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GABRA1 (geneid:2554) - Gene BioActivity Data
Also known as: ECA4, EJM, EJM5.
Filters: All Data » Active      
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BioActivity Outcomes:
Active(683)
 
 
BioAssay Types:
Literature(636)
 
 
BioActivity Types:
Ki(465)
 
 
IC50(40)
 
 
EC50(29)
 
 
Substance Types:
Chemical(683)
 
 
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Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 71    Data Row: 683   Total Pages: 14   Display: Page     
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#StructureSubstanceCompoundActivityBioAssayTargetLinks
OutcomeTypeValue [μM]
1
[SID103484726]
[CID11646612]
Ki 0.0001Displacement of [3H]Ro-151788 from recombinant human GABA-Aalpha1 receptor plus beta3gamma2 [AID262644, Type: Literature] [gi:27808653]
View
2
[SID124968046]
[CID44466078]
Ki 0.00014Displacement of [3H]flumazenil human recombinant alpha1beta3gamma2 GABA(A) receptor expressed in HEK293 cells after 30 mins by glass fiber filtration assay [AID552801, Type: Literature] [gi:27808653]
View
3
[SID103479487]
[CID11524362]
Ki 0.00015Displacement of [3H]Ro 15-1788 from recombinant human GABAA alpha-1 receptor plus beta3gamma2 expressed in L(tk-) cells [AID260334, Type: Literature] [gi:27808653]
View
4
[SID103482895]
[CID44409159]
Ki 0.00016Displacement of [3H]Ro-151788 from human recombinant GABA-Aalpha1 receptor plus beta3gamma2 [AID262295, Type: Literature] [gi:27808653]
View
5
[SID103482437]
[CID10000391]
Ki 0.0002Displacement of [3H]Ro 15-1788 from human GABA-Aalpha1 receptor plus beta-3-gamma-2 expressed in mouse L(tk-) cells [AID262219, Type: Literature] [gi:27808653]
View
6
[SID103226602]
[CID44291154]
Ki 0.0002Displacement of [3H]Ro-151788 from human GABA-A receptor alpha-1-beta-3-gamma-2 subunits expressed in L(tk) cells [AID72914, Type: Literature] [gi:27808653]
View
7
[SID103513034]
[CID9799023]
Ki 0.00023Displacement of [3H]Ro 15-1788 from human recombinant GABAA alpha-1-beta-3-gamma-2 receptor expressed in L(tk-) cells [AID282665, Type: Literature] [gi:27808653]
View
8
[SID103479915]
[CID11611050]
Ki 0.00025Displacement of [3H]Ro 15-1788 from recombinant human GABAA alpha-1 receptor plus beta3gamma2 expressed in L(tk-) cells [AID260334, Type: Literature] [gi:27808653]
View
9
[SID103476287]
[CID9908684]
Ki 0.00026Displacement of [3H]-Ro15-1788 from human recombinant GABAA alpha1 in combination with beta-3-gamma-2 expressed in L(tk-) cells [AID259129, Type: Literature] [gi:27808653]
View
10
[SID103476287]
[CID9908684]
Ki 0.00027Displacement of [3H]Ro 15-1788 from human recombinant GABAA alpha-1-beta-3-gamma-2 receptor expressed in L(tk-) cells [AID282665, Type: Literature] [gi:27808653]
View
11
[SID103483578]
[CID11529633]
Ki 0.00027Displacement of [3H]Flumazenil from human GABA-Aalpha1 receptor plus beta-2-gamma-2 expressed in HEK293 cells [AID262560, Type: Literature] [gi:27808653]
View
12
[SID103483133]
[CID11501697]
Ki 0.00028Displacement of [3H]Ro-151788 from human recombinant GABA-Aalpha1 receptor plus beta3gamma2 [AID262295, Type: Literature] [gi:27808653]
View
13
[SID103340411]
[CID128064]
Ki 0.00029Inhibition of [3H]-Ro- 15-1788 binding to human GABA-A receptor alpha-1-beta-3-gamma-2 expressed in L(tk-) cells [AID254510, Type: Literature] [gi:27808653]
View
14
[SID103480930]
[CID9928025]
Ki 0.00031Displacement of [3H]Ro 15-1788 from recombinant human GABA-Aalpha1 receptor plus beta-3-gamma-2 expressed in L(tk-) cells [AID261197, Type: Literature] [gi:27808653]
View
15
[SID103480931]
[CID9945466]
