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F2RL3 (geneid:9002) - Gene BioActivity Data
Also known as: PAR4.
BioActivity Outcomes:
Probe(2)
 
 
Active(16)
 
 
Inactive(188)
 
 
Unspecified(14)
 
 
BioAssay Types:
Confirmatory(201)
 
 
 
 
Literature(19)
 
 
 
 
BioActivity Types:
IC50(201)
 
 
 
 
Substance Types:
Chemical(213)
 
 
 
 
 
RNAi(7)
 
 
 
 
Data download

Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 14    Data Row: 220   Total Pages: 5   Display: Page     
Sort: [Click the result table header to sort]
#StructureSubstanceCompoundActivityBioAssayTargetLinks
OutcomeTypeValue [μM]
1
[SID144241412]
[CID60210843]
Average_IC50_uM 0.139Discovery of Novel Antagonists of Protease activated receptor 4: CRC Assay [AID652253, Type: confirmatory] [gi:89353783]
View
2
[SID161004645]
[CID752812]
IC50_uM 0.139Discovery of Novel Antagonists of Protease activated receptor 4: Single Point [AID652250, Type: confirmatory] [gi:89353783]
View
3
[SID161780288]
[CID71148612]
IC50_uM 0.83Discovery of Novel Antagonists of Protease activated receptor 4: Single Point [AID652250, Type: confirmatory] [gi:89353783]
View
4
[SID161780288]
[CID71148612]
Average_IC50_uM 0.83Discovery of Novel Antagonists of Protease activated receptor 4: CRC Assay [AID652253, Type: confirmatory] [gi:89353783]
View
5
[SID160870425]
[CID70702166]
IC50_uM 3.13Discovery of Novel Antagonists of Protease activated receptor 4: Single Point [AID652250, Type: confirmatory] [gi:89353783]
View
6
[SID160870447]
[CID70702182]
IC50_uM 3.85Discovery of Novel Antagonists of Protease activated receptor 4: Single Point [AID652250, Type: confirmatory] [gi:89353783]
View
7
[SID160870446]
[CID70702192]
IC50_uM 5.27Discovery of Novel Antagonists of Protease activated receptor 4: Single Point [AID652250, Type: confirmatory] [gi:89353783]
View
8
[SID152145946]
[CID66552991]
IC50_uM 5.4Discovery of Novel Antagonists of Protease activated receptor 4: Single Point [AID652250, Type: confirmatory] [gi:89353783]
View
9
[SID152145949]
[CID66552993]
IC50_uM 10Discovery of Novel Antagonists of Protease activated receptor 4: Single Point [AID652250, Type: confirmatory] [gi:89353783]
View
10
[SID152145947]
[CID66552992]
IC50_uM 10Discovery of Novel Antagonists of Protease activated receptor 4: Single Point [AID652250, Type: confirmatory] [gi:89353783]
View
11
[SID160870443]
[CID70702170]
IC50_uM 10Discovery of Novel Antagonists of Protease activated receptor 4: Single Point [AID652250, Type: confirmatory] [gi:89353783]
View
12
[SID160870449]
[CID70702172]
IC50_uM 14.6Discovery of Novel Antagonists of Protease activated receptor 4: Single Point [AID652250, Type: confirmatory] [gi:89353783]
View
13
[SID160721261]
Genome-wide high-content siRNA screens for regulators of Parkin translocation in selective mitophagy (Ambion Library) [AID651811, Type: Literature] [geneid:9002]
View
14
[SID160724205]
Genome-wide high-content siRNA screens for regulators of Parkin translocation in selective mitophagy (Ambion Library) [AID651811, Type: Literature] [geneid:9002]
View
15
[SID161004552]
[CID1150319]
IC50_uM Discovery of Novel Antagonists of Protease activated receptor 4: Single Point [AID652250, Type: confirmatory] [gi:89353783]
View
16
[SID161004578]
[CID4342667]
IC50_uM Discovery of Novel Antagonists of Protease activated receptor 4: Single Point [AID652250, Type: confirmatory] [gi:89353783]
View
17
[SID161004647]
[CID987967]
IC50_uM Discovery of Novel Antagonists of Protease activated receptor 4: Single Point [AID652250, Type: confirmatory] [gi:89353783]
View
18
[SID161004613]
[CID6603619]
IC50_uM Discovery of Novel Antagonists of Protease activated receptor 4: Single Point [AID652250, Type: confirmatory] [gi:89353783]
View
19
[SID85104896]
siRNA Circadian Assay [AID1904, Type: Literature] [geneid:9002]
View
20
[SID85112119]
siRNA Circadian Assay [AID1904, Type: Literature] [geneid:9002]
View
21
[SID103353632]
[CID10132921]
Inhibition of PAR4-mediated GYPGKF-induced ATP release in human platelet assessed per 3*10^8 platelets at 0.2 uM [AID323470, Type: Literature] [gi:116242700]
View
22
[SID103353632]
[CID10132921]
Inhibition of PAR4-mediated GYPGKF-induced ATP release in human platelet assessed per 3*10^8 platelets at 0.1 uM [AID323471, Type: Literature] [gi:116242700]
View
23
[SID103353632]
[CID10132921]
Inhibition of PAR4-mediated GYPGKF-induced P-selectin expression in human platelet at 0.1 uM [AID323474, Type: Literature] [gi:116242700]
View
24
[SID103353632]
[CID10132921]
Inhibition of PAR4-mediated GYPGKF-induced P-selectin expression in human platelet at 0.05 uM [AID323475, Type: Literature] [gi:116242700]
