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BioActivity Data for Targets
Filters: All Data » Active      
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BioActivity Outcomes:
Active(378)
 
 
BioAssay Types:
Literature(377)
 
 
BioActivity Types:
IC50(259)
 
 
Ki(50)
 
 
Kd(36)
 
 
Substance Types:
Chemical(378)
 
 
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Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 68    Data Row: 378   Total Pages: 19   Display: Page     
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#StructureSubstanceCompoundActivityBioAssayLinks
OutcomeTypeValue [μM]
1
[SID103501363]
[CID6918852]
Kd 0.00061Binding constant for CDK4-cyclinD1 kinase domain [AID624780, Type: Literature]
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2
[SID103501363]
[CID6918852]
Kd 0.00081Binding constant for CDK4-cyclinD3 kinase domain [AID624781, Type: Literature]
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3
[SID103501363]
[CID6918852]
Ki 0.001Inhibition of CDK4/Cyclin D1 [AID271733, Type: Literature]
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4
[SID103501396]
[CID10479319]
Ki 0.001Inhibition of CDK4/Cyclin D1 [AID271733, Type: Literature]
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5
[SID103461562]
[CID5330279]
IC50 0.002Inhibition of [32P]ATP binding to Cyclin dependant kinase 4-cyclin D [AID241660, Type: Literature]
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6
[SID103382741]
[CID5330583]
IC50 0.0023Inhibition of CDK4 [AID271344, Type: Literature]
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7
[SID194153632]
[CID76317846]
IC50 0.0023Inhibition of CDK4/cyclinD1 (unknown origin) [AID1069265, Type: Literature]
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8
[SID160692025]
[CID46937330]
IC50 0.003Inhibition of human CDK4/cyclin D1 expressed in baculovirus infected Sf9 cells assessed as inhibition of pRb Ser780 phosphorylation after 60 mins by TR-FRET assay [AID682622, Type: Literature]
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9
[SID103501330]
[CID11743030]
Ki 0.003Inhibition of CDK4/Cyclin D1 [AID271733, Type: Literature]
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10
[SID104234154]
[CID5287969]
Kd 0.0033Binding constant for CDK4-cyclinD3 kinase domain [AID624781, Type: Literature]
View
11
[SID103499353]
[CID44416598]
IC50 0.0036Inhibition of CDK4 [AID271344, Type: Literature]
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12
[SID194139911]
[CID56649281]
IC50 0.0038Inhibition of CDK4/cyclinD1 (unknown origin) [AID1069265, Type: Literature]
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13
[SID194139911]
[CID56649281]
IC50 0.00387Inhibition of CDK4/cyclinD1 (unknown origin) using retinoblastoma as substrate after 30 mins by autoradiography in presence of [gamma-32P]ATP [AID1069225, Type: Literature]
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14
[SID174516437]
[CID66553053]
IC50 0.004Inhibition of CDK4/Cyclin D1 (unknown origin)-mediated phosphorylation of peptide substrate incubated for 15 mins prior to substrate addition measured after 90 mins by P33-radiolabeled assay [AID745525, Type: Literature]
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15
[SID103461870]
[CID5330358]
IC50 0.004Inhibition of [32P]ATP binding to Cyclin dependant kinase 4-cyclin D [AID241660, Type: Literature]
View
16
[SID103492722]
[CID44413509]
IC50 0.0042Inhibition of CDK4 [AID266563, Type: Literature]
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17
[SID103461766]
[CID5330278]
IC50 0.005Inhibition of [32P]ATP binding to Cyclin dependant kinase 4-cyclin D [AID241660, Type: Literature]
View
18
[SID103461687]
[CID5330356]
IC50 0.005Inhibition of [32P]ATP binding to Cyclin dependant kinase 4-cyclin D [AID241660, Type: Literature]
View
19
[SID123083941]
[CID49840037]
IC50 0.005Inhibition of human CDK4/cyclin D1 expressed in baculovirus infected Sf21 cells after 60 mins by TR-FRET assay [AID528447, Type: Literature]
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20
[SID103461613]
[CID5330286]
IC50 0.00536Inhibition of CDK4/cyclinD1 (unknown origin) using retinoblastoma as substrate after 30 mins by autoradiography in presence of [gamma-32P]ATP [AID1069225, Type: Literature]
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