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BioActivity Data for Targets
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BioActivity Outcomes:
Active(311)
 
 
BioAssay Types:
Literature(311)
 
 
BioActivity Types:
IC50(226)
 
 
Ki(41)
 
 
Kd(1)
 
 
Substance Types:
Chemical(311)
 
 
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Total Bioassays: 42    Data Row: 311   Total Pages: 16   Display: Page     
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#StructureSubstanceCompoundActivityBioAssayLinks
OutcomeTypeValue [μM]
1
[SID103274195]
[CID478573]
IC50 1.8e-05Inhibition of human IDO1 expressed in HEK293 cells assessed as kynurenine release after 5 hrs by spectrophotometry [AID1053471, Type: Literature]
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2
[SID103700367]
[CID44597383]
IC50 0.012Inhibition of indoleamine 2,3-dioxygenase in IFN-gamma-stimulated human HeLa cells assessed as kynurenine formation by spectrophotometry [AID439709, Type: Literature]
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3
[SID103700254]
[CID11977720]
IC50 0.017Inhibition of indoleamine 2,3-dioxygenase in IFN-gamma-stimulated human HeLa cells assessed as kynurenine formation by spectrophotometry [AID439709, Type: Literature]
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4
[SID103700211]
[CID11978511]
IC50 0.019Inhibition of indoleamine 2,3-dioxygenase in IFN-gamma-stimulated human HeLa cells assessed as kynurenine formation by spectrophotometry [AID439709, Type: Literature]
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5
[SID103700349]
[CID11978742]
IC50 0.019Inhibition of indoleamine 2,3-dioxygenase in IFN-gamma-stimulated human HeLa cells assessed as kynurenine formation by spectrophotometry [AID439709, Type: Literature]
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6
[SID103753306]
[CID478574]
IC50 0.023Inhibition of human IDO1 expressed in HEK293 cells assessed as kynurenine release after 5 hrs by spectrophotometry [AID1053471, Type: Literature]
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7
[SID194158814]
[CID76320783]
IC50 0.0243Inhibition of human IDO1 expressed in HEK293 cells assessed as kynurenine release after 5 hrs by spectrophotometry [AID1053471, Type: Literature]
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8
[SID194138110]
[CID478647]
IC50 0.0271Inhibition of human IDO1 expressed in HEK293 cells assessed as kynurenine release after 5 hrs by spectrophotometry [AID1053471, Type: Literature]
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9
[SID104242225]
[CID49864297]
Ki 0.041Inhibition of human recombinant indoleamine-2,3-dioxygenase [AID500586, Type: Literature]
View
10
[SID103621382]
[CID24825243]
Ki 0.041Inhibition of human recombinant indoleamine 2,3-dioxygenase [AID384942, Type: Literature]
View
11
[SID103274177]
[CID73549]
IC50 0.0537Inhibition of human IDO1 expressed in HEK293 cells assessed as kynurenine release after 5 hrs by spectrophotometry [AID1053471, Type: Literature]
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12
[SID103273712]
[CID478572]
IC50 0.0539Inhibition of human IDO1 expressed in HEK293 cells assessed as kynurenine release after 5 hrs by spectrophotometry [AID1053471, Type: Literature]
View
13
[SID103700272]
[CID11977838]
IC50 0.054Inhibition of indoleamine 2,3-dioxygenase in IFN-gamma-stimulated human HeLa cells assessed as kynurenine formation by spectrophotometry [AID439709, Type: Literature]
View
14
[SID103700367]
[CID44597383]
IC50 0.059Inhibition of N-terminal his-tagged human indoleamine 2,3-dioxygenase expressed in Escherichia coli assessed as N'-formylkynurenine formation by spectrophotometry [AID439708, Type: Literature]
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15
[SID103700349]
[CID11978742]
IC50 0.06Inhibition of human IDO1 transfected in mouse P815B clone-6 cells by HPLC analysis [AID687187, Type: Literature]
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16
[SID103700349]
[CID11978742]
IC50 0.067Inhibition of N-terminal his-tagged human indoleamine 2,3-dioxygenase expressed in Escherichia coli assessed as N'-formylkynurenine formation by spectrophotometry [AID439708, Type: Literature]
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17
[SID163337181]
[CID60154723]
IC50 0.071Inhibition of human recombinant N-terminal His-tagged IDO1 (Ala2 to Gly403) overexpressed in Escherichia coli BL21 at pH 7.4 after 60 mins by HPLC analysis [AID687182, Type: Literature]
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18
[SID103700254]
[CID11977720]
IC50 0.073Inhibition of N-terminal his-tagged human indoleamine 2,3-dioxygenase expressed in Escherichia coli assessed as N'-formylkynurenine formation by spectrophotometry [AID439708, Type: Literature]
View
19
[SID104242226]
[CID24856336]
Ki 0.08Inhibition of human recombinant indoleamine-2,3-dioxygenase [AID500586, Type: Literature]
View
20
[SID104242227]
[CID49864298]
Ki 0.08Inhibition of human recombinant indoleamine-2,3-dioxygenase [AID500586, Type: Literature]
View