Ki 0.00031Displacement of [3H]Ro 15-1788 from recombinant human GABA-Aalpha1 receptor plus beta-3-gamma-2 expressed in L(tk-) cells [AID261197, Type: Literature] [gi:27808653]
View
16
[SID103481016]
[CID10292263]
Ki 0.00036Displacement of [3H]Ro 15-1788 from recombinant human GABA-Aalpha1 receptor plus beta-3-gamma-2 expressed in L(tk-) cells [AID261197, Type: Literature] [gi:27808653]
View
17
[SID103513035]
[CID11631938]
Ki 0.00036Displacement of [3H]Ro 15-1788 from human recombinant GABAA alpha-1-beta-3-gamma-2 receptor expressed in L(tk-) cells [AID282665, Type: Literature] [gi:27808653]
View
18
[SID103513026]
[CID11675202]
Ki 0.00038Displacement of [3H]Ro 15-1788 from human recombinant GABAA alpha-1-beta-3-gamma-2 receptor expressed in L(tk-) cells [AID282665, Type: Literature] [gi:27808653]
View
19
[SID103491332]
[CID9865768]
Ki 0.00039Inhibition of [3H]Ro15-1788 binding to human recombinant GABA-Aalpha1 plus beta-3-gamma-2 receptor expressed in L(tk-) cells [AID267887, Type: Literature] [gi:27808653]
View
20
[SID103476516]
[CID9839679]
Ki 0.00039Displacement of [3H]-Ro15-1788 from human recombinant GABAA alpha1 in combination with beta-3-gamma-2 expressed in L(tk-) cells [AID259129, Type: Literature] [gi:27808653]
View
21
[SID103476516]
[CID9839679]
Ki 0.0004Displacement of [3H]Ro 15-1788 from recombinant human GABAA alpha-1 receptor plus beta3gamma2 expressed in L(tk-) cells [AID260334, Type: Literature] [gi:27808653]
View
22
[SID103484271]
[CID11632351]
Ki 0.0004Displacement of [3H]Ro-151788 from recombinant human GABA-Aalpha1 receptor plus beta3gamma2 [AID262644, Type: Literature] [gi:27808653]
View
23
[SID124965338]
[CID44466077]
Ki 0.00043Displacement of [3H]flumazenil human recombinant alpha1beta3gamma2 GABA(A) receptor expressed in HEK293 cells after 30 mins by glass fiber filtration assay [AID552801, Type: Literature] [gi:27808653]
View
24
[SID164147009]
[CID71584335]
Ki 0.00045Displacement of [3H]Ro15-1788 from recombinant GABA-A alpha1beta2gamma2 receptor benzodiazepine binding site (unknown origin) after 1 hr [AID739949, Type: Literature] [gi:27808653]
View
25
[SID103484354]
[CID11646630]
Ki 0.0005Displacement of [3H]Ro-151788 from recombinant human GABA-Aalpha1 receptor plus beta3gamma2 [AID262644, Type: Literature] [gi:27808653]
View
26
[SID103484270]
[CID11530663]
Ki 0.0005Displacement of [3H]Ro-151788 from recombinant human GABA-Aalpha1 receptor plus beta3gamma2 [AID262644, Type: Literature] [gi:27808653]
View
27
[SID103476533]
[CID9970131]
Ki 0.0005Displacement of [3H]-Ro15-1788 from human recombinant GABAA alpha1 in combination with beta-3-gamma-2 expressed in L(tk-) cells [AID259129, Type: Literature] [gi:27808653]
View
28
[SID103238503]
[CID11394173]
Ki 0.00051Binding affinity for human GABA-A receptor alpha-4-beta-3-gamma-2 subunits in L(tk-) cells [AID72467, Type: Literature] [gi:27808653]
View
29
[SID103482888]
[CID9841060]
Ki 0.00053Displacement of [3H]Ro-151788 from human recombinant GABA-Aalpha1 receptor plus beta3gamma2 [AID262295, Type: Literature] [gi:27808653]
View
30
[SID103482576]
[CID10154824]
Ki 0.00055Displacement of [3H]Ro 15-1788 from recombinant human GABA-Aalpha1 receptor plus beta3gamma2 expressed in mouse L(tk-) cells [AID262144, Type: Literature] [gi:27808653]
View
31
[SID103480016]
[CID9865233]
Ki 0.0006Displacement of [3H]Ro-151788 from human recombinant GABA-Aalpha1 receptor plus beta3gamma2 [AID262295, Type: Literature] [gi:27808653]
View
32
[SID103482601]
[CID44409020]
Ki 0.0006Displacement of [3H]Ro 15-1788 from recombinant human GABA-Aalpha1 receptor plus beta3gamma2 expressed in mouse L(tk-) cells [AID262144, Type: Literature] [gi:27808653]
View
33
[SID103476480]
[CID10200975]
