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TRPM2 (geneid:7226) - Gene BioActivity Data
Also known as: EREG1, KNP3, LTRPC2, NUDT9H, NUDT9L1, TRPC7.
BioActivity Outcomes:
Active(5)
 
 
Inactive(19)
 
 
Unspecified(8)
 
 
BioAssay Types:
Literature(20)
 
 
 
 
Screening(10)
 
 
BioActivity Types:
IC50(11)
 
 
 
Substance Types:
Chemical(21)
 
 
 
 
RNAi(11)
 
 
 
Data download

Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 16    Data Row: 32   Total Pages: 2   Display: Page     
Sort: [Click the result table header to sort]
#StructureSubstanceCompoundActivityBioAssayTargetLinks
OutcomeTypeValue [μM]
1
[SID103424618]
[CID1598]
IC50 1Inhibition of human TRPM2 expressed in HEK293 cells [AID1065919, Type: Literature] [gi:160381681]
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2
[SID103430866]
[CID5353376]
IC50 1.7Inhibition of human TRPM2 expressed in HEK293 cells assessed as inhibition of H2O2-induced intracellular calcium level by patch clamp technique [AID1065920, Type: Literature] [gi:160381681]
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3
[SID103244070]
IC50 2.6Inhibition of TRPM2 (unknown origin) expressed in HEK293 cells assessed as inhibition of ADP-ribose-induced current by patch clamp technique [AID1065918, Type: Literature] [gi:160381681]
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4
[SID103176241]
[CID2812]
IC50 3Inhibition of TRPM2 (unknown origin) [AID1065914, Type: Literature] [gi:160381681]
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5
[SID103212333]
[CID3198]
IC50 3Inhibition of TRPM2 (unknown origin) [AID1065914, Type: Literature] [gi:160381681]
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6
[SID103201463]
[CID6083]
IC50 70Inhibition of TRPM2 (unknown origin) [AID1065914, Type: Literature] [gi:160381681]
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7
[SID103191339]
[CID3371]
IC50 70Inhibition of human recombinant TRPM2 [AID1065922, Type: Literature] [gi:160381681]
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8
[SID103191721]
[CID85472]
IC50 76Inhibition of human TRPM2 expressed in HEK293 cells assessed as inhibition of ADP-ribose-induced current by patch clamp electrophysiology [AID1065921, Type: Literature] [gi:160381681]
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9
[SID103476697]
[CID636430]
IC50 100Antagonist activity at human TRPM2 expressed in HEK293 cells assessed as inhibition of ADPR-induced maximum outward potassium current at +15 mV by whole-cell patch-clamp electrophysiology [AID1065917, Type: Literature] [gi:160381681]
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10
[SID103191448]
[CID4044]
IC50 124Inhibition of human recombinant TRPM2 [AID1065922, Type: Literature] [gi:160381681]
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11
[SID103253261]
[CID4488]
IC50 149Inhibition of human recombinant TRPM2 [AID1065922, Type: Literature] [gi:160381681]
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12
[SID85101237]
siRNA Circadian Assay [AID1904, Type: other] [geneid:7226]
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13
[SID85108460]
siRNA Circadian Assay [AID1904, Type: other] [geneid:7226]
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14
[SID87692368]
[CID776924]
Late stage counterscreen results from the probe development effort to identify selective agonists of the Transient Receptor Potential Channels 3 (TRPML3): other ion channel Fura-2 profiling assay [AID2770, Type: screening] [gi:4507689]
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15
[SID87692368]
[CID776924]
Late stage counterscreen results from the probe development effort to identify selective agonists of the Transient Receptor Potential Channels 3 (TRPML3): other ion channel Fura-2 profiling assay [AID2770_5, Type: screening] [gi:4507689]
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16
[SID87692370]
[CID801435]
Late stage counterscreen results from the probe development effort to identify selective agonists of the Transient Receptor Potential Channels 3 (TRPML3): other ion channel Fura-2 profiling assay [AID2770, Type: screening] [gi:4507689]
View
17
[SID87692370]
[CID801435]
Late stage counterscreen results from the probe development effort to identify selective agonists of the Transient Receptor Potential Channels 3 (TRPML3): other ion channel Fura-2 profiling assay [AID2770_5, Type: screening] [gi:4507689]
View
18
[SID87692372]
[CID2745583]
Late stage counterscreen results from the probe development effort to identify selective agonists of the Transient Receptor Potential Channels 3 (TRPML3): other ion channel Fura-2 profiling assay [AID2770, Type: screening] [gi:4507689]
View
19
[SID87692372]
[CID2745583]
Late stage counterscreen results from the probe development effort to identify selective agonists of the Transient Receptor Potential Channels 3 (TRPML3): other ion channel Fura-2 profiling assay [AID2770_5, Type: screening] [gi:4507689]
View
20
[SID134310306]
An siRNA screen for human genes that are involved in human papilloma virus (HPV) E2 transcriptional repression of the E6 and E7 oncogenes [AID624099, Type: Literature] [geneid:7226]
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