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PPARA (geneid:5465) - Gene BioActivity Data
Also known as: SC22CB-5E3.5, NR1C1, PPAR, PPARalpha, hPPAR.
BioActivity Outcomes:
Active(2446)
 
 
Inactive(3088)
 
 
Inconclusive(201)
 
 
Unspecified(1741)
 
 
BioAssay Types:
Literature(4395)
 
 
 
 
 
Confirmatory(3055)
 
 
 
 
 
Screening(18)
 
 
 
BioActivity Types:
Potency(2864)
 
 
 
 
EC50(2353)
 
 
 
 
 
IC50(781)
 
 
 
 
 
Ki(60)
 
 
 
 
 
Kd(17)
 
 
 
Substance Types:
Chemical(7464)
 
 
 
 
 
RNAi(12)
 
 
 
Data download

Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 426    Data Row: 7476   Total Pages: 374   Display: Page     
Sort: [Click the result table header to sort]
#StructureSubstanceCompoundActivityBioAssayTargetLinks
OutcomeTypeValue [μM]
1
[SID103283308]
[CID10004270]
EC50 2e-11Transactivation of GAL4-fused Homo sapiens (human) PPARalpha/PPARgamma DNA binding domain expressed in African green monkey CV1 cells by luciferase reporter gene assay [AID1105617, Type: confirmatory] [gi:3041727]
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2
[SID103282873]
[CID9890585]
EC50 4e-11Transactivation of GAL4-fused Homo sapiens (human) PPARalpha/PPARgamma DNA binding domain expressed in African green monkey CV1 cells by luciferase reporter gene assay [AID1105617, Type: confirmatory] [gi:3041727]
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3
[SID194136726]
[CID76309038]
EC50 1.1e-10Transactivation of GAL4-fused Homo sapiens (human) PPARalpha/PPARgamma DNA binding domain expressed in African green monkey CV1 cells by luciferase reporter gene assay [AID1105617, Type: confirmatory] [gi:3041727]
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4
[SID194143594]
[CID76312721]
EC50 1.6e-10Transactivation of GAL4-fused Homo sapiens (human) PPARalpha/PPARgamma DNA binding domain expressed in African green monkey CV1 cells by luciferase reporter gene assay [AID1105617, Type: confirmatory] [gi:3041727]
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5
[SID194178084]
[CID76330830]
EC50 2.51e-09Transactivation of GAL4-fused Homo sapiens (human) PPARalpha/PPARgamma DNA binding domain expressed in African green monkey CV1 cells by luciferase reporter gene assay [AID1105617, Type: confirmatory] [gi:3041727]
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6
[SID194143593]
[CID76312720]
EC50 8.32e-09Transactivation of GAL4-fused Homo sapiens (human) PPARalpha/PPARgamma DNA binding domain expressed in African green monkey CV1 cells by luciferase reporter gene assay [AID1105617, Type: confirmatory] [gi:3041727]
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7
[SID103422205]
[CID11049998]
EC50 9.77e-09Transactivation of GAL4-fused Homo sapiens (human) PPARalpha/PPARgamma DNA binding domain expressed in African green monkey CV1 cells by luciferase reporter gene assay [AID1105617, Type: confirmatory] [gi:3041727]
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8
[SID194184892]
[CID76334424]
EC50 1.7e-08Transactivation of GAL4-fused Homo sapiens (human) PPARalpha/PPARgamma DNA binding domain expressed in African green monkey CV1 cells by luciferase reporter gene assay [AID1105617, Type: confirmatory] [gi:3041727]
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9
[SID194184891]
[CID76334423]
EC50 2.57e-08Transactivation of GAL4-fused Homo sapiens (human) PPARalpha/PPARgamma DNA binding domain expressed in African green monkey CV1 cells by luciferase reporter gene assay [AID1105617, Type: confirmatory] [gi:3041727]
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10
[SID134436215]
[CID56659348]
EC50 5e-08Transactivation of human PPARalpha expressed in human HepG2 cells co-transfected with PPRE3-TK-Luc by luciferase reporter gene assay [AID610309, Type: Literature] [gi:3041727]
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11
[SID134459372]
[CID56679849]
EC50 6e-08Transactivation of human PPARalpha expressed in human HepG2 cells co-transfected with PPRE3-TK-Luc by luciferase reporter gene assay [AID610309, Type: Literature] [gi:3041727]
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12
[SID103295006]
[CID446758]
EC50 6.17e-08Transactivation of GAL4-fused Homo sapiens (human) PPARalpha/PPARgamma DNA binding domain expressed in African green monkey CV1 cells by luciferase reporter gene assay [AID1105617, Type: confirmatory] [gi:3041727]
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13
[SID134447814]
[CID56669690]
EC50 7e-08Transactivation of human PPARalpha expressed in human HepG2 cells co-transfected with PPRE3-TK-Luc by luciferase reporter gene assay [AID610309, Type: Literature] [gi:3041727]
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14
[SID194136727]
[CID76309039]
EC50 1.66e-07Transactivation of GAL4-fused Homo sapiens (human) PPARalpha/PPARgamma DNA binding domain expressed in African green monkey CV1 cells by luciferase reporter gene assay [AID1105617, Type: confirmatory] [gi:3041727]
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15
[SID103295111]
[CID44321572]
EC50 2.69e-07Transactivation of GAL4-fused Homo sapiens (human) PPARalpha/PPARgamma DNA binding domain expressed in African green monkey CV1 cells by luciferase reporter gene assay [AID1105617, Type: confirmatory] [gi:3041727]
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16
[SID134455510]
[CID53233135]
EC50 3.1e-07Transactivation of human PPARalpha expressed in human HepG2 cells co-transfected with PPRE3-TK-Luc by luciferase reporter gene assay [AID610309, Type: Literature] [gi:3041727]
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17
[SID103294065]
[CID44320978]
EC50 5.37e-07Transactivation of GAL4-fused Homo sapiens (human) PPARalpha/PPARgamma DNA binding domain expressed in African green monkey CV1 cells by luciferase reporter gene assay [AID1105617, Type: confirmatory] [gi:3041727]
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18
[SID103422072]
[CID10896153]
EC50 7.94e-07Transactivation of GAL4-fused Homo sapiens (human) PPARalpha/PPARgamma DNA binding domain expressed in African green monkey CV1 cells by luciferase reporter gene assay [AID1105617, Type: confirmatory] [gi:3041727]
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19
[SID103295062]
[CID44321548]
EC50 1.2e-06Transactivation of GAL4-fused Homo sapiens (human) PPARalpha/PPARgamma DNA binding domain expressed in African green monkey CV1 cells by luciferase reporter gene assay [AID1105617, Type: confirmatory] [gi:3041727]
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20
[SID103293909]
[CID44320897]
EC50 1.66e-06Transactivation of GAL4-fused Homo sapiens (human) PPARalpha/PPARgamma DNA binding domain expressed in African green monkey CV1 cells by luciferase reporter gene assay [AID1105617, Type: confirmatory] [gi:3041727]
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