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mast/stem cell growth factor receptor Kit iso.. [gi:4557695] - Target BioActivity Data
Also known as: mast/stem cell growth factor receptor Kit isoform 1 precursor [Homo sapiens].
Filters: All Data » Active      
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BioActivity Outcomes:
Active(905)
 
 
BioAssay Types:
Literature(867)
 
 
Confirmatory(32)
 
 
BioActivity Types:
Kd(479)
 
 
IC50(353)
 
 
Ki(19)
 
 
Substance Types:
Chemical(905)
 
 
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Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 85    Data Row: 905   Total Pages: 46   Display: Page     
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#StructureSubstanceCompoundActivityBioAssayLinks
OutcomeTypeValue [μM]
1
[SID134461981]
[CID56593836]
Ki 1e-06Displacement of [33P]ATP from human recombinant c-KIT domain after 20 mins by scintillation counting [AID623446, Type: Literature]
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2
[SID103175813]
[CID5329102]
Kd 0.00021Binding constant for KIT(V559D,V654A) kinase domain [AID435802, Type: Literature]
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3
[SID103175813]
[CID5329102]
Kd 0.00021Binding constant for KIT(V559D,V654A) kinase domain [AID624793, Type: Literature]
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4
[SID131277755]
[CID10138259]
Kd 0.00025Binding constant for KIT(V559D,V654A) kinase domain [AID624793, Type: Literature]
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5
[SID131277755]
[CID10138259]
Kd 0.00025Binding constant for KIT(V559D,V654A) kinase domain [AID435802, Type: Literature]
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6
[SID103592924]
[CID9933475]
Kd 0.00027Binding constant for KIT(V559D) kinase domain [AID624791, Type: Literature]
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7
[SID103175813]
[CID5329102]
Kd 0.00028Binding constant for KIT(V559D,T670I) kinase domain [AID435675, Type: Literature]
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8
[SID103175813]
[CID5329102]
Kd 0.00028Binding constant for KIT(V559D,T670I) kinase domain [AID624792, Type: Literature]
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9
[SID131277755]
[CID10138259]
Kd 0.00029Binding constant for KIT(L576P) kinase domain [AID624790, Type: Literature]
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10
[SID103592924]
[CID9933475]
Kd 0.00031Binding constant for KIT(V559D,V654A) kinase domain [AID624793, Type: Literature]
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11
[SID103592924]
[CID9933475]
Kd 0.00032Binding constant for KIT(V559D,T670I) kinase domain [AID624792, Type: Literature]
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12
[SID103175813]
[CID5329102]
Kd 0.00037Binding constant for KIT kinase domain [AID435410, Type: Literature]
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13
[SID103175813]
[CID5329102]
Kd 0.00037Binding affinity to human KIT incubated for 1 hr by kinase binding assay [AID599957, Type: Literature]
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14
[SID103175813]
[CID5329102]
Kd 0.00037Binding constant for KIT kinase domain [AID624786, Type: Literature]
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15
[SID103592924]
[CID9933475]
Kd 0.00038Binding constant for KIT kinase domain [AID624786, Type: Literature]
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16
[SID103175813]
[CID5329102]
Kd 0.00041Binding constant for KIT(V559D) kinase domain [AID624791, Type: Literature]
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17
[SID103175813]
[CID5329102]
Kd 0.00041Binding constant for KIT(V559D) kinase domain [AID435167, Type: Literature]
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18
[SID123092436]
[CID44259]
Kd 0.00043Binding constant for KIT(D816H) kinase domain [AID624788, Type: Literature]
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19
[SID136931825]
[CID9869779]
Kd 0.00046Binding constant for KIT(V559D) kinase domain [AID624791, Type: Literature]
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20
[SID123098392]
[CID6450551]
Kd 0.00049Binding constant for KIT(V559D) kinase domain [AID624791, Type: Literature]
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