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F2 (geneid:2147) - Gene BioActivity Data
Also known as: PT, RPRGL2, THPH1.
BioActivity Outcomes:
Active(2272)
 
 
Inactive(217144)
 
 
Inconclusive(85)
 
 
Unspecified(941)
 
 
BioAssay Types:
Screening(217250)
 
 
 
Literature(2630)
 
 
 
 
 
Confirmatory(529)
 
 
 
 
BioActivity Types:
IC50(1310)
 
 
 
 
 
Ki(1001)
 
 
 
 
 
Kd(15)
 
 
 
 
 
Substance Types:
Chemical(220435)
 
 
 
 
 
RNAi(7)
 
 
 
 
Data download

Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 234    Data Row: 220442   Total Pages: 4409   Display: Page     
Sort: [Click the result table header to sort]
#StructureSubstanceCompoundActivityBioAssayTargetLinks
OutcomeTypeValue [μM]
1
[SID103467135]
[CID10074165]
Ki 1e-06Binding affinity against thrombin in human plasma [AID238307, Type: Literature] [gi:135807]
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2
[SID103467095]
[CID10029817]
Ki 2e-06Binding affinity against thrombin in human plasma [AID238307, Type: Literature] [gi:135807]
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3
[SID103466840]
[CID11755549]
Ki 1e-05Binding affinity against thrombin in human plasma [AID238307, Type: Literature] [gi:135807]
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4
[SID103467596]
[CID44402668]
Ki 1e-05Binding affinity against thrombin in human plasma [AID238307, Type: Literature] [gi:135807]
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5
[SID103467426]
[CID10027333]
Ki 4e-05Binding affinity against thrombin in human plasma [AID238307, Type: Literature] [gi:135807]
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6
[SID103471019]
[CID10367956]
Ki 4e-05Inhibitory constant against thrombin [AID254280, Type: Literature] [gi:135807]
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7
[SID103471133]
[CID9954791]
Ki 4e-05Inhibitory constant against thrombin [AID254280, Type: Literature] [gi:135807]
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8
[SID103223097]
[CID9872549]
Ki 4e-05Inhibition of thrombin in human plasma [AID211176, Type: Literature] [gi:135807]
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9
[SID103220074]
[CID122296]
Ki 4.2e-05Inhibition of Coagulation factor II [AID51156, Type: Literature] [gi:135807]
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10
[SID103467199]
[CID10098601]
Ki 5e-05Binding affinity against thrombin in human plasma [AID238307, Type: Literature] [gi:135807]
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11
[SID163315727]
[CID46899738]
Ki 5.2e-05Inhibition of human thrombin using Tos-Gly-Pro-Arg-AMC as substrate after 600 secs by fluorimetric method [AID690519, Type: Literature] [gi:135807]
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12
[SID103471079]
[CID10390121]
Ki 6e-05Inhibitory constant against thrombin [AID254280, Type: Literature] [gi:135807]
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13
[SID103470978]
[CID10098302]
Ki 7e-05Inhibitory constant against thrombin [AID254280, Type: Literature] [gi:135807]
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14
[SID103223054]
[CID44289618]
Ki 7e-05Inhibition of thrombin in human plasma [AID211176, Type: Literature] [gi:135807]
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15
[SID103470977]
[CID44404152]
Ki 8e-05Inhibitory constant against thrombin [AID254280, Type: Literature] [gi:135807]
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16
[SID103467599]
[CID44402671]
Ki 8e-05Binding affinity against thrombin in human plasma [AID238307, Type: Literature] [gi:135807]
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17
[SID103385141]
[CID11762017]
Ki 0.0001Binding affinity to human thrombin [AID331733, Type: Literature] [gi:135807]
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18
[SID104241273]
[CID46899735]
Ki 0.000102Inhibition of human thrombin [AID499183, Type: Literature] [gi:135807]
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19
[SID104241274]
[CID46899737]
Ki 0.000108Inhibition of human thrombin [AID499183, Type: Literature] [gi:135807]
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20
[SID134441768]
[CID46899736]
Ki 0.000119Inhibition of human thrombin using Tos-Gly-Pro-Arg-AMC as substrate after 600 secs by fluorimetric method [AID690519, Type: Literature] [gi:135807]
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21
[SID103439872]
[CID23646580]
Ki 0.00012Binding affinity determined against human alpha thrombin [AID238527, Type: Literature] [gi:135807]
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22
[SID103439893]
[CID23646608]
Ki 0.00014Binding affinity determined against human alpha thrombin [AID238527, Type: Literature] [gi:135807]
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23
[SID103466775]
[CID10255447]
Ki 0.00014Binding affinity against thrombin in human plasma [AID238307, Type: Literature] [gi:135807]
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24
[SID103470972]
[CID10324635]
Ki 0.00014Inhibitory constant against thrombin [AID254280, Type: Literature] [gi:135807]
