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BioActivity Data for Targets
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BioActivity Outcomes:
Active(346)
 
 
BioAssay Types:
Literature(339)
 
 
BioActivity Types:
IC50(238)
 
 
Ki(50)
 
 
Kd(36)
 
 
Substance Types:
Chemical(346)
 
 
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Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 54    Data Row: 346   Total Pages: 7   Display: Page     
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#StructureSubstanceCompoundActivityBioAssayLinks
OutcomeTypeValue [μM]
1
[SID103501363]
[CID6918852]
Kd 0.00061Binding constant for CDK4-cyclinD1 kinase domain [AID624780, Type: Literature]
View
2
[SID103501363]
[CID6918852]
Kd 0.00081Binding constant for CDK4-cyclinD3 kinase domain [AID624781, Type: Literature]
View
3
[SID103501363]
[CID6918852]
Ki 0.001Inhibition of CDK4/Cyclin D1 [AID271733, Type: Literature]
View
4
[SID103501396]
[CID10479319]
Ki 0.001Inhibition of CDK4/Cyclin D1 [AID271733, Type: Literature]
View
5
[SID103461562]
[CID5330279]
IC50 0.002Inhibition of [32P]ATP binding to Cyclin dependant kinase 4-cyclin D [AID241660, Type: Literature]
View
6
[SID103382741]
[CID5330583]
IC50 0.0023Inhibition of CDK4 [AID271344, Type: Literature]
View
7
[SID103501330]
[CID11743030]
Ki 0.003Inhibition of CDK4/Cyclin D1 [AID271733, Type: Literature]
View
8
[SID160692025]
[CID46937330]
IC50 0.003Inhibition of human CDK4/cyclin D1 expressed in baculovirus infected Sf9 cells assessed as inhibition of pRb Ser780 phosphorylation after 60 mins by TR-FRET assay [AID682622, Type: other]
View
9
[SID104234154]
[CID5287969]
Kd 0.0033Binding constant for CDK4-cyclinD3 kinase domain [AID624781, Type: Literature]
View
10
[SID103499353]
[CID44416598]
IC50 0.0036Inhibition of CDK4 [AID271344, Type: Literature]
View
11
[SID103461870]
[CID5330358]
IC50 0.004Inhibition of [32P]ATP binding to Cyclin dependant kinase 4-cyclin D [AID241660, Type: Literature]
View
12
[SID103492722]
[CID44413509]
IC50 0.0042Inhibition of CDK4 [AID266563, Type: Literature]
View
13
[SID103461766]
[CID5330278]
IC50 0.005Inhibition of [32P]ATP binding to Cyclin dependant kinase 4-cyclin D [AID241660, Type: Literature]
View
14
[SID103461687]
[CID5330356]
IC50 0.005Inhibition of [32P]ATP binding to Cyclin dependant kinase 4-cyclin D [AID241660, Type: Literature]
View
15
[SID123083941]
[CID49840037]
IC50 0.005Inhibition of human CDK4/cyclin D1 expressed in baculovirus infected Sf21 cells after 60 mins by TR-FRET assay [AID528447, Type: Literature]
View
16
[SID103501386]
[CID11975206]
Ki 0.006Inhibition of CDK4/Cyclin D1 [AID271733, Type: Literature]
View
17
[SID103461620]
[CID5330333]
IC50 0.006Inhibition of [32P]ATP binding to Cyclin dependant kinase 4-cyclin D [AID241660, Type: Literature]
View
18
[SID103461732]
[CID5330280]
IC50 0.006Inhibition of [32P]ATP binding to Cyclin dependant kinase 4-cyclin D [AID241660, Type: Literature]
View
19
[SID103499106]
[CID44416439]
IC50 0.006Inhibition of CDK4 [AID271344, Type: Literature]
View
20
[SID103499685]
[CID10292184]
IC50 0.006Inhibition of CDK4 [AID271344, Type: Literature]
View
21
[SID160692024]
[CID49786055]
IC50 0.006Inhibition of human CDK4/cyclin D1 expressed in baculovirus infected Sf9 cells assessed as inhibition of pRb Ser780 phosphorylation after 60 mins by TR-FRET assay [AID682622, Type: other]
View
22
[SID103499387]
[CID16046126]
IC50 0.0064Inhibition of CDK4 [AID271344, Type: Literature]
View
23
[SID103501306]
[CID9979700]
Ki 0.007Inhibition of CDK4/Cyclin D1 [AID271733, Type: Literature]
View
24
[SID103382397]
[CID5330254]
IC50 0.007Inhibition of [32P]ATP binding to Cyclin dependant kinase 4-cyclin D [AID241660, Type: Literature]
View
25
[SID123085735]
[CID49840176]