View
25
[SID103568898]
[CID9967881]
Inhibition of PAR4-mediated GYPGKF-induced ATP release in human platelet assessed per 3*10^8 platelets at 5 uM [AID323473, Type: Literature] [gi:116242700]
View
26
[SID103568898]
[CID9967881]
Inhibition of PAR4-mediated GYPGKF-induced P-selectin expression in human platelet at 5 uM [AID323477, Type: Literature] [gi:116242700]
View
27
[SID103569233]
[CID24873525]
Inhibition of PAR4-mediated GYPGKF-induced ATP release in human platelet assessed per 3*10^8 platelets at 0.2 uM [AID323470, Type: Literature] [gi:116242700]
View
28
[SID103569233]
[CID24873525]
Inhibition of PAR4-mediated GYPGKF-induced ATP release in human platelet assessed per 3*10^8 platelets at 0.1 uM [AID323471, Type: Literature] [gi:116242700]
View
29
[SID103569233]
[CID24873525]
Inhibition of PAR4-mediated GYPGKF-induced P-selectin expression in human platelet at 0.1 uM [AID323474, Type: Literature] [gi:116242700]
View
30
[SID103569233]
[CID24873525]
Inhibition of PAR4-mediated GYPGKF-induced P-selectin expression in human platelet at 0.05 uM [AID323475, Type: Literature] [gi:116242700]
View
31
[SID103569372]
[CID44451921]
Inhibition of PAR4-mediated GYPGKF-induced ATP release in human platelet assessed per 3*10^8 platelets at 1 uM [AID323472, Type: Literature] [gi:116242700]
View
32
[SID103569372]
[CID44451921]
Inhibition of PAR4-mediated GYPGKF-induced P-selectin expression in human platelet at 1 uM [AID323476, Type: Literature] [gi:116242700]
View
33
[SID160870425]
[CID70702166]
Average_IC50_uM 3.13Discovery of Novel Antagonists of Protease activated receptor 4: CRC Assay [AID652253, Type: confirmatory] [gi:89353783]
View
34
[SID160870447]
[CID70702182]
Average_IC50_uM 3.85Discovery of Novel Antagonists of Protease activated receptor 4: CRC Assay [AID652253, Type: confirmatory] [gi:89353783]
View
35
[SID160870446]
[CID70702192]
Average_IC50_uM 5.27Discovery of Novel Antagonists of Protease activated receptor 4: CRC Assay [AID652253, Type: confirmatory] [gi:89353783]
View
36
[SID152145946]
[CID66552991]
Average_IC50_uM 5.4Discovery of Novel Antagonists of Protease activated receptor 4: CRC Assay [AID652253, Type: confirmatory] [gi:89353783]
View
37
[SID160870448]
[CID70702186]
Average_IC50_uM 14.6Discovery of Novel Antagonists of Protease activated receptor 4: CRC Assay [AID652253, Type: confirmatory] [gi:89353783]
View
38
[SID161004646]
[CID5098252]
IC50_uM Discovery of Novel Antagonists of Protease activated receptor 4: Single Point [AID652250, Type: confirmatory] [gi:89353783]
View
39
[SID161004648]
[CID3956524]
IC50_uM Discovery of Novel Antagonists of Protease activated receptor 4: Single Point [AID652250, Type: confirmatory] [gi:89353783]
View
40
[SID161004649]
[CID4637020]
IC50_uM Discovery of Novel Antagonists of Protease activated receptor 4: Single Point [AID652250, Type: confirmatory] [gi:89353783]
View
41
[SID161004650]
[CID2921458]
IC50_uM Discovery of Novel Antagonists of Protease activated receptor 4: Single Point [AID652250, Type: confirmatory] [gi:89353783]
View
42
[SID161004651]
[CID15997028]
IC50_uM Discovery of Novel Antagonists of Protease activated receptor 4: Single Point [AID652250, Type: confirmatory] [gi:89353783]
View
43
[SID161004652]
[CID15987694]
IC50_uM Discovery of Novel Antagonists of Protease activated receptor 4: Single Point [AID652250, Type: confirmatory] [gi:89353783]
View
44
[SID161004653]
[CID15997031]
IC50_uM Discovery of Novel Antagonists of Protease activated receptor 4: Single Point [AID652250, Type: confirmatory] [gi:89353783]
View
45
[SID161004654]
[CID16000499]
IC50_uM Discovery of Novel Antagonists of Protease activated receptor 4: Single Point [AID652250, Type: confirmatory] [gi:89353783]
View
46
[SID161004655]
[CID752157]
IC50_uM Discovery of Novel Antagonists of Protease activated receptor 4: Single Point [AID652250, Type: confirmatory] [gi:89353783]
View
47
[SID161004656]
[CID2056642]
IC50_uM Discovery of Novel Antagonists of Protease activated receptor 4: Single Point [AID652250, Type: confirmatory] [gi:89353783]
View
48
[SID161004657]
[CID4230002]
IC50_uM Discovery of Novel Antagonists of Protease activated receptor 4: Single Point [AID652250, Type: confirmatory] [gi:89353783]
View
49
[SID161004658]
[CID4610922]
IC50_uM Discovery of Novel Antagonists of Protease activated receptor 4: Single Point [AID652250, Type: confirmatory] [gi:89353783]
View
50
[SID161004659]
[CID4523395]
IC50_uM Discovery of Novel Antagonists of Protease activated receptor 4: Single Point [AID652250, Type: confirmatory] [gi:89353783]
View