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OPRK1 (geneid:4986) - Gene BioActivity Data
Also known as: K-OR-1, KOR, KOR-1, OPRK.
BioActivity Outcomes:
Probe(4)
 
 
Active(3837)
 
 
Inactive(591108)
 
 
Inconclusive(307)
 
 
Unspecified(2548)
 
 
BioAssay Types:
Confirmatory(576477)
 
 
 
 
 
Screening(16007)
 
 
 
 
Literature(5230)
 
 
 
 
 
Summary(4)
 
 
BioActivity Types:
IC50(292300)
 
 
 
 
 
EC50(285247)
 
 
 
 
 
Ki(2166)
 
 
 
 
 
Kd(1)
 
 
Substance Types:
Chemical(597792)
 
 
 
 
 
 
RNAi(12)
 
 
 
 
Data download

Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 589    Data Row: 597804   Total Pages: 29891   Display: Page     
Sort: [Click the result table header to sort]
#StructureSubstanceCompoundActivityBioAssayTargetLinks
OutcomeTypeValue [μM]
1
[SID87218782]
[CID5236771]
Summary of small molecule agonists of the kappa opioid receptor [AID1786, Type: summary] [gi:39725940]
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2
[SID87218794]
[CID3342390]
Summary of small molecule antagonists of the kappa opioid receptor [AID1785, Type: summary] [gi:39725940]
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3
[SID87334039]
[CID44601470]
Summary of small molecule agonists of the kappa opioid receptor [AID1786, Type: summary] [gi:39725940]
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4
[SID88442997]
[CID44665680]
Summary of small molecule antagonists of the kappa opioid receptor [AID1785, Type: summary] [gi:39725940]
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5
[SID103500899]
[CID16087270]
IC50 3e-06Activity at human recombinant kappa opioid receptor expressed in CHO cells assessed as stimulation of [35S]GTP-gamma-S binding [AID273145, Type: Literature] [gi:116242691]
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6
[SID134434099]
[CID6602241]
Ki 3e-06Displacement of [3H]U69593 from human kappa opioid receptor expressed in CHO cells [AID259396, Type: Literature] [gi:116242691]
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7
[SID103500785]
[CID16087283]
IC50 6e-06Activity at human recombinant kappa opioid receptor expressed in CHO cells assessed as stimulation of [35S]GTP-gamma-S binding [AID273145, Type: Literature] [gi:116242691]
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8
[SID164132787]
[CID71625152]
EC50 6.1e-06Agonist activity at human KOR expressed in CHO cells assessed as stimulation of [35S]GTPgammaS binding [AID735221, Type: Literature] [gi:116242691]
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9
[SID164132788]
[CID71625277]
EC50 7e-06Agonist activity at human KOR expressed in CHO cells assessed as stimulation of [35S]GTPgammaS binding [AID735221, Type: Literature] [gi:116242691]
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10
[SID164144042]
[CID71625278]
EC50 7.7e-06Agonist activity at human KOR expressed in CHO cells assessed as stimulation of [35S]GTPgammaS binding [AID735221, Type: Literature] [gi:116242691]
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11
[SID164129948]
[CID71625279]
EC50 9.8e-06Agonist activity at human KOR expressed in CHO cells assessed as stimulation of [35S]GTPgammaS binding [AID735221, Type: Literature] [gi:116242691]
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12
[SID164135610]
[CID71624552]
EC50 1.1e-05Agonist activity at human KOR expressed in CHO cells assessed as stimulation of [35S]GTPgammaS binding [AID735221, Type: Literature] [gi:116242691]
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13
[SID164149695]
[CID71625151]
EC50 1.3e-05Agonist activity at human KOR expressed in CHO cells assessed as stimulation of [35S]GTPgammaS binding [AID735221, Type: Literature] [gi:116242691]
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14
[SID164146758]
[CID71625027]
Ki 1.5e-05Displacement of [3H]-diprenorphine from human KOR expressed in CHO cells [AID735689, Type: Literature] [gi:116242691]
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15
[SID164135611]
[CID71624663]
EC50 1.6e-05Agonist activity at human KOR expressed in CHO cells assessed as stimulation of [35S]GTPgammaS binding [AID735221, Type: Literature] [gi:116242691]
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16
[SID164138476]
[CID71624555]
EC50 1.7e-05Agonist activity at human KOR expressed in CHO cells assessed as stimulation of [35S]GTPgammaS binding [AID735221, Type: Literature] [gi:116242691]
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17
[SID164149694]
[CID71625028]
Ki 1.9e-05Displacement of [3H]-diprenorphine from human KOR expressed in CHO cells [AID735689, Type: Literature] [gi:116242691]
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18
[SID103328513]
[CID44337683]
Ki 2e-05Ratio of kappa/delta-opioid receptors Binding affinity [AID228131, Type: Literature] [gi:116242691]
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19
[SID164138472]
[CID71625029]
Ki 2e-05Displacement of [3H]-diprenorphine from human KOR expressed in CHO cells [AID735689, Type: Literature] [gi:116242691]
View
20
[SID164138473]
[CID71625393]
EC50 2e-05Agonist activity at human KOR expressed in CHO cells assessed as stimulation of [35S]GTPgammaS binding [AID735221, Type: Literature] [gi:116242691]
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