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PPARD (geneid:5467) - Gene BioActivity Data
Also known as: FAAR, NR1C2, NUC1, NUCI, NUCII, PPARB.
BioActivity Outcomes:
Active(1800)
 
 
Inactive(35566)
 
 
Inconclusive(7359)
 
 
Unspecified(1015)
 
 
BioAssay Types:
Confirmatory(24408)
 
 
 
 
 
Summary(18610)
 
 
 
 
Literature(2701)
 
 
 
 
 
Screening(18)
 
 
 
BioActivity Types:
Potency(33631)
 
 
 
 
EC50(1329)
 
 
 
 
 
IC50(477)
 
 
 
 
 
Ki(30)
 
 
 
Kd(12)
 
 
 
Substance Types:
Chemical(45729)
 
 
 
 
 
RNAi(11)
 
 
 
Data download

Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 243    Data Row: 45740   Total Pages: 2287   Display: Page     
Sort: [Click the result table header to sort]
#StructureSubstanceCompoundActivityBioAssayTargetLinks
OutcomeTypeValue [μM]
1
[SID103522681]
[CID16726113]
EC50 3e-05Agonist activity at human PPARdelta receptor by cell based transactivation assay [AID290903, Type: Literature] [gi:417522]
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2
[SID103522679]
[CID11418941]
EC50 6e-05Agonist activity at human PPARdelta receptor by cell based transactivation assay [AID290903, Type: Literature] [gi:417522]
View
3
[SID103215363]
[CID9934458]
Kd 0.0004Binding affinity to human PPARdelta (unknown origin) by competitive TR-FRET assay [AID731520, Type: Literature] [gi:417522]
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4
[SID124969632]
[CID50942698]
EC50 0.0005Agonist activity at Gal4-fused human PPARdelta DNA binding domain expressed in HEK293 cells by luciferase reporter gene assay [AID551019, Type: Literature] [gi:417522]
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5
[SID103508878]
[CID16110483]
EC50 0.00058Agonist activity at human PPAR delta by FRET assay [AID279989, Type: Literature] [gi:417522]
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6
[SID103635314]
[CID44143330]
Ki 0.0006Displacement of [3H]GW2433 from human PPARdelta receptor by scintillation proximity assay [AID375472, Type: Literature] [gi:417522]
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7
[SID103519494]
[CID16220190]
EC50 0.00072Transactivation of Gal4-fused human PPARdelta expressed in HEK293 cells after 16 to 20 hrs by luciferase reporter gene assay [AID554247, Type: Literature] [gi:417522]
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8
[SID103766417]
[CID11620299]
EC50 0.0009Agonist activity at human PPAR-delta expressed in african green monkey CV-1 cells after 24 hrs by luciferase reporter gene assay [AID547900, Type: Literature] [gi:417522]
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9
[SID103519494]
[CID16220190]
EC50 0.00091Effect on PPARdelta transactivation activity in HEK293 cells [AID288974, Type: Literature] [gi:417522]
View
10
[SID103508871]
[CID16110444]
EC50 0.00095Agonist activity at human PPAR delta by FRET assay [AID279989, Type: Literature] [gi:417522]
View
11
[SID103215363]
[CID9934458]
EC50 0.001Maximum transcriptional activation of human PPAR delta receptor [AID156617, Type: Literature] [gi:417522]
View
12
[SID103215363]
[CID9934458]
IC50 0.001Binding affinity for human PPAR delta receptor [AID156625, Type: Literature] [gi:417522]
View
13
[SID103215364]
[CID9803963]
EC50 0.001Maximum transcriptional activation of human PPAR delta receptor [AID156617, Type: Literature] [gi:417522]
View
14
[SID103215364]
[CID9803963]
IC50 0.001Binding affinity for human PPAR delta receptor [AID156625, Type: Literature] [gi:417522]
View
15
[SID144212728]
[CID9934458]
Ratio Potency (uM) 0.001qHTS assay to identify small molecule agonists of the peroxisome proliferator-activated receptor delta (PPARd) signaling pathway: Summary [AID743227, Type: summary] [gi:216409690]
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16
[SID103736027]
[CID44627948]
EC50 0.001Agonist activity at human PPARdelta ligand binding domain expressed in human 293T cells co-transfected with Gal4-DBD by luciferase transactivation assay [AID469785, Type: Literature] [gi:417522]
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17
[SID103736415]
[CID16722365]
EC50 0.001Agonist activity at human PPARdelta ligand binding domain expressed in human 293T cells co-transfected with Gal4-DBD by luciferase transactivation assay [AID469785, Type: Literature] [gi:417522]
View
18
[SID103736417]
[CID44627529]
EC50 0.001Agonist activity at human PPARdelta ligand binding domain expressed in human 293T cells co-transfected with Gal4-DBD by luciferase transactivation assay [AID469785, Type: Literature] [gi:417522]
View
19
[SID160689487]
[CID60166650]
EC50 0.001Transactivation activity at human PPARdelta expressed in african green monkey CV1 cells after 24 hrs by luciferase reporter gene assay [AID663629, Type: Literature] [gi:417522]
View
20
[SID124957999]
[CID50925503]
EC50 0.001Agonist activity at human PPAR-delta expressed in african green monkey CV-1 cells after 24 hrs by luciferase reporter gene assay [AID547900, Type: Literature] [gi:417522]
View