Bookmark and Share
cyclin-dependent kinase 9 [Homo sapiens] [gi:4502747] - Target BioActivity Data
Filters: All Data » Active      
Filter selected
BioActivity Outcomes:
Active(167)
 
 
BioAssay Types:
Literature(166)
 
 
Confirmatory(1)
 
 
BioActivity Types:
IC50(103)
 
 
Kd(20)
 
 
Ki(20)
 
 
Substance Types:
Chemical(167)
 
 
Data download

Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 40    Data Row: 167   Total Pages: 4   Display: Page     
Sort: [Click the result table header to sort]
#StructureSubstanceCompoundActivityBioAssayLinks
OutcomeTypeValue [μM]
1
[SID103492722]
[CID44413509]
IC50 0.0025Inhibition of CDK9 [AID266569, Type: Literature]
View
2
[SID104234154]
[CID5287969]
Ki 0.003Inhibition of CDK9/Cyclin T (1 to 330 amino acid residues) (unknown origin) by differential scanning fluorimetry assay [AID723735, Type: Literature]
View
3
[SID104234154]
[CID5287969]
Ki 0.003Inhibition of CDK9 (unknown origin) [AID723739, Type: Literature]
View
4
[SID103229612]
[CID3025986]
Ki 0.004Inhibition of CDK9 (unknown origin) [AID723739, Type: Literature]
View
5
[SID103578264]
[CID23727982]
IC50 0.0056Inhibition of human recombinant CDK9/cyclin T expressed in insect cells [AID315302, Type: Literature]
View
6
[SID103578259]
[CID24801185]
IC50 0.0056Inhibition of human recombinant CDK9/cyclin T expressed in insect cells [AID315302, Type: Literature]
View
7
[SID103643679]
[CID11338033]
Kd 0.0058Binding constant for CDK9 kinase domain [AID624830, Type: Literature]
View
8
[SID103578262]
[CID23727981]
IC50 0.006Inhibition of human recombinant CDK9/cyclin T expressed in insect cells [AID315302, Type: Literature]
View
9
[SID164133474]
[CID44253323]
Ki 0.006Inhibition of CDK9/Cyclin T (1 to 330 amino acid residues) (unknown origin) by differential scanning fluorimetry assay [AID723735, Type: Literature]
View
10
[SID164133475]
[CID44253325]
Ki 0.006Inhibition of CDK9/Cyclin T (1 to 330 amino acid residues) (unknown origin) by differential scanning fluorimetry assay [AID723735, Type: Literature]
View
11
[SID104234154]
[CID5287969]
Kd 0.0064Binding constant for full-length CDK9 [AID435279, Type: Literature]
View
12
[SID104234154]
[CID5287969]
Kd 0.0064Binding constant for CDK9 kinase domain [AID624830, Type: Literature]
View
13
[SID103578263]
[CID24801697]
IC50 0.007Inhibition of human recombinant CDK9/cyclin T expressed in insect cells [AID315302, Type: Literature]
View
14
[SID103243222]
[CID44299148]
Ki 0.007Inhibition of CDK9/Cyclin T (1 to 330 amino acid residues) (unknown origin) by differential scanning fluorimetry assay [AID723735, Type: Literature]
View
15
[SID164147480]
[CID71720363]
Ki 0.007Inhibition of CDK9/Cyclin T (1 to 330 amino acid residues) (unknown origin) by differential scanning fluorimetry assay [AID723735, Type: Literature]
View
16
[SID164147481]
[CID71300299]
Ki 0.007Inhibition of CDK9/Cyclin T (1 to 330 amino acid residues) (unknown origin) by differential scanning fluorimetry assay [AID723735, Type: Literature]
View
17
[SID164130668]
[CID44253324]
Ki 0.008Inhibition of CDK9/Cyclin T (1 to 330 amino acid residues) (unknown origin) by differential scanning fluorimetry assay [AID723735, Type: Literature]
View
18
[SID164144686]
[CID44253465]
Ki 0.008Inhibition of CDK9/Cyclin T (1 to 330 amino acid residues) (unknown origin) by differential scanning fluorimetry assay [AID723735, Type: Literature]
View
19
[SID164136244]
[CID44253187]
Ki 0.011Inhibition of CDK9/Cyclin T (1 to 330 amino acid residues) (unknown origin) by differential scanning fluorimetry assay [AID723735, Type: Literature]
View
20
[SID164147481]
[CID71300299]
IC50 0.014Inhibition of human recombinant His6 tagged CDK9/CyclinT1 expressed in Sf21 insect cells after 40 mins by scintillation counting analysis [AID741495, Type: Literature]
View
21
[SID103501363]
[CID6918852]
Kd 0.015Binding constant for CDK9 kinase domain [AID624830, Type: Literature]
View
22
[SID103578267]
[CID24801699]
IC50 0.018Inhibition of human recombinant CDK9/cyclin T expressed in insect cells [AID315302, Type: Literature]
View
23
[SID164139129]
[CID44224280]
Ki 0.022Inhibition of CDK9/Cyclin T (1 to 330 amino acid residues) (unknown origin) by differential scanning fluorimetry assay [AID723735, Type: Literature]
View
24
