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BioActivity Data for Targets
Filters: All Data » Active      
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BioActivity Outcomes:
Active(106)
 
 
BioAssay Types:
Literature(93)
 
 
BioActivity Types:
Ki(12)
 
 
IC50(3)
 
 
Substance Types:
Chemical(106)
 
 
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Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 7    Data Row: 106   Total Pages: 6   Display: Page     
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#StructureSubstanceCompoundActivityBioAssayLinks
OutcomeTypeValue [μM]
1
[SID103215832]
[CID9948785]
Ki 0.025Affinity for inactive human SkM1 sodium channel expressed in HEK293 cells [AID205290, Type: Literature]
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2
[SID103585628]
[CID11174599]
IC50 0.03Inhibition of voltage-gated Na channel 1.4 (unknown origin) [AID726289, Type: Literature]
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3
[SID103216185]
[CID9861009]
Ki 0.031Affinity for inactive human SkM1 sodium channel expressed in HEK293 cells [AID205290, Type: Literature]
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4
[SID103215833]
[CID9818665]
Ki 0.031Affinity for inactive human SkM1 sodium channel expressed in HEK293 cells [AID205290, Type: Literature]
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5
[SID103215939]
[CID11300443]
Ki 0.035Affinity for inactive human SkM1 sodium channel expressed in HEK293 cells [AID205290, Type: Literature]
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6
[SID103216153]
[CID11738446]
Ki 0.15Affinity for inactive human SkM1 sodium channel expressed in HEK293 cells [AID205290, Type: Literature]
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7
[SID103215238]
[CID9816959]
Ki 0.18Affinity for inactive human SkM1 sodium channel expressed in HEK293 cells [AID205290, Type: Literature]
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8
[SID103215976]
[CID9816478]
Ki 0.2Affinity for inactive human SkM1 sodium channel expressed in HEK293 cells [AID205290, Type: Literature]
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9
[SID103215977]
[CID2806138]
Ki 0.24Affinity for inactive human SkM1 sodium channel expressed in HEK293 cells [AID205290, Type: Literature]
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10
[SID103216152]
[CID11198140]
Ki 0.34Affinity for inactive human SkM1 sodium channel expressed in HEK293 cells [AID205290, Type: Literature]
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11
[SID134459314]
[CID53361524]
IC50 0.4Inhibition of 20% inactivated TTX-resistant human sodium channel Nav1.4 expressed in human HEK293 cells at 1 uM by patch-clamp electrophysiological assay [AID612194, Type: Literature]
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12
[SID103215975]
[CID11242617]
Ki 0.69Affinity for inactive human SkM1 sodium channel expressed in HEK293 cells [AID205290, Type: Literature]
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13
[SID103169867]
[CID3676]
IC50 2Modulation of human Nav1.4 in open-inactivated state assessed as inhibition of inward current after 4 mins by whole-cell electrophysiology [AID1069530, Type: Literature]
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14
[SID103199382]
[CID3878]
Ki 17Affinity for inactive human SkM1 sodium channel expressed in HEK293 cells [AID205290, Type: Literature]
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15
[SID103164546]
[CID1775]
Ki 24Affinity for inactive human SkM1 sodium channel expressed in HEK293 cells [AID205290, Type: Literature]
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16
[SID103164546]
[CID1775]
Sodium channel alpha subunit blocker [AID742738, Type: Literature]
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17
[SID103164546]
[CID1775]
Sodium channel alpha subunit blocker [AID742738, Type: Literature]
View
18
[SID103169867]
[CID3676]
Sodium channel alpha subunit blocker [AID742738, Type: Literature]
View
19
[SID103169867]
[CID3676]
Sodium channel alpha subunit blocker [AID742738, Type: Literature]
View
20
[SID103177753]
[CID2554]
Sodium channel alpha subunit blocker [AID742738, Type: Literature]
View