IC50 0.009Inhibition of human CDK4/cyclin D1 expressed in baculovirus infected Sf21 cells after 60 mins by TR-FRET assay [AID528447, Type: Literature]
View
26
[SID104234154]
[CID5287969]
Kd 0.009Binding constant for CDK4-cyclinD1 kinase domain [AID624780, Type: Literature]
View
27
[SID103492790]
[CID16037675]
IC50 0.0092Inhibition of CDK4 [AID266563, Type: Literature]
View
28
[SID103461819]
[CID5330331]
IC50 0.01Inhibition of [32P]ATP binding to Cyclin dependant kinase 4-cyclin D [AID241660, Type: Literature]
View
29
[SID103461702]
[CID5330332]
IC50 0.01Inhibition of [32P]ATP binding to Cyclin dependant kinase 4-cyclin D [AID241660, Type: Literature]
View
30
[SID103454690]
[CID6539369]
Ki 0.01Binding affinity for human cyclin-dependent kinase 4 [AID238431, Type: Literature]
View
31
[SID103455011]
[CID6539373]
Ki 0.01Binding affinity for human cyclin-dependent kinase 4 [AID238431, Type: Literature]
View
32
[SID103455041]
[CID11163861]
Ki 0.01Binding affinity for human cyclin-dependent kinase 4 [AID238431, Type: Literature]
View
33
[SID123097252]
[CID49765254]
IC50 0.01Inhibition of human CDK4/cyclin D1 expressed in baculovirus infected Sf21 cells after 60 mins by TR-FRET assay [AID528447, Type: Literature]
View
34
[SID103499384]
[CID44416618]
IC50 0.011Inhibition of CDK4 [AID271344, Type: Literature]
View
35
[SID104246363]
[CID49800100]
IC50 0.011Inhibition of human CDK4/cyclin D1 expressed in baculovirus infected Sf21 cells after 60 mins by TR-FRET assay [AID528447, Type: Literature]
View
36
[SID123085742]
[CID49840236]
IC50 0.011Inhibition of human CDK4/cyclin D1 expressed in baculovirus infected Sf21 cells after 60 mins by TR-FRET assay [AID528447, Type: Literature]
View
37
[SID103679305]
[CID45265861]
IC50 0.011Inhibition of CDK4 [AID271344, Type: Literature]
View
38
[SID104246362]
[CID49800099]
IC50 0.012Inhibition of human CDK4/cyclin D1 expressed in baculovirus infected Sf21 cells after 60 mins by TR-FRET assay [AID528447, Type: Literature]
View
39
[SID103643679]
[CID11338033]
Kd 0.012Binding constant for CDK4-cyclinD3 kinase domain [AID624781, Type: Literature]
View
40
[SID123099581]
[CID49840175]
IC50 0.012Inhibition of human CDK4/cyclin D1 expressed in baculovirus infected Sf21 cells after 60 mins by TR-FRET assay [AID528447, Type: Literature]
View
41
[SID160702826]
[CID49785477]
IC50 0.012Inhibition of human CDK4/cyclin D1 expressed in baculovirus infected Sf9 cells assessed as inhibition of pRb Ser780 phosphorylation after 60 mins by TR-FRET assay [AID682622, Type: other]
View
42
[SID123092643]
[CID49840235]
IC50 0.013Inhibition of human CDK4/cyclin D1 expressed in baculovirus infected Sf21 cells after 60 mins by TR-FRET assay [AID528447, Type: Literature]
View
43
[SID123099151]
[CID49840239]
IC50 0.013Inhibition of human CDK4/cyclin D1 expressed in baculovirus infected Sf21 cells after 60 mins by TR-FRET assay [AID528447, Type: Literature]
View
44
[SID103679213]
[CID45265807]
IC50 0.013Inhibition of CDK4 [AID271344, Type: Literature]
View
45
[SID103492759]
[CID44413527]
IC50 0.013Inhibition of CDK4 [AID266563, Type: Literature]
View
46
[SID103446454]
[CID5330329]
IC50 0.014Inhibition of [32P]ATP binding to Cyclin dependant kinase 4-cyclin D [AID241660, Type: Literature]
View
47
[SID103501375]
[CID10319097]
Ki 0.014Inhibition of CDK4/Cyclin D1 [AID271733, Type: Literature]
View
48
[SID160686554]
[CID66599617]
IC50 0.015Inhibition of human CDK4/cyclin D1 expressed in baculovirus infected Sf9 cells assessed as inhibition of pRb Ser780 phosphorylation after 60 mins by TR-FRET assay [AID682622, Type: other]
View
49
[SID103501395]
[CID10251513]
Ki 0.016Inhibition of CDK4/Cyclin D1 [AID271733, Type: Literature]
View
50
[SID123083466]
[CID49840237]
IC50 0.016Inhibition of human CDK4/cyclin D1 expressed in baculovirus infected Sf21 cells after 60 mins by TR-FRET assay [AID528447, Type: Literature]
View