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CXCR6 (geneid:10663) - Gene BioActivity Data
Also known as: BONZO, CD186, STRL33, TYMSTR.
BioActivity Outcomes:
Active(2049)
 
 
Inactive(362437)
 
 
Unspecified(1514)
 
 
BioAssay Types:
Screening(363092)
 
 
 
Confirmatory(2897)
 
 
 
 
Literature(11)
 
 
 
BioActivity Types:
IC50(2897)
 
 
 
 
Substance Types:
Chemical(365993)
 
 
 
 
RNAi(7)
 
 
 
Data download

Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 15    Data Row: 366000   Total Pages: 7320   Display: Page     
Sort: [Click the result table header to sort]
#StructureSubstanceCompoundActivityBioAssayTargetLinks
OutcomeTypeValue [μM]
1
[SID150864418]
[CID60202254]
IC50_CXCR6_Mean 0.137SAR analysis of small molecule antagonists of the CXCR6 receptor in a screening panel assay - 4 [AID651919, Type: confirmatory] [gi:5730106]
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2
[SID144220967]
[CID60202254]
IC50_CXCR6_Mean 0.338SAR analysis of small molecule antagonists of the CXCR6 receptor in a screening panel assay - 3 [AID651708, Type: confirmatory] [gi:5730106]
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3
[SID144220967]
[CID60202254]
IC50_CXCR6_Mean 0.338SAR analysis of small molecule antagonists of the CXCR6 receptor in a screening panel assay - 3 [AID651708_7, Type: confirmatory] [gi:5730106]
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4
[SID144220967]
[CID60202254]
IC50_CXCR6_Mean 0.356SAR analysis of small molecule antagonists of the CXCR6 receptor in a screening panel assay - 4 [AID651919, Type: confirmatory] [gi:5730106]
View
5
[SID16953942]
[CID2055076]
IC50_CXCR6_Mean 1.07Dose Response confirmation of uHTS hits from a small molecule antagonists of the CXCR6 receptor in a screening assay [AID624129, Type: confirmatory] [gi:5730106]
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6
[SID144220963]
[CID60202215]
IC50_CXCR6_Mean 1.46SAR analysis of small molecule antagonists of the CXCR6 receptor in a screening panel assay - 3 [AID651708, Type: confirmatory] [gi:5730106]
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7
[SID144220963]
[CID60202215]
IC50_CXCR6_Mean 1.46SAR analysis of small molecule antagonists of the CXCR6 receptor in a screening panel assay - 3 [AID651708_7, Type: confirmatory] [gi:5730106]
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8
[SID144220963]
[CID60202215]
IC50_CXCR6_Mean 1.48SAR analysis of small molecule antagonists of the CXCR6 receptor in a screening panel assay - 4 [AID651919, Type: confirmatory] [gi:5730106]
View
9
[SID144220966]
[CID60202261]
IC50_CXCR6_Mean 1.85SAR analysis of small molecule antagonists of the CXCR6 receptor in a screening panel assay - 4 [AID651919, Type: confirmatory] [gi:5730106]
View
10
[SID144220966]
[CID60202261]
IC50_CXCR6_Mean 1.95SAR analysis of small molecule antagonists of the CXCR6 receptor in a screening panel assay - 3 [AID651708, Type: confirmatory] [gi:5730106]
View
11
[SID144220966]
[CID60202261]
IC50_CXCR6_Mean 1.95SAR analysis of small molecule antagonists of the CXCR6 receptor in a screening panel assay - 3 [AID651708_7, Type: confirmatory] [gi:5730106]
View
12
[SID99361013]
[CID6511382]
IC50_CXCR6_Mean 2.41Dose Response confirmation of uHTS hits from a small molecule antagonists of the CXCR6 receptor in a screening assay [AID624129, Type: confirmatory] [gi:5730106]
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13
[SID49673350]
[CID9684646]
IC50_CXCR6_Mean 3.33Dose Response confirmation of uHTS hits from a small molecule antagonists of the CXCR6 receptor in a screening assay [AID624129, Type: confirmatory] [gi:5730106]
View
14
