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GLP1R (geneid:2740) - Gene BioActivity Data
BioActivity Outcomes:
Active(6723)
 
 
Inactive(696571)
 
 
Inconclusive(83184)
 
 
Unspecified(97)
 
 
BioAssay Types:
Confirmatory(786211)
 
 
 
 
Literature(354)
 
 
 
 
 
Screening(5)
 
 
BioActivity Types:
Potency(786211)
 
 
 
 
EC50(157)
 
 
 
 
IC50(102)
 
 
 
 
Ki(5)
 
 
Kd(1)
 
 
Substance Types:
Chemical(786563)
 
 
 
 
 
RNAi(12)
 
 
 
Data download

Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 54    Data Row: 786575   Total Pages: 39329   Display: Page     
Sort: [Click the result table header to sort]
#StructureSubstanceCompoundActivityBioAssayTargetLinks
OutcomeTypeValue [μM]
1
[SID194146381]
[CID76314012]
EC50 1.5e-06Activation of human GLP-1 receptor overexpressed in HEK293 cells assessed as cAMP accumulation after 20 mins by HTRF assay [AID1066039, Type: Literature] [gi:311033387]
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2
[SID103529204]
[CID16157882]
EC50 1.5e-06Activation of human GLP-1 receptor overexpressed in HEK293 cells assessed as cAMP accumulation after 20 mins by HTRF assay [AID1066039, Type: Literature] [gi:311033387]
View
3
[SID103645615]
[CID44588329]
EC50 2e-06Activation of human GLP1R expressed in HEK293 cells assessed as effect on cAMP responsive element promoter driven luciferase expression [AID388010, Type: Literature] [gi:311033387]
View
4
[SID103645623]
[CID44588337]
EC50 2.1e-06Activation of human GLP1R expressed in HEK293 cells assessed as effect on cAMP responsive element promoter driven luciferase expression [AID388010, Type: Literature] [gi:311033387]
View
5
[SID103645622]
[CID44588336]
EC50 2.8e-06Activation of human GLP1R expressed in HEK293 cells assessed as effect on cAMP responsive element promoter driven luciferase expression [AID388010, Type: Literature] [gi:311033387]
View
6
[SID103645621]
[CID44588335]
EC50 2.9e-06Activation of human GLP1R expressed in HEK293 cells assessed as effect on cAMP responsive element promoter driven luciferase expression [AID388010, Type: Literature] [gi:311033387]
View
7
[SID194146382]
[CID76314013]
EC50 3e-06Activation of human GLP-1 receptor overexpressed in HEK293 cells assessed as cAMP accumulation after 20 mins by HTRF assay [AID1066039, Type: Literature] [gi:311033387]
View
8
[SID103621977]
[CID44577331]
EC50 3e-06Agonist activity at human GLP1R expressed in CHO cells assessed as increase in cAMP level by cAMP-response element/luciferase activation assay [AID385218, Type: Literature] [gi:311033387]
View
9
[SID194167152]
[CID76324901]
EC50 3.2e-06Activation of human GLP-1 receptor overexpressed in HEK293 cells assessed as cAMP accumulation after 20 mins by HTRF assay [AID1066039, Type: Literature] [gi:311033387]
View
10
[SID194160215]
[CID76321286]
EC50 3.2e-06Activation of human GLP-1 receptor overexpressed in HEK293 cells assessed as cAMP accumulation after 20 mins by HTRF assay [AID1066039, Type: Literature] [gi:311033387]
View
11
[SID103645627]
[CID44588341]
EC50 3.3e-06Activation of human GLP1R expressed in HEK293 cells assessed as effect on cAMP responsive element promoter driven luciferase expression [AID388010, Type: Literature] [gi:311033387]
View
12
[SID103450617]
[CID16135499]
EC50 3.3e-06Activation of human GLP-1 receptor overexpressed in HEK293 cells assessed as cAMP accumulation after 20 mins by HTRF assay [AID1066039, Type: Literature] [gi:311033387]
View
13
[SID194180860]
[CID76332142]
EC50 3.4e-06Activation of human GLP-1 receptor overexpressed in HEK293 cells assessed as cAMP accumulation after 20 mins by HTRF assay [AID1066039, Type: Literature] [gi:311033387]
View
14
[SID103645608]
[CID44588322]
EC50 3.63e-06Activation of human GLP1R expressed in HEK293 cells assessed as effect on cAMP responsive element promoter driven luciferase expression [AID388010, Type: Literature] [gi:311033387]
View
15
[SID103645616]
[CID44588330]
EC50 3.8e-06Activation of human GLP1R expressed in HEK293 cells assessed as effect on cAMP responsive element promoter driven luciferase expression [AID388010, Type: Literature] [gi:311033387]
View
16
[SID194173972]
[CID76328461]
EC50 3.8e-06Activation of human GLP-1 receptor overexpressed in HEK293 cells assessed as cAMP accumulation after 20 mins by HTRF assay [AID1066039, Type: Literature] [gi:311033387]
View
17
[SID103621991]
[CID44577345]
EC50 4e-06Agonist activity at human GLP1R expressed in CHO cells assessed as increase in cAMP level by cAMP-response element/luciferase activation assay [AID385218, Type: Literature] [gi:311033387]
View
18
[SID103529204]
[CID16157882]
EC50 4e-06Agonist activity at human GLP1R expressed in CHO cells assessed as increase in cAMP level by cAMP-response element/luciferase activation assay [AID385218, Type: Literature] [gi:311033387]
View
19
[SID103645624]
[CID44588338]
EC50 4.8e-06Activation of human GLP1R expressed in HEK293 cells assessed as effect on cAMP responsive element promoter driven luciferase expression [AID388010, Type: Literature] [gi:311033387]
View
20
[SID194146379]
[CID76314010]
EC50 4.9e-06Activation of human GLP-1 receptor overexpressed in HEK293 cells assessed as cAMP accumulation after 20 mins by HTRF assay [AID1066039, Type: Literature] [gi:311033387]
View