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HTR5A (geneid:3361) - Gene BioActivity Data
Also known as: 5-HT5A.
BioActivity Outcomes:
Active(2758)
 
 
Inactive(671783)
 
 
Inconclusive(3)
 
 
Unspecified(118)
 
 
BioAssay Types:
Screening(674137)
 
 
 
Confirmatory(269)
 
 
Literature(250)
 
 
 
 
 
BioActivity Types:
EC50(269)
 
 
Ki(138)
 
 
 
 
IC50(16)
 
 
 
Kd(6)
 
 
 
Substance Types:
Chemical(674655)
 
 
 
 
 
RNAi(7)
 
 
 
Data download

Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 91    Data Row: 674662   Total Pages: 13494   Display: Page     
Sort: [Click the result table header to sort]
#StructureSubstanceCompoundActivityBioAssayTargetLinks
OutcomeTypeValue [μM]
1
[SID103307762]
[CID4106]
Ki 0.001Binding affinity towards human 5-hydroxytryptamine 5A receptor [AID6479, Type: Literature] [gi:1345607]
View
2
[SID103307762]
[CID4106]
Ki 0.001Binding affinity towards human 5-hydroxytryptamine 5A receptor was evaluated using [3H]-5-CT as radioligand [AID6480, Type: Literature] [gi:1345607]
View
3
[SID104238293]
[CID44469677]
IC50 0.001Displacement of [3H]LSD from human recombinant 5HT5A receptor expressed in CHO cells [AID493596, Type: Literature] [gi:1345607]
View
4
[SID103575411]
[CID44456033]
Ki 0.0016Binding affinity to human 5HT5A receptor [AID316378, Type: Literature] [gi:1345607]
View
5
[SID103575647]
[CID44456230]
Ki 0.0018Binding affinity to human 5HT5A receptor [AID316378, Type: Literature] [gi:1345607]
View
6
[SID103575301]
[CID16093484]
Ki 0.002Displacement of [3H]LSD from human recombinant 5HT5A receptor expressed in HEK293-EBNA cells [AID315623, Type: Literature] [gi:1345607]
View
7
[SID103575344]
[CID16006492]
Kd 0.00302Antagonist activity at human recombinant 5HT5A receptor expressed in HEK293-EBNA cells by [35S]GTP-gamma-S binding assay [AID315637, Type: Literature] [gi:1345607]
View
8
[SID103575344]
[CID16006492]
Kd 0.00316Antagonist activity at human 5HT5A receptor by [35S]GTP-gamma-S binding assay [AID316379, Type: Literature] [gi:1345607]
View
9
[SID103575834]
[CID16093485]
Ki 0.0047Displacement of [3H]LSD from human recombinant 5HT5A receptor expressed in HEK293-EBNA cells [AID315623, Type: Literature] [gi:1345607]
View
10
[SID103575344]
[CID16006492]
Ki 0.0051Displacement of [3H]LSD from human recombinant 5HT5A receptor expressed in HEK293-EBNA cells [AID315623, Type: Literature] [gi:1345607]
View
11
[SID103575690]
[CID16006599]
Ki 0.0057Binding affinity to human 5HT5A receptor [AID316378, Type: Literature] [gi:1345607]
View
12
[SID103575920]
[CID16006496]
Ki 0.0063Displacement of [3H]LSD from human recombinant 5HT5A receptor expressed in HEK293-EBNA cells [AID315623, Type: Literature] [gi:1345607]
View
13
[SID103575921]
[CID16006606]
Ki 0.0063Displacement of [3H]LSD from human recombinant 5HT5A receptor expressed in HEK293-EBNA cells [AID315623, Type: Literature] [gi:1345607]
View
14
[SID103575789]
[CID16006605]
Ki 0.0065Displacement of [3H]LSD from human recombinant 5HT5A receptor expressed in HEK293-EBNA cells [AID315623, Type: Literature] [gi:1345607]
View
15
[SID103575371]
[CID44456001]
Ki 0.0068Binding affinity to human 5HT5A receptor [AID316378, Type: Literature] [gi:1345607]
View
16
[SID103575304]
[CID16006493]
Kd 0.00741Antagonist activity at human recombinant 5HT5A receptor expressed in HEK293-EBNA cells by [35S]GTP-gamma-S binding assay [AID315637, Type: Literature] [gi:1345607]
View
17
[SID103575837]
[CID16006607]
Ki 0.01Displacement of [3H]LSD from human recombinant 5HT5A receptor expressed in HEK293-EBNA cells [AID315623, Type: Literature] [gi:1345607]
View
18
[SID103575731]
[CID16006495]
Ki 0.0101Binding affinity to human 5HT5A receptor [AID316378, Type: Literature] [gi:1345607]
View
19
[SID103575304]
[CID16006493]
Ki 0.0108Displacement of [3H]LSD from human recombinant 5HT5A receptor expressed in HEK293-EBNA cells [AID315623, Type: Literature] [gi:1345607]
View
20
[SID103183384]
[CID1809]
Ki 0.02Binding affinity towards human 5-hydroxytryptamine 5A receptor [AID6479, Type: Literature] [gi:1345607]
View
21
[SID103183384]
[CID1809]
Ki 0.02Binding affinity towards human 5-hydroxytryptamine 5A receptor was evaluated using [3H]-5-CT as radioligand [AID6480, Type: Literature] [gi:1345607]
View
22
[SID103575542]
[CID16006709]
Ki 0.0222Binding affinity to human 5HT5A receptor [AID316378, Type: Literature] [gi:1345607]
