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OPRD1 (geneid:4985) - Gene BioActivity Data
Also known as: OPRD.
BioActivity Outcomes:
Active(4965)
 
 
Inactive(674008)
 
 
Inconclusive(157)
 
 
Unspecified(2307)
 
 
BioAssay Types:
Screening(674934)
 
 
 
 
Literature(4250)
 
 
 
 
 
Confirmatory(2234)
 
 
 
 
BioActivity Types:
Ki(1854)
 
 
 
 
IC50(1631)
 
 
 
 
 
EC50(1439)
 
 
 
 
 
Kd(6)
 
 
Substance Types:
Chemical(681425)
 
 
 
 
 
RNAi(12)
 
 
 
Data download

Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 499    Data Row: 681437   Total Pages: 34072   Display: Page     
Sort: [Click the result table header to sort]
#StructureSubstanceCompoundActivityBioAssayTargetLinks
OutcomeTypeValue [μM]
1
[SID103225178]
[CID9875567]
EC50 1e-05Activity at delta opioid receptor assessed as increase in calcium level in CHO cells by aequorin luminescence based calcium assay [AID277680, Type: Literature] [gi:311033488]
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2
[SID163337288]
[CID54669894]
EC50 1.6e-05Agonist activity at human DOR expressed in HEK293 cell membrane assessed as inhibition of forskolin-induced cAMP accumulation by by liquid scintillation counting [AID690647, Type: Literature] [gi:311033488]
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3
[SID103720324]
[CID46227362]
EC50 1.74e-05Agonist activity at human delta opioid receptor expressed in HN9.10 cells assessed as stimulation of [35S]GTPgammaS binding [AID452780, Type: Literature] [gi:311033488]
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4
[SID103682580]
[CID23642304]
EC50 1.8e-05Agonist activity at human recombinant delta opioid receptor expressed in human HEK293 cells by [35S]GTPgammaS binding assay [AID636101, Type: Literature] [gi:311033488]
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5
[SID103682580]
[CID23642304]
EC50 1.8e-05Agonist activity at human recombinant delta opioid receptor expressed in HEK293 cells by [35S]GTPgammaS binding assay [AID424039, Type: Literature] [gi:311033488]
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6
[SID103328513]
[CID44337683]
Ki 2e-05Ratio of kappa/delta-opioid receptors Binding affinity [AID228131, Type: Literature] [gi:311033488]
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7
[SID131283791]
[CID5360515]
Ki 2e-05Ratio of mu/delta-opioid receptors Binding affinity [AID228132, Type: Literature] [gi:311033488]
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8
[SID103500785]
[CID16087283]
IC50 2e-05Activity at human recombinant delta opioid receptor expressed in CHO cells assessed as stimulation of [35S]GTP-gamma-S binding [AID273143, Type: Literature] [gi:311033488]
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9
[SID103653367]
[CID44138064]
Ki 2.5e-05Displacement of [3H]naltrindole from human delta opioid receptor expressed in CHO cells after 3 hrs by scintillation counting [AID416814, Type: Literature] [gi:311033488]
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10
[SID103328773]
[CID44337800]
Ki 3e-05Ratio of kappa/delta-opioid receptors Binding affinity [AID228131, Type: Literature] [gi:311033488]
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11
[SID103500899]
[CID16087270]
IC50 3e-05Activity at human recombinant delta opioid receptor expressed in CHO cells assessed as stimulation of [35S]GTP-gamma-S binding [AID273143, Type: Literature] [gi:311033488]
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12
[SID103629454]
[CID10864183]
Ki 3.1e-05Binding affinity to delta opioid receptor [AID266690, Type: Literature] [gi:311033488]
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13
[SID174490420]
[CID73347271]
Ki 3.5e-05Binding affinity to delta opioid receptor [AID266690, Type: Literature] [gi:311033488]
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14
[SID103328370]
[CID44337613]
Ki 4e-05Ratio of kappa/delta-opioid receptors Binding affinity [AID228131, Type: Literature] [gi:311033488]
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15
[SID131283791]
[CID5360515]
Ki 4e-05Ratio of kappa/delta-opioid receptors Binding affinity [AID228131, Type: Literature] [gi:311033488]
View
16
[SID103642507]
[CID11016572]
Ki 4.2e-05Binding affinity to delta opioid receptor [AID266690, Type: Literature] [gi:311033488]
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17
[SID103689528]
[CID44467662]
EC50 4.7e-05Agonist activity at human recombinant delta opioid receptor expressed in HEK293 cells by [35S]GTPgammaS binding assay [AID424039, Type: Literature] [gi:311033488]
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18
[SID103689528]
[CID44467662]
EC50 4.7e-05Agonist activity at human recombinant delta opioid receptor expressed in human HEK293 cells by [35S]GTPgammaS binding assay [AID636101, Type: Literature] [gi:311033488]
View
19
[SID103687877]
[CID45270599]
EC50 6e-05Agonist activity at human recombinant delta opioid receptor expressed in human HEK293 cells by [35S]GTPgammaS binding assay [AID636101, Type: Literature] [gi:311033488]
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20
[SID103687877]
[CID45270599]
EC50 6e-05Agonist activity at human recombinant delta opioid receptor expressed in HEK293 cells by [35S]GTPgammaS binding assay [AID424039, Type: Literature] [gi:311033488]
View