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OPRM1 (geneid:4988) - Gene BioActivity Data
Also known as: LMOR, M-OR-1, MOP, MOR, MOR1, OPRM.
BioActivity Outcomes:
Active(5987)
 
 
Inactive(676219)
 
 
Inconclusive(329)
 
 
Unspecified(2548)
 
 
BioAssay Types:
Screening(677199)
 
 
 
 
Literature(5502)
 
 
 
 
 
Confirmatory(2335)
 
 
 
 
BioActivity Types:
Ki(2218)
 
 
 
 
 
EC50(1817)
 
 
 
 
 
IC50(1711)
 
 
 
 
 
Kd(24)
 
 
 
Substance Types:
Chemical(685071)
 
 
 
 
 
RNAi(12)
 
 
 
 
Data download

Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 646    Data Row: 685083   Total Pages: 34255   Display: Page     
Sort: [Click the result table header to sort]
#StructureSubstanceCompoundActivityBioAssayTargetLinks
OutcomeTypeValue [μM]
1
[SID164129496]
[CID71605589]
EC50 4.2e-08Agonist activity at FLAG-tagged mu-type opioid receptor (unknown origin) expressed in HEK293 cells assessed as inhibition of forskolin-stimulated cAMP accumulation after 30 mins by liquid scintillation counting analysis [AID730862, Type: Literature] [gi:2851402]
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2
[SID164140762]
[CID71605588]
EC50 9.12e-08Agonist activity at FLAG-tagged mu-type opioid receptor (unknown origin) expressed in HEK293 cells assessed as inhibition of forskolin-stimulated cAMP accumulation after 30 mins by liquid scintillation counting analysis [AID730862, Type: Literature] [gi:2851402]
View
3
[SID164129460]
[CID71605755]
EC50 1.07e-07Agonist activity at FLAG-tagged mu-type opioid receptor (unknown origin) expressed in HEK293 cells assessed as inhibition of forskolin-stimulated cAMP accumulation after 30 mins by liquid scintillation counting analysis [AID730862, Type: Literature] [gi:2851402]
View
4
[SID164140761]
[CID71605756]
EC50 1.09e-07Agonist activity at FLAG-tagged mu-type opioid receptor (unknown origin) expressed in HEK293 cells assessed as inhibition of forskolin-stimulated cAMP accumulation after 30 mins by liquid scintillation counting analysis [AID730862, Type: Literature] [gi:2851402]
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5
[SID164149159]
[CID71720682]
EC50 1.3e-07Agonist activity at FLAG-tagged mu-type opioid receptor (unknown origin) expressed in HEK293 cells assessed as inhibition of forskolin-stimulated cAMP accumulation after 30 mins by liquid scintillation counting analysis [AID730862, Type: Literature] [gi:2851402]
View
6
[SID164143536]
[CID71719454]
EC50 5.16e-07Agonist activity at FLAG-tagged mu-type opioid receptor (unknown origin) expressed in HEK293 cells assessed as inhibition of forskolin-stimulated cAMP accumulation after 30 mins by liquid scintillation counting analysis [AID730862, Type: Literature] [gi:2851402]
View
7
[SID103293205]
[CID5311080]
EC50 1e-06Activity at mu opioid receptor assessed as increase in calcium level in CHO cells by aequorin luminescence based calcium assay [AID277678, Type: Literature] [gi:2851402]
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8
[SID163339747]
[CID58443234]
Ki 1.6e-06Displacement of [3H]DAMGO from human mu opioid receptor expressed in CHO cells after 60 mins by scintillation counting [AID719453, Type: Literature] [gi:2851402]
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9
[SID163337288]
[CID54669894]
EC50 1.74e-06Agonist activity at human MOR expressed in HEK293 cell membrane assessed as inhibition of forskolin-induced cAMP accumulation by by liquid scintillation counting [AID690645, Type: Literature] [gi:2851402]
View
10
[SID134434099]
[CID6602241]
Ki 3e-06Displacement of [3H]DAMGO from human mu opioid receptor expressed in CHO cells [AID259394, Type: Literature] [gi:2851402]
View
11
[SID164129496]
[CID71605589]
Ki 3.72e-06Displacement of [3H]DAMGO from FLAG-tagged mu-type opioid receptor (unknown origin) expressed in HEK293 cells after 60 mins by liquid scintillation counting analysis [AID730870, Type: Literature] [gi:2851402]
View
12
[SID163322529]
[CID71454361]
Ki 4.9e-06Displacement of [3H]DAMGO from human mu opioid receptor expressed in CHO cells after 60 mins by scintillation counting [AID719453, Type: Literature] [gi:2851402]
View
13
[SID163322528]
[CID58443225]
Ki 5.6e-06Displacement of [3H]DAMGO from human mu opioid receptor expressed in CHO cells after 60 mins by scintillation counting [AID719453, Type: Literature] [gi:2851402]
View
14
[SID163325912]
[CID71456106]
Ki 5.6e-06Displacement of [3H]DAMGO from human mu opioid receptor expressed in CHO cells after 60 mins by scintillation counting [AID719453, Type: Literature] [gi:2851402]
View
15
[SID163322530]
[CID71454362]
Ki 7.1e-06Displacement of [3H]DAMGO from human mu opioid receptor expressed in CHO cells after 60 mins by scintillation counting [AID719453, Type: Literature] [gi:2851402]
View
16
[SID164137991]
[CID71605419]
EC50 8.53e-06Agonist activity at FLAG-tagged mu-type opioid receptor (unknown origin) expressed in HEK293 cells assessed as inhibition of forskolin-stimulated cAMP accumulation after 30 mins by liquid scintillation counting analysis [AID730862, Type: Literature] [gi:2851402]
View
17
[SID164140762]
[CID71605588]
Ki 9.86e-06Displacement of [3H]DAMGO from FLAG-tagged mu-type opioid receptor (unknown origin) expressed in HEK293 cells after 60 mins by liquid scintillation counting analysis [AID730870, Type: Literature] [gi:2851402]
View
18
[SID103248656]
[CID44301701]
Ki 1e-05Binding affinity to mu opioid receptor (unknown origin) [AID754478, Type: Literature] [gi:2851402]
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19
[SID103476378]
[CID44406663]
Ki 1e-05Displacement of [3H]DAMGO from human mu opioid receptor expressed in CHO cells [AID259394, Type: Literature] [gi:2851402]
View
20
[SID103500785]
[CID16087283]
IC50 1.25e-05Activity at human recombinant mu opioid receptor expressed in CHO cells assessed as stimulation of [35S]GTP-gamma-S binding [AID273141, Type: Literature] [gi:2851402]
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