[SID144220951]
[CID653186]
IC50_CXCR6_Mean 3.4SAR analysis of small molecule antagonists of the CXCR6 receptor in a screening panel assay - 4 [AID651919, Type: confirmatory] [gi:5730106]
View
15
[SID144220962]
[CID60202201]
IC50_CXCR6_Mean 3.51SAR analysis of small molecule antagonists of the CXCR6 receptor in a screening panel assay - 3 [AID651708, Type: confirmatory] [gi:5730106]
View
16
[SID144220962]
[CID60202201]
IC50_CXCR6_Mean 3.51SAR analysis of small molecule antagonists of the CXCR6 receptor in a screening panel assay - 3 [AID651708_7, Type: confirmatory] [gi:5730106]
View
17
[SID17414893]
[CID887191]
IC50_CXCR6_Mean 4.62Dose Response confirmation of uHTS hits from a small molecule antagonists of the CXCR6 receptor in a screening assay [AID624129, Type: confirmatory] [gi:5730106]
View
18
[SID144220973]
[CID653186]
IC50_CXCR6_Mean 4.74SAR analysis of small molecule antagonists of the CXCR6 receptor in a screening panel assay - 4 [AID651919, Type: confirmatory] [gi:5730106]
View
19
[SID144220973]
[CID653186]
IC50_CXCR6_Mean 4.75SAR analysis of small molecule antagonists of the CXCR6 receptor in a screening panel assay - 3 [AID651708, Type: confirmatory] [gi:5730106]
View
20
[SID144220973]
[CID653186]
IC50_CXCR6_Mean 4.75SAR analysis of small molecule antagonists of the CXCR6 receptor in a screening panel assay - 3 [AID651708_7, Type: confirmatory] [gi:5730106]
View
21
[SID144220951]
[CID653186]
IC50_CXCR6_Mean 4.78SAR analysis of small molecule antagonists of the CXCR6 receptor in a screening panel assay - 3 [AID651708, Type: confirmatory] [gi:5730106]
View
22
[SID144220951]
[CID653186]
IC50_CXCR6_Mean 4.78SAR analysis of small molecule antagonists of the CXCR6 receptor in a screening panel assay - 3 [AID651708_7, Type: confirmatory] [gi:5730106]
View
23
[SID89854985]
[CID2817]
IC50_CXCR6_Mean 4.82Dose Response confirmation of uHTS hits from a small molecule antagonists of the CXCR6 receptor in a screening assay [AID624129, Type: confirmatory] [gi:5730106]
View
24
[SID47200567]
[CID3544398]
IC50_CXCR6_Mean 5.44Dose Response confirmation of uHTS hits from a small molecule antagonists of the CXCR6 receptor in a screening assay [AID624129, Type: confirmatory] [gi:5730106]
View
25
[SID49680007]
[CID2796987]
IC50_CXCR6_Mean 5.58Dose Response confirmation of uHTS hits from a small molecule antagonists of the CXCR6 receptor in a screening assay [AID624129, Type: confirmatory] [gi:5730106]
View
26
[SID144220964]
[CID60202246]
IC50_CXCR6_Mean 5.69SAR analysis of small molecule antagonists of the CXCR6 receptor in a screening panel assay - 3 [AID651708, Type: confirmatory] [gi:5730106]
View
27
[SID144220964]
[CID60202246]
IC50_CXCR6_Mean 5.69SAR analysis of small molecule antagonists of the CXCR6 receptor in a screening panel assay - 3 [AID651708_7, Type: confirmatory] [gi:5730106]
View
28
[SID144088974]
[CID653186]
IC50_CXCR6_Mean 6.08SAR analysis of small molecule antagonists of the CXCR6 receptor in an APJ-DiscoveRx counter screen panel assay [AID651598, Type: confirmatory] [gi:5730106]
View
29
[SID92763750]
[CID373493]
IC50_CXCR6_Mean 6.38Dose Response confirmation of uHTS hits from a small molecule antagonists of the CXCR6 receptor in a screening assay [AID624129, Type: confirmatory] [gi:5730106]
View
30
[SID7970265]
[CID3694793]
IC50_CXCR6_Mean 7.46Dose Response confirmation of uHTS hits from a small molecule antagonists of the CXCR6 receptor in a screening assay [AID624129, Type: confirmatory] [gi:5730106]
View
31
[SID24832501]
[CID2106098]
IC50_CXCR6_Mean 7.48Dose Response confirmation of uHTS hits from a small molecule antagonists of the CXCR6 receptor in a screening assay [AID624129, Type: confirmatory] [gi:5730106]
