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BioActivity Data for Targets

Filters: All Data » Active      
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BioActivity Outcomes:
Active(122)
 
 
BioAssay Types:
Literature(109)
 
 
BioAssay Categories:
Biochemical(41)
 
 
Cell-based(27)
 
 
BioActivity Types:
IC50(19)
 
 
Ki(12)
 
 
Substance Types:
Chemical(122)
 
 
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Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 11    Data Row: 122   Total Pages: 7   Display: Page     
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#StructureSubstanceCompoundActivityBioAssayLinks
OutcomeTypeValue [μM]
1
[SID103215832]
[CID9948785]
Ki 0.025Affinity for inactive human SkM1 sodium channel expressed in HEK293 cells [AID205290, Type: Literature]
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2
[SID103585628]
[CID11174599]
IC50 0.03Inhibition of voltage-gated Na channel 1.4 (unknown origin) [AID726289, Type: Literature]
View
3
[SID103215833]
[CID9818665]
Ki 0.031Affinity for inactive human SkM1 sodium channel expressed in HEK293 cells [AID205290, Type: Literature]
View
4
[SID103216185]
[CID9861009]
Ki 0.031Affinity for inactive human SkM1 sodium channel expressed in HEK293 cells [AID205290, Type: Literature]
View
5
[SID103215939]
[CID11300443]
Ki 0.035Affinity for inactive human SkM1 sodium channel expressed in HEK293 cells [AID205290, Type: Literature]
View
6
[SID103216153]
[CID11738446]
Ki 0.15Affinity for inactive human SkM1 sodium channel expressed in HEK293 cells [AID205290, Type: Literature]
View
7
[SID103215238]
[CID9816959]
Ki 0.18Affinity for inactive human SkM1 sodium channel expressed in HEK293 cells [AID205290, Type: Literature]
View
8
[SID103215976]
[CID9816478]
Ki 0.2Affinity for inactive human SkM1 sodium channel expressed in HEK293 cells [AID205290, Type: Literature]
View
9
[SID103215977]
[CID2806138]
Ki 0.24Affinity for inactive human SkM1 sodium channel expressed in HEK293 cells [AID205290, Type: Literature]
View
10
[SID103216152]
[CID11198140]
Ki 0.34Affinity for inactive human SkM1 sodium channel expressed in HEK293 cells [AID205290, Type: Literature]
View
11
[SID134459314]
[CID53361524]
IC50 0.4Inhibition of 20% inactivated TTX-resistant human sodium channel Nav1.4 expressed in human HEK293 cells at 1 uM by patch-clamp electrophysiological assay [AID612194, Type: Literature]
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12
[SID103215975]
[CID11242617]
Ki 0.69Affinity for inactive human SkM1 sodium channel expressed in HEK293 cells [AID205290, Type: Literature]
View
13
[SID103169867]
[CID3676]
IC50 2Modulation of human Nav1.4 in open-inactivated state assessed as inhibition of inward current after 4 mins by whole-cell electrophysiology [AID1069530, Type: Literature]
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14
[SID242623116]
[CID53239561]
IC50 4.58Inhibition of human Nav1.4 assessed as inactivated-state block by patch-clamp electrophysiology/cell based assay [AID1129319, Type: Literature]
View
15
[SID194158690]
[CID76320732]
IC50 8Modulation of human Nav1.4 by automated patch clamp electrophysiology assay [AID1054865, Type: Literature]
View
16
[SID242623116]
[CID53239561]
IC50 10.5Inhibition of human Nav1.4 assessed as 10 Hz block by patch-clamp electrophysiology/cell based assay [AID1129318, Type: Literature]
View
17
[SID194153317]
[CID60167367]
IC50 14Modulation of human Nav1.4 in open-inactivated state assessed as inhibition of inward current after 4 mins by whole-cell electrophysiology [AID1069530, Type: Literature]
View
18
[SID194158692]
[CID76320734]
IC50 15Modulation of human Nav1.4 by automated patch clamp electrophysiology assay [AID1054865, Type: Literature]
View
19
[SID194180948]
[CID76332198]
IC50 15Modulation of human Nav1.4 in open-inactivated state assessed as inhibition of inward current after 4 mins by whole-cell electrophysiology [AID1069530, Type: Literature]
View
20
[SID194151690]
[CID76317019]
IC50 16Modulation of human Nav1.4 by automated patch clamp electrophysiology assay [AID1054865, Type: Literature]
View