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BioActivity Data for Target mitogen-activated protein kinase 1 [Homo sapi.. [gi:66932916]

Also known as: mitogen-activated protein kinase 1 [Homo sapiens].
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BioActivity Outcomes:
Active(1658)
 
 
BioAssay Types:
Confirmatory(1357)
 
 
Literature(287)
 
 
BioAssay Categories:
In vitro(28)
 
 
Biochemical(303)
 
 
Cell-based(136)
 
 
BioActivity Types:
Potency(1332)
 
 
IC50(167)
 
 
Ki(52)
 
 
Kd(10)
 
 
Substance Types:
Chemical(1658)
 
 
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Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 83    Data Row: 1658   Total Pages: 83   Display: Page     
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#StructureSubstanceCompoundActivityBioAssayLinks
OutcomeTypeValue [μM]
1
[SID103320641]
[CID10303277]
IC50 1e-05Inhibit ion of MAPK phosphorylation in LoVo cells [AID102178, Type: Literature]
View
2
[SID174523273]
[CID71555244]
IC50 0.000205Inhibition of human ERK2 pre-incubation for 15 mins before substrate addition measured after 60 mins by IMAP-FP assay [AID760524, Type: Literature]
View
3
[SID174518062]
[CID71555167]
IC50 0.000286Inhibition of human ERK2 pre-incubation for 15 mins before substrate addition measured after 60 mins by IMAP-FP assay [AID760524, Type: Literature]
View
4
[SID14729642]
[CID9550014]
Potency 0.0004qHTS Assay for Inhibitors of the ERK Signaling Pathway using a Homogeneous Screening Assay; Stimulation with EGF [AID1454, Type: confirmatory]
View
5
[SID174518061]
[CID71555247]
IC50 0.000851Inhibition of human ERK2 pre-incubation for 15 mins before substrate addition measured after 60 mins by IMAP-FP assay [AID760524, Type: Literature]
View
6
[SID242650899]
[CID90645249]
IC50 0.001Inhibition of human recombinant N-terminal 6-His-tagged ERK2 expressed in Escherichia coli using S/T17 as substrate after 30 mins by spectrophotometry [AID1157610, Type: Literature]
View
7
[SID242651010]
[CID60198530]
IC50 0.001Inhibition of human recombinant N-terminal 6-His-tagged ERK2 expressed in Escherichia coli using S/T17 as substrate after 30 mins by spectrophotometry [AID1157610, Type: Literature]
View
8
[SID242651011]
[CID90645253]
IC50 0.001Inhibition of human recombinant N-terminal 6-His-tagged ERK2 expressed in Escherichia coli using S/T17 as substrate after 30 mins by spectrophotometry [AID1157610, Type: Literature]
View
9
[SID242651012]
[CID90645254]
IC50 0.001Inhibition of human recombinant N-terminal 6-His-tagged ERK2 expressed in Escherichia coli using S/T17 as substrate after 30 mins by spectrophotometry [AID1157610, Type: Literature]
View
10
[SID242651580]
[CID86705475]
IC50 0.001Inhibition of human recombinant N-terminal 6-His-tagged ERK2 expressed in Escherichia coli using S/T17 as substrate after 30 mins by spectrophotometry [AID1157610, Type: Literature]
View
11
[SID242651582]
[CID90645256]
IC50 0.001Inhibition of human recombinant N-terminal 6-His-tagged ERK2 expressed in Escherichia coli using S/T17 as substrate after 30 mins by spectrophotometry [AID1157610, Type: Literature]
View
12
[SID242651583]
[CID90645247]
IC50 0.001Inhibition of human recombinant N-terminal 6-His-tagged ERK2 expressed in Escherichia coli using S/T17 as substrate after 30 mins by spectrophotometry [AID1157610, Type: Literature]
View
13
[SID242651006]
[CID60198532]
IC50 0.001Inhibition of human recombinant N-terminal 6-His-tagged ERK2 expressed in Escherichia coli using S/T17 as substrate after 30 mins by spectrophotometry [AID1157610, Type: Literature]
View
14
[SID242650903]
[CID90645252]
IC50 0.002Inhibition of human recombinant N-terminal 6-His-tagged ERK2 expressed in Escherichia coli using S/T17 as substrate after 30 mins by spectrophotometry [AID1157610, Type: Literature]
View
15
[SID242650441]
[CID90645270]
IC50 0.002Inhibition of human recombinant N-terminal 6-His-tagged ERK2 expressed in Escherichia coli using S/T17 as substrate after 30 mins by spectrophotometry [AID1157610, Type: Literature]
View
16
[SID242650438]
[CID90645267]
IC50 0.002Inhibition of human recombinant N-terminal 6-His-tagged ERK2 expressed in Escherichia coli using S/T17 as substrate after 30 mins by spectrophotometry [AID1157610, Type: Literature]
View
17
[SID242651581]
[CID90645255]
IC50 0.002Inhibition of human recombinant N-terminal 6-His-tagged ERK2 expressed in Escherichia coli using S/T17 as substrate after 30 mins by spectrophotometry [AID1157610, Type: Literature]
View
18
[SID242650901]
[CID60198399]
IC50 0.002Inhibition of human recombinant N-terminal 6-His-tagged ERK2 expressed in Escherichia coli using S/T17 as substrate after 30 mins by spectrophotometry [AID1157610, Type: Literature]
View
19
[SID242651009]
[CID90645280]
IC50 0.002Inhibition of human recombinant N-terminal 6-His-tagged ERK2 expressed in Escherichia coli using S/T17 as substrate after 30 mins by spectrophotometry [AID1157610, Type: Literature]
View
20
[SID242650789]
[CID90645248]
IC50 0.002Inhibition of human recombinant N-terminal 6-His-tagged ERK2 expressed in Escherichia coli using S/T17 as substrate after 30 mins by spectrophotometry [AID1157610, Type: Literature]
View