View
32
[SID24809101]
[CID4879304]
IC50_CXCR6_Mean 7.79Dose Response confirmation of uHTS hits from a small molecule antagonists of the CXCR6 receptor in a screening assay [AID624129, Type: confirmatory] [gi:5730106]
View
33
[SID17409458]
[CID6418635]
IC50_CXCR6_Mean 8.46Dose Response confirmation of uHTS hits from a small molecule antagonists of the CXCR6 receptor in a screening assay [AID624129, Type: confirmatory] [gi:5730106]
View
34
[SID24807520]
[CID3157015]
IC50_CXCR6_Mean 8.56Dose Response confirmation of uHTS hits from a small molecule antagonists of the CXCR6 receptor in a screening assay [AID624129, Type: confirmatory] [gi:5730106]
View
35
[SID4244637]
[CID3239208]
IC50_CXCR6_Mean 9.15Dose Response confirmation of uHTS hits from a small molecule antagonists of the CXCR6 receptor in a screening assay [AID624129, Type: confirmatory] [gi:5730106]
View
36
[SID26726053]
[CID653186]
IC50_CXCR6_Mean 10.7Dose Response confirmation of uHTS hits from a small molecule antagonists of the CXCR6 receptor in a screening assay [AID624129, Type: confirmatory] [gi:5730106]
View
37
[SID144088970]
[CID653186]
IC50_CXCR6_Mean 14.3SAR analysis of small molecule antagonists of the CXCR6 receptor in a screening panel assay [AID651601, Type: confirmatory] [gi:5730106]
View
38
[SID144088970]
[CID653186]
IC50_CXCR6_Mean 14.3SAR analysis of small molecule antagonists of the CXCR6 receptor in a screening panel assay [AID651601_9, Type: confirmatory] [gi:5730106]
View
39
[SID99495631]
[CID56643191]
uHTS identification of CXCR6 Inhibitors in a B-arrestin luminescence assay [AID602244, Type: screening] [gi:5730106]
View
40
[SID99495631]
[CID56643191]
Single concentration confirmation of uHTS hits from a small molecule antagonists of the CXCR6 receptor via a luminescent beta-arrestin assay [AID602409, Type: screening] [gi:5730106]
View
41
[SID99495764]
[CID56643207]
uHTS identification of CXCR6 Inhibitors in a B-arrestin luminescence assay [AID602244, Type: screening] [gi:5730106]
View
42
[SID99495764]
[CID56643207]
Single concentration confirmation of uHTS hits from a small molecule antagonists of the CXCR6 receptor via a luminescent beta-arrestin assay [AID602409, Type: screening] [gi:5730106]
View
43
[SID144088974]
[CID653186]
IC50_CXCR6_Mean SAR analysis of small molecule antagonists of the CXCR6 receptor in an APJ-DiscoveRx counter screen panel assay [AID651598_8, Type: confirmatory] [gi:5730106]
View
44
[SID144220951]
[CID653186]
IC50_CXCR6_Mean SAR analysis of small molecule antagonists of the CXCR6 receptor in a screening panel assay - 4 [AID651919_1, Type: confirmatory] [gi:5730106]
View
45
[SID99494475]
[CID4853667]
uHTS identification of CXCR6 Inhibitors in a B-arrestin luminescence assay [AID602244, Type: screening] [gi:5730106]
View
46
[SID99495536]
[CID2888835]
uHTS identification of CXCR6 Inhibitors in a B-arrestin luminescence assay [AID602244, Type: screening] [gi:5730106]
View
47
[SID57261406]
[CID16955]
uHTS identification of CXCR6 Inhibitors in a B-arrestin luminescence assay [AID602244, Type: screening] [gi:5730106]
View
48
[SID57261279]
[CID3279941]
uHTS identification of CXCR6 Inhibitors in a B-arrestin luminescence assay [AID602244, Type: screening] [gi:5730106]
View
49
[SID57261279]
[CID3279941]
Single concentration confirmation of uHTS hits from a small molecule antagonists of the CXCR6 receptor via a luminescent beta-arrestin assay [AID602409, Type: screening] [gi:5730106]
View
50
[SID57261556]
[CID16328916]
uHTS identification of CXCR6 Inhibitors in a B-arrestin luminescence assay [AID602244, Type: screening] [gi:5730106]
View