Bookmark and Share
EPAS1 (geneid:2034) - Gene BioActivity Data
Also known as: ECYT4, HIF2A, HLF, MOP2, PASD2, bHLHe73.
BioActivity Outcomes:
Active(3996)
 
 
Inactive(362854)
 
 
Inconclusive(2)
 
 
Unspecified(1114)
 
 
BioAssay Types:
Screening(365932)
 
 
 
Confirmatory(1932)
 
 
 
 
Literature(100)
 
 
 
 
BioActivity Types:
IC50(1932)
 
 
 
 
Kd(22)
 
 
 
EC50(22)
 
 
 
 
Substance Types:
Chemical(367954)
 
 
 
 
RNAi(12)
 
 
 
Data download

Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 56    Data Row: 367966   Total Pages: 18399   Display: Page     
Sort: [Click the result table header to sort]
#StructureSubstanceCompoundActivityBioAssayTargetLinks
OutcomeTypeValue [μM]
1
[SID164133446]
[CID70697712]
Kd 0.09Binding affinity to wild type PAS-B domain of HIF-2alpha (unknown origin) by isothermal calorimetry analysis [AID723542, Type: Literature] [gi:32470617]
View
2
[SID164144653]
[CID71575455]
Kd 0.16Binding affinity to wild type PAS-B domain of HIF-2alpha (unknown origin) by isothermal calorimetry analysis [AID723542, Type: Literature] [gi:32470617]
View
3
[SID164139102]
[CID2842377]
Kd 0.17Binding affinity to wild type PAS-B domain of HIF-2alpha (unknown origin) by isothermal calorimetry analysis [AID723542, Type: Literature] [gi:32470617]
View
4
[SID164141863]
[CID71575558]
Kd 0.17Binding affinity to wild type PAS-B domain of HIF-2alpha (unknown origin) by isothermal calorimetry analysis [AID723542, Type: Literature] [gi:32470617]
View
5
[SID4254515]
[CID972733]
IC50_HIF-2a_PANC_Mean 0.19Dose response confirmation of uHTS identification of HIF-2a Inhibitors in screening - selectivity counterscreen assays [AID651581_7, Type: confirmatory] [gi:40254439]
View
6
[SID103061877]
[CID666941]
IC50_Mean_HIF2a (PANC cells) 0.19SAR Analysis small molecule inhibitors of HIF-1a in a panel assay [AID652011, Type: confirmatory] [gi:40254439]
View
7
[SID103061905]
[CID1994282]
IC50_Mean_HIF2a (PANC cells) 0.19SAR Analysis small molecule inhibitors of HIF-1a in a panel assay [AID652011, Type: confirmatory] [gi:40254439]
View
8
[SID103061912]
[CID1943900]
IC50_Mean_HIF2a (PANC cells) 0.19SAR Analysis small molecule inhibitors of HIF-1a in a panel assay [AID652011, Type: confirmatory] [gi:40254439]
View
9
[SID103061963]
[CID2037423]
IC50_Mean_HIF2a (PANC cells) 0.19SAR Analysis small molecule inhibitors of HIF-1a in a panel assay [AID652011, Type: confirmatory] [gi:40254439]
View
10
[SID103061971]
[CID3159504]
IC50_Mean_HIF2a (PANC cells) 0.19SAR Analysis small molecule inhibitors of HIF-1a in a panel assay [AID652011, Type: confirmatory] [gi:40254439]
View
11
[SID103061973]
[CID666941]
IC50_Mean_HIF2a (PANC cells) 0.19SAR Analysis small molecule inhibitors of HIF-1a in a panel assay [AID652011, Type: confirmatory] [gi:40254439]
View
12
[SID110067516]
[CID50898046]
IC50_Mean_HIF2a (PANC cells) 0.19SAR Analysis small molecule inhibitors of HIF-1a in a panel assay [AID652011, Type: confirmatory] [gi:40254439]
View
13
[SID110067538]
[CID50898044]
IC50_Mean_HIF2a (PANC cells) 0.19SAR Analysis small molecule inhibitors of HIF-1a in a panel assay [AID652011, Type: confirmatory] [gi:40254439]
View
14
[SID110067542]
[CID50898039]
IC50_Mean_HIF2a (PANC cells) 0.19SAR Analysis small molecule inhibitors of HIF-1a in a panel assay [AID652011, Type: confirmatory] [gi:40254439]
View
15
[SID49675252]
[CID854968]
IC50_HIF-2a_PANC_Mean 0.247Dose response confirmation of uHTS identification of HIF-2a Inhibitors in screening - selectivity counterscreen assays [AID651581_7, Type: confirmatory] [gi:40254439]
View
16
[SID22411729]
[CID15945494]
IC50_HIF-2a_PANC_Mean 0.25Dose response confirmation of uHTS identification of HIF-2a Inhibitors in screening - selectivity counterscreen assays [AID651581_7, Type: confirmatory] [gi:40254439]
View
17
[SID49665726]
[CID2767825]
IC50_1_HIF-1a 0.274Dose response confirmation of uHTS identification of HIF-2a Inhibitors in screening - selectivity counterscreen assays [AID651581, Type: confirmatory] [gi:40254439]
View
18
[SID49725274]
[CID1991339]
IC50_HIF-2a_PANC_Mean 0.3Dose response confirmation of uHTS identification of HIF-2a Inhibitors in screening - selectivity counterscreen assays [AID651581_7, Type: confirmatory] [gi:40254439]
View
19
[SID17510599]
[CID9657888]
IC50_HIF-2a_PANC_Mean 0.3Dose response confirmation of uHTS identification of HIF-2a Inhibitors in screening - selectivity counterscreen assays [AID651581_7, Type: confirmatory] [gi:40254439]
View
20
[SID865680]
[CID666941]
IC50_HIF-2a_PANC_Mean 0.3Dose response confirmation of uHTS identification of HIF-2a Inhibitors in screening - selectivity counterscreen assays [AID651581_7, Type: confirmatory] [gi:40254439]
View