View
23
[SID103575544]
[CID44456149]
Ki 0.0222Binding affinity to human 5HT5A receptor [AID316378, Type: Literature] [gi:1345607]
View
24
[SID103575835]
[CID44456395]
Ki 0.0229Displacement of [3H]LSD from human recombinant 5HT5A receptor expressed in HEK293-EBNA cells [AID315623, Type: Literature] [gi:1345607]
View
25
[SID103575350]
[CID44455986]
Ki 0.024Displacement of [3H]LSD from human recombinant 5HT5A receptor expressed in HEK293-EBNA cells [AID315623, Type: Literature] [gi:1345607]
View
26
[SID103575836]
[CID44456396]
Ki 0.0254Displacement of [3H]LSD from human recombinant 5HT5A receptor expressed in HEK293-EBNA cells [AID315623, Type: Literature] [gi:1345607]
View
27
[SID103575300]
[CID44455943]
Ki 0.0265Displacement of [3H]LSD from human recombinant 5HT5A receptor expressed in HEK293-EBNA cells [AID315623, Type: Literature] [gi:1345607]
View
28
[SID103575599]
[CID16006711]
Ki 0.0282Binding affinity to human 5HT5A receptor [AID316378, Type: Literature] [gi:1345607]
View
29
[SID103575455]
[CID44456071]
Ki 0.0334Binding affinity to human 5HT5A receptor [AID316378, Type: Literature] [gi:1345607]
View
30
[SID103575600]
[CID44456195]
Ki 0.037Binding affinity to human 5HT5A receptor [AID316378, Type: Literature] [gi:1345607]
View
31
[SID103679503]
[CID45265979]
Ki 0.038Displacement of [3H]LSD from human recombinant 5HT5A receptor expressed in HEK293-EBNA cells [AID315623, Type: Literature] [gi:1345607]
View
32
[SID103679503]
[CID45265979]
Ki 0.038Binding affinity to human 5HT5A receptor [AID316378, Type: Literature] [gi:1345607]
View
33
[SID103575731]
[CID16006495]
Kd 0.0389Antagonist activity at human 5HT5A receptor by [35S]GTP-gamma-S binding assay [AID316379, Type: Literature] [gi:1345607]
View
34
[SID103575519]
[CID9904281]
Ki 0.043Displacement of [3H]LSD from human recombinant 5HT5A receptor expressed in HEK293-EBNA cells [AID315623, Type: Literature] [gi:1345607]
View
35
[SID103308379]
[CID10382508]
Ki 0.055Binding affinity towards human 5-hydroxytryptamine 5A receptor [AID6479, Type: Literature] [gi:1345607]
View
36
[SID103575343]
[CID44455973]
Ki 0.0844Displacement of [3H]LSD from human recombinant 5HT5A receptor expressed in HEK293-EBNA cells [AID315623, Type: Literature] [gi:1345607]
View
37
[SID103575779]
[CID44456354]
Ki 0.087Binding affinity to human 5HT5A receptor [AID316378, Type: Literature] [gi:1345607]
View
38
[SID103575545]
[CID44456150]
Ki 0.096Binding affinity to human 5HT5A receptor [AID316378, Type: Literature] [gi:1345607]
View
39
[SID103679506]
[CID45265982]
Ki 0.097Displacement of [3H]LSD from human recombinant 5HT5A receptor expressed in HEK293-EBNA cells [AID315623, Type: Literature] [gi:1345607]
View
40
[SID103575518]
[CID13702393]
Ki 0.099Displacement of [3H]LSD from human recombinant 5HT5A receptor expressed in HEK293-EBNA cells [AID315623, Type: Literature] [gi:1345607]
View
41
[SID103676404]
[CID45263888]
Ki 0.099Displacement of [3H]LSD from human recombinant 5HT5A receptor expressed in HEK293-EBNA cells [AID315623, Type: Literature] [gi:1345607]
View
42
[SID103575241]
[CID44455897]
Ki 0.103Binding affinity to human 5HT5A receptor [AID316378, Type: Literature] [gi:1345607]
View
43
[SID103575330]
[CID44455963]
Ki 0.122Binding affinity to human 5HT5A receptor [AID316378, Type: Literature] [gi:1345607]
View
44
[SID103575502]
[CID44456111]
Ki 0.124Binding affinity to human 5HT5A receptor [AID316378, Type: Literature] [gi:1345607]
View
45
[SID103165719]
[CID5202]
Ki 0.126Binding affinity towards human 5-hydroxytryptamine 5A receptor was evaluated using [3H]-5-CT as radioligand [AID6480, Type: Literature] [gi:1345607]
View
46
[SID103676403]
[CID45263887]
Ki 0.145Displacement of [3H]LSD from human recombinant 5HT5A receptor expressed in HEK293-EBNA cells [AID315623, Type: Literature] [gi:1345607]
View
47
[SID103575900]
[CID44456463]
Ki 0.153Binding affinity to human 5HT5A receptor [AID316378, Type: Literature] [gi:1345607]
View
48
[SID103575547]
[CID44456152]
Ki 0.163Binding affinity to human 5HT5A receptor [AID316378, Type: Literature] [gi:1345607]
View
49
[SID103677945]
[CID10392062]
Ki 0.168Binding affinity towards 5-hydroxytryptamine 5A receptor [AID6498, Type: Literature] [gi:1345607]
View
50
[SID103165719]
[CID5202]
Ki 0.17Displacement of [3H]LSD from human 5HT5A receptor [AID611937, Type: Literature] [gi:1345607]
View