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PRKACA (geneid:5566) - Gene BioActivity Data
Also known as: PKACA.
BioActivity Outcomes:
Active(642)
 
 
Inactive(65670)
 
 
Inconclusive(20)
 
 
Unspecified(1353)
 
 
BioAssay Types:
Screening(64926)
 
 
 
Literature(1486)
 
 
 
 
 
Confirmatory(211)
 
 
 
 
BioActivity Types:
AC50(111)
 
 
 
 
Kd(110)
 
 
 
IC50(77)
 
 
 
 
Ki(20)
 
 
 
Substance Types:
Chemical(67676)
 
 
 
 
 
RNAi(9)
 
 
 
 
Data download

Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 82    Data Row: 67685   Total Pages: 1354   Display: Page     
Sort: [Click the result table header to sort]
#StructureSubstanceCompoundActivityBioAssayTargetLinks
OutcomeTypeValue [μM]
1
[SID103469179]
[CID44403669]
Ki 0.0034Inhibitory constant against the protein kinase A [AID254305, Type: Literature] [gi:125205]
View
2
[SID103469178]
[CID5327966]
Ki 0.0039Inhibitory constant against the protein kinase A [AID254305, Type: Literature] [gi:125205]
View
3
[SID103252142]
[CID5287736]
Ki 0.0047Inhibitory constant against the protein kinase A [AID254305, Type: Literature] [gi:125205]
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4
[SID103520504]
[CID16732279]
IC50 0.005Inhibition of PKA [AID290880, Type: Literature] [gi:125205]
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5
[SID104543587]
[CID44537813]
AC50_uM 0.005Protein Kinase A Activity Assay Measured in Biochemical System Using Plate Reader - 2052-04_Inhibitor_Dose_DryPowder_Activity [AID504583, Type: confirmatory] [gi:4506055]
View
6
[SID103517955]
[CID23647431]
IC50 0.0068Inhibition of PKA [AID287580, Type: Literature] [gi:125205]
View
7
[SID103520531]
[CID16731841]
IC50 0.007Inhibition of PKA [AID290880, Type: Literature] [gi:125205]
View
8
[SID103520457]
[CID16732881]
IC50 0.009Inhibition of PKA [AID290880, Type: Literature] [gi:125205]
View
9
[SID103520530]
[CID11327794]
IC50 0.013Inhibition of PKA [AID290880, Type: Literature] [gi:125205]
View
10
[SID103520529]
[CID16732276]
IC50 0.015Inhibition of PKA [AID290880, Type: Literature] [gi:125205]
View
11
[SID103517961]
[CID23647380]
IC50 0.015Inhibition of PKA [AID287580, Type: Literature] [gi:125205]
View
12
[SID103516311]
[CID44422924]
IC50 0.015Inhibition of PKA by radiometric filter binding assay [AID286920, Type: Literature] [gi:125205]
View
13
[SID103517956]
[CID23647432]
IC50 0.016Inhibition of PKA [AID287580, Type: Literature] [gi:125205]
View
14
[SID103491101]
[CID11314340]
Ki 0.016Inhibition of PKA [AID266592, Type: Literature] [gi:125205]
View
15
[SID103517954]
[CID10126464]
IC50 0.018Inhibition of PKA [AID287580, Type: Literature] [gi:125205]
View
16
[SID103243222]
[CID44299148]
Kd 0.019Binding constant for PKAC-alpha kinase domain [AID624881, Type: Literature] [gi:125205]
View
17
[SID103604655]
[CID16725726]
Kd 0.019Binding constant for PKAC-alpha kinase domain [AID624881, Type: Literature] [gi:125205]
View
18
[SID103243222]
[CID44299148]
IC50 0.019Inhibition of human neutrophil protein kinase A (PKA) [AID164478, Type: Literature] [gi:125205]
View
19
[SID103243222]
[CID44299148]
Kd 0.019Binding constant for PKAC-alpha kinase domain [AID435932, Type: Literature] [gi:125205]
View
20
[SID103436463]
[CID44386181]
IC50 0.03Inhibition of cAMP-dependent protein kinase (PKA) [AID155687, Type: other] [gi:125205]
View
21
[SID103517963]
[CID23647437]
IC50 0.032Inhibition of PKA [AID287580, Type: Literature] [gi:125205]
View
22
[SID103517966]
[CID23647440]
IC50 0.032Inhibition of PKA [AID287580, Type: Literature] [gi:125205]
View
23
[SID103516318]
[CID16122633]
IC50 0.033Inhibition of PKA by radiometric filter binding assay [AID286920, Type: Literature] [gi:125205]
View
24
[SID103517964]
[CID23647438]