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25
[SID103439936]
[CID23646610]
Ki 0.00015Binding affinity determined against human alpha thrombin [AID238527, Type: Literature] [gi:135807]
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26
[SID103471001]
[CID10051489]
Ki 0.00016Inhibitory constant against thrombin [AID254280, Type: Literature] [gi:135807]
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27
[SID103439901]
[CID23646582]
Ki 0.00018Binding affinity determined against human alpha thrombin [AID238527, Type: Literature] [gi:135807]
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28
[SID103439901]
[CID23646582]
Ki 0.00018Inhibition constant against human alpha thrombin [AID238705, Type: Literature] [gi:135807]
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29
[SID103571922]
[CID9872263]
Ki 0.00018Inhibition constant against human alpha thrombin [AID238705, Type: Literature] [gi:135807]
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30
[SID103741053]
Kd 0.00018Binding affinity to human thrombin after 30 mins by non-equilibrium capillary electrophoresis [AID463302, Type: Literature] [gi:135807]
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31
[SID103571922]
[CID9872263]
Ki 0.00019Inhibition of human alpha-thrombin. [AID211230, Type: Literature] [gi:135807]
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32
[SID103571922]
[CID9872263]
Ki 0.0002Binding affinity determined against human alpha thrombin [AID238527, Type: Literature] [gi:135807]
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33
[SID103439941]
[CID73346747]
Ki 0.0002Binding affinity determined against human alpha thrombin [AID238527, Type: Literature] [gi:135807]
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34
[SID103741055]
Kd 0.00021Binding affinity to human thrombin after 30 mins by non-equilibrium capillary electrophoresis [AID463302, Type: Literature] [gi:135807]
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35
[SID103439920]
[CID23646609]
Ki 0.00023Binding affinity determined against human alpha thrombin [AID238527, Type: Literature] [gi:135807]
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36
[SID103467531]
[CID10435712]
Ki 0.00023Binding affinity against thrombin in human plasma [AID238307, Type: Literature] [gi:135807]
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37
[SID103471018]
[CID10390490]
Ki 0.00025Inhibitory constant against thrombin [AID254280, Type: Literature] [gi:135807]
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38
[SID103741052]
Kd 0.00025Binding affinity to human thrombin after 30 mins by non-equilibrium capillary electrophoresis [AID463302, Type: Literature] [gi:135807]
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39
[SID163323508]
[CID57411954]
Ki 0.000259Inhibition of human thrombin using Tos-Gly-Pro-Arg-AMC as substrate after 600 secs by fluorimetric method [AID690519, Type: Literature] [gi:135807]
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40
[SID103741054]
Kd 0.00027Binding affinity to human thrombin after 30 mins by non-equilibrium capillary electrophoresis [AID463302, Type: Literature] [gi:135807]
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41
[SID103448932]
[CID44393000]
Ki 0.00027Inhibition constant against human Thrombin [AID238244, Type: Literature] [gi:135807]
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42
[SID103351330]
[CID44347623]
Ki 0.00028Inhibition of Thrombin [AID211234, Type: Literature] [gi:135807]
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43
[SID103741056]
Kd 0.00028Binding affinity to human thrombin after 30 mins by non-equilibrium capillary electrophoresis [AID463302, Type: Literature] [gi:135807]
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44
[SID103471002]
[CID10004800]
Ki 0.00031Inhibitory constant against thrombin [AID254280, Type: Literature] [gi:135807]
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45
[SID103439917]
[CID23646594]
Ki 0.00034Binding affinity determined against human alpha thrombin [AID238527, Type: Literature] [gi:135807]
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46
[SID103439954]
[CID23646586]
Ki 0.00036Binding affinity determined against human alpha thrombin [AID238527, Type: Literature] [gi:135807]
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47
[SID103439956]
[CID23646611]
Ki 0.00037Binding affinity determined against human alpha thrombin [AID238527, Type: Literature] [gi:135807]
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48
[SID103563457]
[CID44448740]
Ki 0.00038Binding affinity to human thrombin [AID331733, Type: Literature] [gi:135807]
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49
[SID103166154]
[CID9913629]
Ki 0.00038Binding affinity towards human thrombin [AID210997, Type: Literature] [gi:135807]
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50
[SID103467303]
[CID10479448]
Ki 0.0004Binding affinity against thrombin in human plasma [AID238307, Type: Literature] [gi:135807]
View