2 expressed in HEK293 cells [AID262560, Type: Literature] [gi:27808653]
View
12
[SID103483133]
[CID11501697]
Ki 0.00028Displacement of [3H]Ro-151788 from human recombinant GABA-Aalpha1 receptor plus beta3gamma2 [AID262295, Type: Literature] [gi:27808653]
View
13
[SID103340411]
[CID128064]
Ki 0.00029Inhibition of [3H]-Ro- 15-1788 binding to human GABA-A receptor alpha-1-beta-3-gamma-2 expressed in L(tk-) cells [AID254510, Type: Literature] [gi:27808653]
View
14
[SID103480930]
[CID9928025]
Ki 0.00031Displacement of [3H]Ro 15-1788 from recombinant human GABA-Aalpha1 receptor plus beta-3-gamma-2 expressed in L(tk-) cells [AID261197, Type: Literature] [gi:27808653]
View
15
[SID103480931]
[CID9945466]
Ki 0.00031Displacement of [3H]Ro 15-1788 from recombinant human GABA-Aalpha1 receptor plus beta-3-gamma-2 expressed in L(tk-) cells [AID261197, Type: Literature] [gi:27808653]
View
16
[SID103481016]
[CID10292263]
Ki 0.00036Displacement of [3H]Ro 15-1788 from recombinant human GABA-Aalpha1 receptor plus beta-3-gamma-2 expressed in L(tk-) cells [AID261197, Type: Literature] [gi:27808653]
View
17
[SID103513035]
[CID11631938]
Ki 0.00036Displacement of [3H]Ro 15-1788 from human recombinant GABAA alpha-1-beta-3-gamma-2 receptor expressed in L(tk-) cells [AID282665, Type: Literature] [gi:27808653]
View
18
[SID103513026]
[CID11675202]
Ki 0.00038Displacement of [3H]Ro 15-1788 from human recombinant GABAA alpha-1-beta-3-gamma-2 receptor expressed in L(tk-) cells [AID282665, Type: Literature] [gi:27808653]
View
19
[SID103491332]
[CID9865768]
Ki 0.00039Inhibition of [3H]Ro15-1788 binding to human recombinant GABA-Aalpha1 plus beta-3-gamma-2 receptor expressed in L(tk-) cells [AID267887, Type: Literature] [gi:27808653]
View
20
[SID103476516]
[CID9839679]
Ki 0.00039Displacement of [3H]-Ro15-1788 from human recombinant GABAA alpha1 in combination with beta-3-gamma-2 expressed in L(tk-) cells [AID259129, Type: Literature] [gi:27808653]
View