Ki 0.00065Displacement of [3H]-Ro15-1788 from human recombinant GABAA alpha1 in combination with beta-3-gamma-2 expressed in L(tk-) cells [AID259129, Type: Literature] [gi:27808653]
View
34
[SID103476526]
[CID9925268]
Ki 0.00066Displacement of [3H]-Ro15-1788 from human recombinant GABAA alpha1 in combination with beta-3-gamma-2 expressed in L(tk-) cells [AID259129, Type: Literature] [gi:27808653]
View
35
[SID103476526]
[CID9925268]
Ki 0.00066Displacement of [3H]Ro 15-1788 from recombinant human GABA-Aalpha1 receptor plus beta-3-gamma-2 expressed in L(tk-) cells [AID261197, Type: Literature] [gi:27808653]
View
36
[SID103482813]
[CID10271398]
Ki 0.00067Displacement of [3H]Ro 15-1788 from recombinant human GABA-Aalpha1 receptor plus beta3gamma2 expressed in mouse L(tk-) cells [AID262144, Type: Literature] [gi:27808653]
View
37
[SID103482820]
[CID10292839]
Ki 0.00067Displacement of [3H]Ro 15-1788 from recombinant human GABA-Aalpha1 receptor plus beta3gamma2 expressed in mouse L(tk-) cells [AID262144, Type: Literature] [gi:27808653]
View
38
[SID103482232]
[CID10269219]
Ki 0.00068Displacement of [3H]Ro 15-1788 from recombinant human GABA-Aalpha1 receptor plus beta3gamma2 expressed in mouse L(tk-) cells [AID262144, Type: Literature] [gi:27808653]
View
39
[SID124973262]
[CID44466326]
Ki 0.00068Displacement of [3H]flumazenil human recombinant alpha1beta3gamma2 GABA(A) receptor expressed in HEK293 cells after 30 mins by glass fiber filtration assay [AID552801, Type: Literature] [gi:27808653]
View
40
[SID103482889]
[CID10406330]
Ki 0.0007Displacement of [3H]Ro-151788 from human recombinant GABA-Aalpha1 receptor plus beta3gamma2 [AID262295, Type: Literature] [gi:27808653]
View
41
[SID103482429]
[CID9969492]
Ki 0.00071Displacement of [3H]Ro 15-1788 from human GABA-Aalpha1 receptor plus beta-3-gamma-2 expressed in mouse L(tk-) cells [AID262219, Type: Literature] [gi:27808653]
View
42
[SID103585639]
[CID124514]
Ki 0.00072Displacement of [3H]flunitrazepam from human recombinant GABAA alpha-1-beta-3-gamma-2 receptor expressed in HEK cells by liquid scintillation counting [AID527597, Type: Literature] [gi:27808653]
View
43
[SID103480016]
[CID9865233]
Ki 0.00073Displacement of [3H]Ro 15-1788 from recombinant human GABAA alpha-1 receptor plus beta3gamma2 expressed in L(tk-) cells [AID260334, Type: Literature] [gi:27808653]
View
44
[SID103482819]
[CID10199394]
Ki 0.00076Displacement of [3H]Ro 15-1788 from recombinant human GABA-Aalpha1 receptor plus beta3gamma2 expressed in mouse L(tk-) cells [AID262144, Type: Literature] [gi:27808653]
View
45
[SID103513019]
[CID11574515]
Ki 0.00078Displacement of [3H]Ro 15-1788 from human recombinant GABAA alpha-1-beta-3-gamma-2 receptor expressed in L(tk-) cells [AID282665, Type: Literature] [gi:27808653]
View
46
[SID103484781]
[CID11717884]
Ki 0.0008Displacement of [3H]Ro-151788 from recombinant human GABA-Aalpha1 receptor plus beta3gamma2 [AID262644, Type: Literature] [gi:27808653]
View
47
[SID103482302]
[CID10270246]
Ki 0.0008Displacement of [3H]Ro 15-1788 from recombinant human GABA-Aalpha1 receptor plus beta3gamma2 expressed in mouse L(tk-) cells [AID262144, Type: Literature] [gi:27808653]
View
48
[SID103476224]
[CID9908880]
Ki 0.0008Displacement of [3H]-Ro15-1788 from human recombinant GABAA alpha1 in combination with beta-3-gamma-2 expressed in L(tk-) cells [AID259129, Type: Literature] [gi:27808653]
View
49
[SID103458752]
[CID6918583]
Ki 0.0008Positive allosteric modulation of GABAA alpha1 (unknown origin) [AID726242, Type: Literature] [gi:27808653]
View
50
[SID103164270]
[CID3373]
Ki 0.0008Binding affinity against alpha-1-beta-3-gamma-2 GABAA/BzR receptor subtype. [AID219794, Type: Literature] [gi:27808653]
View