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HTR5A (geneid:3361) - Gene BioActivity Data
Also known as: 5-HT5A.
BioActivity Outcomes:
Active(2793)
 
 
Inactive(671784)
 
 
Inconclusive(11)
 
 
Unspecified(157)
 
 
BioAssay Types:
Screening(674138)
 
 
 
Literature(333)
 
 
 
 
 
Confirmatory(269)
 
 
BioActivity Types:
EC50(269)
 
 
Ki(176)
 
 
 
 
IC50(18)
 
 
 
Kd(6)
 
 
 
Substance Types:
Chemical(674737)
 
 
 
 
 
RNAi(8)
 
 
 
Data download

Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 105    Data Row: 674745   Total Pages: 33738   Display: Page     
Sort: [Click the result table header to sort]
#StructureSubstanceCompoundActivityBioAssayTargetLinks
OutcomeTypeValue [μM]
1
[SID104238293]
[CID44469677]
IC50 0.001Displacement of [3H]LSD from human recombinant 5HT5A receptor expressed in CHO cells [AID493596, Type: Literature] [gi:1345607]
View
2
[SID103307762]
[CID4106]
Ki 0.001Binding affinity towards human 5-hydroxytryptamine 5A receptor [AID6479, Type: Literature] [gi:1345607]
View
3
[SID103307762]
[CID4106]
Ki 0.001Binding affinity towards human 5-hydroxytryptamine 5A receptor was evaluated using [3H]-5-CT as radioligand [AID6480, Type: Literature] [gi:1345607]
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4
[SID103575411]
[CID44456033]
Ki 0.0016Binding affinity to human 5HT5A receptor [AID316378, Type: Literature] [gi:1345607]
View
5
[SID103575647]
[CID44456230]
Ki 0.0018Binding affinity to human 5HT5A receptor [AID316378, Type: Literature] [gi:1345607]
View
6
[SID103575301]
[CID16093484]
Ki 0.002Displacement of [3H]LSD from human recombinant 5HT5A receptor expressed in HEK293-EBNA cells [AID315623, Type: Literature] [gi:1345607]
View
7
[SID103575344]
[CID16006492]
Kd 0.00302Antagonist activity at human recombinant 5HT5A receptor expressed in HEK293-EBNA cells by [35S]GTP-gamma-S binding assay [AID315637, Type: Literature] [gi:1345607]
View
8
[SID103575344]
[CID16006492]
Kd 0.00316Antagonist activity at human 5HT5A receptor by [35S]GTP-gamma-S binding assay [AID316379, Type: Literature] [gi:1345607]
View
9
[SID103575834]
[CID16093485]
Ki 0.0047Displacement of [3H]LSD from human recombinant 5HT5A receptor expressed in HEK293-EBNA cells [AID315623, Type: Literature] [gi:1345607]
View
10
[SID103575344]
[CID16006492]
Ki 0.0051Displacement of [3H]LSD from human recombinant 5HT5A receptor expressed in HEK293-EBNA cells [AID315623, Type: Literature] [gi:1345607]
View
11
[SID103575690]
[CID16006599]
Ki 0.0057Binding affinity to human 5HT5A receptor [AID316378, Type: Literature] [gi:1345607]
View
12
[SID103575920]
[CID16006496]
Ki 0.0063Displacement of [3H]LSD from human recombinant 5HT5A receptor expressed in HEK293-EBNA cells [AID315623, Type: Literature] [gi:1345607]
View
13
[SID103575921]
[CID16006606]
Ki 0.0063Displacement of [3H]LSD from human recombinant 5HT5A receptor expressed in HEK293-EBNA cells [AID315623, Type: Literature] [gi:1345607]
View
14
[SID103575789]
[CID16006605]
Ki 0.0065Displacement of [3H]LSD from human recombinant 5HT5A receptor expressed in HEK293-EBNA cells [AID315623, Type: Literature] [gi:1345607]
View
15
[SID103575371]
[CID44456001]
Ki 0.0068Binding affinity to human 5HT5A receptor [AID316378, Type: Literature] [gi:1345607]
View
16
[SID103575304]
[CID16006493]
Kd 0.00741Antagonist activity at human recombinant 5HT5A receptor expressed in HEK293-EBNA cells by [35S]GTP-gamma-S binding assay [AID315637, Type: Literature] [gi:1345607]
View
17
[SID103575837]
[CID16006607]
Ki 0.01Displacement of [3H]LSD from human recombinant 5HT5A receptor expressed in HEK293-EBNA cells [AID315623, Type: Literature] [gi:1345607]
View
18
[SID103575731]
[CID16006495]
Ki 0.0101Binding affinity to human 5HT5A receptor [AID316378, Type: Literature] [gi:1345607]
View
19
[SID103575304]
[CID16006493]
Ki 0.0108Displacement of [3H]LSD from human recombinant 5HT5A receptor expressed in HEK293-EBNA cells [AID315623, Type: Literature] [gi:1345607]
View
20
[SID103183384]
[CID1809]
Ki 0.02Binding affinity towards human 5-hydroxytryptamine 5A receptor [AID6479, Type: Literature] [gi:1345607]
View