IC50 0.046Inhibition of PKA [AID287580, Type: Literature] [gi:125205]
View
25
[SID103491101]
[CID11314340]
Kd 0.056Binding constant for PKAC-alpha kinase domain [AID624881, Type: Literature] [gi:125205]
View
26
[SID103517959]
[CID23647435]
IC50 0.058Inhibition of PKA [AID287580, Type: Literature] [gi:125205]
View
27
[SID103437288]
[CID44386587]
IC50 0.07Inhibition of cAMP-dependent protein kinase (PKA) [AID155687, Type: other] [gi:125205]
View
28
[SID103516244]
[CID9837177]
IC50 0.073Inhibition of PKA by radiometric filter binding assay [AID286920, Type: Literature] [gi:125205]
View
29
[SID103520528]
[CID16731838]
IC50 0.078Inhibition of PKA [AID290880, Type: Literature] [gi:125205]
View
30
[SID103267632]
[CID44310732]
IC50 0.08Inhibition of cAMP-dependent protein kinase (Protein kinase A) [AID164477, Type: other] [gi:125205]
View
31
[SID103517960]
[CID16040274]
IC50 0.11Inhibition of PKA [AID287580, Type: Literature] [gi:125205]
View
32
[SID125299371]
[CID44259]
AC50_uM 0.126Protein Kinase A Activity Assay Measured in Biochemical System Using Plate Reader - 2052-04_Inhibitor_Dose_DryPowder_Activity_Set2 [AID588629, Type: confirmatory] [gi:4506055]
View
33
[SID103516252]
[CID5327109]
IC50 0.17Inhibition of PKA by radiometric filter binding assay [AID286920, Type: Literature] [gi:125205]
View
34
[SID164133368]
[CID71717270]
Kd 0.22Binding constant for PKAC-alpha kinase domain [AID624881, Type: Literature] [gi:125205]
View
35
[SID103517967]
[CID23647441]
IC50 0.274Inhibition of PKA [AID287580, Type: Literature] [gi:125205]
View
36
[SID103240316]
[CID176167]
Kd 0.33Binding constant for PKAC-alpha kinase domain [AID624881, Type: Literature] [gi:125205]
View
37
[SID103567619]
[CID448043]
Ki 0.34Inhibitory constant against PKA [AID435508, Type: Literature] [gi:125205]
View
38
[SID103517969]
[CID23647443]
IC50 0.371Inhibition of PKA [AID287580, Type: Literature] [gi:125205]
View
39
[SID103210437]
[CID3547]
Ki 0.46Inhibitory constant against PKA [AID435508, Type: Literature] [gi:125205]
View
40
[SID103694299]
[CID5154691]
IC50 0.5Inhibition of PKA in the presence of 20uM ATP [AID435212, Type: Literature] [gi:125205]
View
41
[SID103596121]
[CID11213558]
Kd 0.6Binding constant for PKAC-alpha kinase domain [AID624881, Type: Literature] [gi:125205]
View
42
[SID103516289]
[CID11695362]
IC50 0.61Inhibition of PKA by radiometric filter binding assay [AID286920, Type: Literature] [gi:125205]
View
43
[SID164144585]
[CID71719722]
Kd 0.72Binding constant for PKAC-alpha kinase domain [AID435932, Type: Literature] [gi:125205]
View
44
[SID164144585]
[CID71719722]
Kd 0.72Binding constant for PKAC-alpha kinase domain [AID624881, Type: Literature] [gi:125205]
View
45
[SID103232855]
[CID2290]
IC50 0.79Inhibition of cAMP-dependent protein kinase (Protein kinase A) [AID164477, Type: other] [gi:125205]
View
46
[SID92708292]
[CID3547]
AC50_uM 0.837Protein Kinase A Activity Assay Measured in Biochemical System Using Plate Reader - 2052-04_Inhibitor_Dose_DryPowder_Activity_Set2 [AID588629, Type: confirmatory] [gi:4506055]
View
47
[SID99351052]
[CID6489264]
AC50_uM 1.115Protein Kinase A Activity Assay Measured in Biochemical System Using Plate Reader - 2052-04_Inhibitor_Dose_DryPowder_Activity [AID504583, Type: confirmatory] [gi:4506055]
View
48
[SID103313081]
[CID2404]
IC50 1.2Inhibition of human neutrophil protein kinase A (PKA) [AID164478, Type: Literature] [gi:125205]
View
49
[SID92708292]
[CID3547]
AC50_uM 1.558Protein Kinase A Activity Assay Measured in Biochemical System Using Plate Reader - 2052-04_Inhibitor_Dose_DryPowder_Activity [AID504583, Type: confirmatory] [gi:4506055]
View
50
[SID103181324]
[CID5353940]
Kd 1.7Binding constant for PKAC-alpha kinase domain [AID435932, Type: Literature] [gi:125205]
View