[SID164136245]
[CID44253186]
Ki 0.026Inhibition of CDK9/Cyclin T (1 to 330 amino acid residues) (unknown origin) by differential scanning fluorimetry assay [AID723735, Type: Literature]
View
25
[SID103578312]
[CID11637090]
IC50 0.026Inhibition of human recombinant CDK9/cyclin T expressed in insect cells [AID315302, Type: Literature]
View
26
[SID103578350]
[CID9922607]
IC50 0.026Inhibition of human recombinant CDK9/cyclin T expressed in insect cells [AID315302, Type: Literature]
View
27
[SID103492759]
[CID44413527]
IC50 0.026Inhibition of CDK9 [AID266569, Type: Literature]
View
28
[SID164138786]
[CID49838820]
IC50 0.039Inhibition of CDK9/CyclinT1 (unknown origin) using (YSPTSPS)2KK as substrate [AID738800, Type: Literature]
View
29
[SID103609280]
[CID25190761]
IC50 0.043Inhibition of human recombinant CDK9/cyclin T expressed in baculovirus-infected insect cells [AID367871, Type: Literature]
View
30
[SID164147482]
[CID44253188]
Ki 0.043Inhibition of CDK9/Cyclin T (1 to 330 amino acid residues) (unknown origin) by differential scanning fluorimetry assay [AID723735, Type: Literature]
View
31
[SID103578215]
[CID24801183]
IC50 0.05Inhibition of human recombinant CDK9/cyclin T expressed in insect cells [AID315302, Type: Literature]
View
32
[SID103235175]
[CID3820]
IC50 0.064Inhibition of human recombinant CDK9/cyclin T expressed in insect cells assessed as incorporation of [gamma-33P]-ATP in to pRB fragment (773 to 928) substrate after 30 mins by scintillation counting [AID599805, Type: Literature]
View
33
[SID103229612]
[CID3025986]
Kd 0.076Binding constant for full-length CDK9 [AID435279, Type: Literature]
View
34
[SID103229612]
[CID3025986]
Kd 0.076Binding constant for CDK9 kinase domain [AID624830, Type: Literature]
View
35
[SID103243222]
[CID44299148]
Kd 0.1Binding constant for full-length CDK9 [AID435279, Type: Literature]
View
36
[SID103243222]
[CID44299148]
Kd 0.1Binding constant for CDK9 kinase domain [AID624830, Type: Literature]
View
37
[SID164144152]
[CID71579250]
IC50 0.1Inhibition of CDK9/CyclinT1 (unknown origin) using (YSPTSPS)2KK as substrate [AID738800, Type: Literature]
View
38
[SID164135740]
[CID71579251]
IC50 0.106Inhibition of CDK9/CyclinT1 (unknown origin) using (YSPTSPS)2KK as substrate [AID738800, Type: Literature]
View
39
[SID136945930]
[CID9842276]
IC50 0.107Inhibition of CDK9 in human HT29 cells assessed as reduction in RNA polymerase 2 expression [AID633248, Type: Literature]
View
40
[SID164144687]
[CID71719747]
Ki 0.11Inhibition of CDK9/Cyclin T (1 to 330 amino acid residues) (unknown origin) by differential scanning fluorimetry assay [AID723735, Type: Literature]
View
41
[SID103589440]
[CID25169529]
IC50 0.12Inhibition of CDK9-mediated RNA pol 2 phosphorylation at ser2 in human HCT116 cells after 16 hrs by HCS assay [AID409962, Type: Literature]
View
42
[SID160670567]
[CID46912953]
IC50 0.15Inhibition of human recombinant CDK9/cyclin T expressed in baculovirus-infected insect cells [AID682485, Type: Literature]
View
43
[SID164146896]
[CID71579248]
IC50 0.165Inhibition of CDK9/CyclinT1 (unknown origin) using (YSPTSPS)2KK as substrate [AID738800, Type: Literature]
View
44
[SID160708074]
[CID70697479]
IC50 0.18Inhibition of human recombinant CDK9/cyclin T expressed in baculovirus-infected insect cells [AID682485, Type: Literature]
View
45
[SID103491101]
[CID11314340]
Kd 0.18Binding constant for CDK9 kinase domain [AID624830, Type: Literature]
View
46
[SID103694306]
[CID11409972]
Kd 0.19Binding constant for full-length CDK9 [AID435279, Type: Literature]
View
47
[SID103694306]
[CID11409972]
Kd 0.19Binding constant for CDK9 kinase domain [AID624830, Type: Literature]
View
48
[SID103608911]
[CID25190763]
IC50 0.2Inhibition of human recombinant CDK9/cyclin T expressed in baculovirus-infected insect cells [AID367871, Type: Literature]
View
49
[SID103578175]
[CID24801700]
IC50 0.22Inhibition of human recombinant CDK9/cyclin T expressed in insect cells [AID315302, Type: Literature]
View
50
[SID131276151]
[CID54582100]
IC50 0.22Inhibition of human recombinant CDK9/cyclin T expressed in insect cells assessed as incorporation of [gamma-33P]-ATP in to pRB fragment (773 to 928) substrate after 30 mins by scintillation counting [AID599805, Type: Literature]
View