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BioActivity Data for Targets
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BioActivity Outcomes:
Active(279)
 
 
BioAssay Types:
Literature(279)
 
 
BioActivity Types:
IC50(203)
 
 
Ki(40)
 
 
Substance Types:
Chemical(279)
 
 
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Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 33    Data Row: 279   Total Pages: 6   Display: Page     
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#StructureSubstanceCompoundActivityBioAssayLinks
OutcomeTypeValue [μM]
1
[SID103700367]
[CID44597383]
IC50 0.012Inhibition of indoleamine 2,3-dioxygenase in IFN-gamma-stimulated human HeLa cells assessed as kynurenine formation by spectrophotometry [AID439709, Type: Literature]
View
2
[SID103700254]
[CID11977720]
IC50 0.017Inhibition of indoleamine 2,3-dioxygenase in IFN-gamma-stimulated human HeLa cells assessed as kynurenine formation by spectrophotometry [AID439709, Type: Literature]
View
3
[SID103700211]
[CID11978511]
IC50 0.019Inhibition of indoleamine 2,3-dioxygenase in IFN-gamma-stimulated human HeLa cells assessed as kynurenine formation by spectrophotometry [AID439709, Type: Literature]
View
4
[SID103700349]
[CID11978742]
IC50 0.019Inhibition of indoleamine 2,3-dioxygenase in IFN-gamma-stimulated human HeLa cells assessed as kynurenine formation by spectrophotometry [AID439709, Type: Literature]
View
5
[SID103621382]
[CID24825243]
Ki 0.041Inhibition of human recombinant indoleamine 2,3-dioxygenase [AID384942, Type: Literature]
View
6
[SID104242225]
[CID49864297]
Ki 0.041Inhibition of human recombinant indoleamine-2,3-dioxygenase [AID500586, Type: Literature]
View
7
[SID103700272]
[CID11977838]
IC50 0.054Inhibition of indoleamine 2,3-dioxygenase in IFN-gamma-stimulated human HeLa cells assessed as kynurenine formation by spectrophotometry [AID439709, Type: Literature]
View
8
[SID103700367]
[CID44597383]
IC50 0.059Inhibition of N-terminal his-tagged human indoleamine 2,3-dioxygenase expressed in Escherichia coli assessed as N'-formylkynurenine formation by spectrophotometry [AID439708, Type: Literature]
View
9
[SID103700349]
[CID11978742]
IC50 0.06Inhibition of human IDO1 transfected in mouse P815B clone-6 cells by HPLC analysis [AID687187, Type: Literature]
View
10
[SID103700349]
[CID11978742]
IC50 0.067Inhibition of N-terminal his-tagged human indoleamine 2,3-dioxygenase expressed in Escherichia coli assessed as N'-formylkynurenine formation by spectrophotometry [AID439708, Type: Literature]
View
11
[SID163337181]
[CID60154723]
IC50 0.071Inhibition of human recombinant N-terminal His-tagged IDO1 (Ala2 to Gly403) overexpressed in Escherichia coli BL21 at pH 7.4 after 60 mins by HPLC analysis [AID687182, Type: Literature]
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12
[SID103700254]
[CID11977720]
IC50 0.073Inhibition of N-terminal his-tagged human indoleamine 2,3-dioxygenase expressed in Escherichia coli assessed as N'-formylkynurenine formation by spectrophotometry [AID439708, Type: Literature]
View
13
[SID163337181]
[CID60154723]
IC50 0.08Inhibition of human IDO1 transfected in mouse P815B clone-6 cells by HPLC analysis [AID687187, Type: Literature]
View
14
[SID104242226]
[CID24856336]
Ki 0.08Inhibition of human recombinant indoleamine-2,3-dioxygenase [AID500586, Type: Literature]
View
15
[SID104242227]
[CID49864298]
Ki 0.08Inhibition of human recombinant indoleamine-2,3-dioxygenase [AID500586, Type: Literature]
View
16
[SID103577973]
[CID44457253]
IC50 0.082Inhibition of purified human recombinant IDO [AID326467, Type: Literature]
View
17
[SID103700211]
[CID11978511]
IC50 0.086Inhibition of N-terminal his-tagged human indoleamine 2,3-dioxygenase expressed in Escherichia coli assessed as N'-formylkynurenine formation by spectrophotometry [AID439708, Type: Literature]
View
18
[SID103700255]
[CID5852646]
IC50 0.12Inhibition of indoleamine 2,3-dioxygenase in IFN-gamma-stimulated human HeLa cells assessed as kynurenine formation by spectrophotometry [AID439709, Type: Literature]
View
19
[SID103579812]
[CID44559102]
Ki 0.12Inhibition of human indoleamine 2,3-dioxygenase expressed in Escherichia coli by spectrophotometric activity assay [AID379168, Type: Literature]
View
20
[SID103578107]
[CID12239942]
IC50 0.121Inhibition of purified human recombinant IDO [AID326467, Type: Literature]
View
21
[SID103577977]
[CID24824612]
IC50 0.13Inhibition of purified human recombinant IDO [AID326467, Type: Literature]
View
22
[SID103579810]
[CID16091658]
Ki 0.14Inhibition of human indoleamine 2,3-dioxygenase expressed in Escherichia coli by spectrophotometric activity assay [AID379168, Type: Literature]
View
23
[SID103579810]
[CID16091658]
Ki 0.14Inhibition of human recombinant indoleamine 2,3-dioxygenase [AID384942, Type: Literature]
View
24
[SID103577976]
[CID44457255]
IC50 0.186Inhibition of purified human recombinant IDO [AID326467, Type: Literature]
View
25
[SID103578559]
[CID14034883]
IC50 0.19Inhibition of purified human recombinant IDO [AID326467, Type: Literature]
View
26
[SID103621449]
[CID152300]
Ki 0.19Inhibition of human recombinant indoleamine 2,3-dioxygenase [AID384942, Type: Literature]
View
27
[SID103621452]
[CID24825247]
Ki 0.2Inhibition of human recombinant indoleamine 2,3-dioxygenase [AID384942, Type: Literature]
View
28
[SID103707532]
[CID45487181]
IC50 0.2Inhibition of human recombinant IDO expressed in Escherichia coli BL21 AI [AID443993, Type: Literature]
View
29
[SID103621382]
[CID24825243]
Ki 0.21Inhibition of IDO1 (unknown origin) [AID734360, Type: Literature]
View
30
[SID103578028]
[CID72734]
IC50 0.214Inhibition of purified human recombinant IDO [AID326467, Type: Literature]
View
31
[SID103700335]
[CID44597278]
IC50 0.225Inhibition of indoleamine 2,3-dioxygenase in IFN-gamma-stimulated human HeLa cells assessed as kynurenine formation by spectrophotometry [AID439709, Type: Literature]
View
32
[SID103577981]
[CID24822271]
IC50 0.247Inhibition of purified human recombinant IDO [AID326467, Type: Literature]
View
33
[SID103578066]
[CID44457280]
IC50 0.252Inhibition of purified human recombinant IDO [AID326467, Type: Literature]
View
34
[SID103621516]
[CID24825249]
Ki 0.26Inhibition of human recombinant indoleamine 2,3-dioxygenase [AID384942, Type: Literature]
View
35
[SID103621451]
[CID24788785]
Ki 0.26Inhibition of human recombinant indoleamine 2,3-dioxygenase [AID384942, Type: Literature]
View
36
[SID103700213]
[CID11955091]
IC50 0.27Inhibition of indoleamine 2,3-dioxygenase in IFN-gamma-stimulated human HeLa cells assessed as kynurenine formation by spectrophotometry [AID439709, Type: Literature]
View
37
[SID103310959]
[CID8342]
IC50 0.28Inhibition of purified human recombinant IDO [AID326467, Type: Literature]
View
38
[SID163337181]
[CID60154723]
IC50 0.33Inhibition of human recombinant N-terminal His-tagged IDO1 (Ala2 to Gly403) overexpressed in Escherichia coli BL21 at pH 6.5 after 60 mins by HPLC analysis [AID687181, Type: Literature]
View
39
[SID103578145]
[CID21125239]
IC50 0.34Inhibition of purified human recombinant IDO [AID326467, Type: Literature]
View
40
[SID103578560]
[CID44457448]
IC50 0.361Inhibition of purified human recombinant IDO [AID326467, Type: Literature]
View
41
[SID103621450]
[CID24825246]
Ki 0.42Inhibition of human recombinant indoleamine 2,3-dioxygenase [AID384942, Type: Literature]
View
42
[SID103700272]
[CID11977838]
IC50 0.43Inhibition of N-terminal his-tagged human indoleamine 2,3-dioxygenase expressed in Escherichia coli assessed as N'-formylkynurenine formation by spectrophotometry [AID439708, Type: Literature]
View
43
[SID103707531]
[CID45487180]
IC50 0.45Inhibition of human recombinant IDO expressed in Escherichia coli BL21 AI [AID443993, Type: Literature]
View
44
[SID164142572]
[CID114918]
IC50 0.46Inhibition of human recombinant N-terminus 6X-histidine-tagged indoleamine 2,3-dioxygenase expressed in Escherichia coli assessed as inhibition of L-tryptophan to N-formylkynurenine formation measured as residual enzyme activity incubated for 15 mins prior to substrate addition measured after 30 mins by UV-vis spectrophotometric analysis relative to DMSO-treated control [AID728969, Type: Literature]
View
45
[SID103700399]
[CID5367120]
IC50 0.49Inhibition of indoleamine 2,3-dioxygenase in IFN-gamma-stimulated human HeLa cells assessed as kynurenine formation by spectrophotometry [AID439709, Type: Literature]
View
46
[SID103700213]
[CID11955091]
IC50 0.5Inhibition of N-terminal his-tagged human indoleamine 2,3-dioxygenase expressed in Escherichia coli assessed as N'-formylkynurenine formation by spectrophotometry [AID439708, Type: Literature]
View
47
[SID103578475]
[CID44457419]
IC50 0.512Inhibition of purified human recombinant IDO [AID326467, Type: Literature]
View
48
[SID103707641]
[CID45487224]
IC50 0.52Inhibition of human recombinant IDO expressed in Escherichia coli BL21 AI [AID443993, Type: Literature]
View
49
[SID103700255]
[CID5852646]
IC50 0.55Inhibition of N-terminal his-tagged human indoleamine 2,3-dioxygenase expressed in Escherichia coli assessed as N'-formylkynurenine formation by spectrophotometry [AID439708, Type: Literature]
View
50
[SID104245094]
[CID68342]
IC50 0.6Inhibition of indoleamine-2,3-dioxygenase in human A431 cells assessed as inhibition of IFN-gamma-stimulated kynurenine production [AID502207, Type: Literature]
View