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multidrug resistance protein 1 [Homo sapiens] [gi:42741659] - Target BioActivity Data
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BioActivity Outcomes:
Probe(1)
 
 
Active(1617)
 
 
BioAssay Types:
Literature(660)
 
 
Confirmatory(452)
 
 
Screening(148)
 
 
Summary(1)
 
 
BioActivity Types:
EC50(672)
 
 
IC50(191)
 
 
Ki(13)
 
 
AC50(6)
 
 
Substance Types:
Chemical(1618)
 
 
 
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Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 86    Data Row: 1618   Total Pages: 81   Display: Page     
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#StructureSubstanceCompoundActivityBioAssayLinks
OutcomeTypeValue [μM]
1
[SID88095709]
[CID44640177]
Summary of High-throughput multiplex screening for ABC transporter inhibitors [AID1818, Type: summary]
View
2
[SID174525548]
[CID73357268]
EC50 0.00562SUPPLEMENTARY: Inhibition of P-glycoprotein expressed in MDR CCRF vcr1000 cells by daunorubicin efflux assay. Same assay as CHEMBL914418 [AID781331, Type: confirmatory]
View
3
[SID103510495]
[CID44420815]
EC50 0.006Inhibition of P-glycoprotein expressed in MDR CCRF vcr1000 cells by daunorubicin efflux assay [AID281137, Type: Literature]
View
4
[SID103168561]
[CID5351344]
IC50 0.0115Inhibition of MDR1 (unknown origin) transfected in human SKOV3 cells assessed as growth inhibition after 48 hrs by SRB assay [AID751512, Type: Literature]
View
5
[SID174510069]
[CID73352712]
EC50 0.01288SUPPLEMENTARY: Inhibition of P-glycoprotein expressed in MDR CCRF vcr1000 cells by daunorubicin efflux assay. Same assay as CHEMBL914418 [AID781331, Type: confirmatory]
View
6
[SID103510515]
[CID44420823]
EC50 0.013Inhibition of P-glycoprotein expressed in MDR CCRF vcr1000 cells by daunorubicin efflux assay [AID281137, Type: Literature]
View
7
[SID103511366]
[CID44421042]
EC50 0.014Inhibition of P-glycoprotein expressed in MDR CCRF vcr1000 cells by daunorubicin efflux assay [AID281137, Type: Literature]
View
8
[SID174504912]
[CID73351217]
EC50 0.01413SUPPLEMENTARY: Inhibition of P-glycoprotein expressed in MDR CCRF vcr1000 cells by daunorubicin efflux assay. Same assay as CHEMBL914418 [AID781331, Type: confirmatory]
View
9
[SID174525542]
[CID73357263]
EC50 0.01698SUPPLEMENTARY: Inhibition of P-glycoprotein expressed in MDR CCRF vcr1000 cells by daunorubicin efflux assay. Same assay as CHEMBL914418 [AID781331, Type: confirmatory]
View
10
[SID103511350]
[CID44421033]
EC50 0.017Inhibition of P-glycoprotein expressed in MDR CCRF vcr1000 cells by daunorubicin efflux assay [AID281137, Type: Literature]
View
11
[SID174525558]
[CID73357278]
EC50 0.01778SUPPLEMENTARY: Inhibition of P-glycoprotein expressed in MDR CCRF vcr1000 cells by daunorubicin efflux assay. Same assay as CHEMBL914418 [AID781331, Type: confirmatory]
View
12
[SID103511365]
[CID44421041]
EC50 0.018Inhibition of P-glycoprotein expressed in MDR CCRF vcr1000 cells by daunorubicin efflux assay [AID281137, Type: Literature]
View
13
[SID174515185]
[CID73354204]
EC50 0.0182SUPPLEMENTARY: Inhibition of P-glycoprotein expressed in MDR CCRF vcr1000 cells by daunorubicin efflux assay. Same assay as CHEMBL914418 [AID781331, Type: confirmatory]
View
14
[SID103511361]
[CID44421039]
EC50 0.019Inhibition of P-glycoprotein expressed in MDR CCRF vcr1000 cells by daunorubicin efflux assay [AID281137, Type: Literature]
View
15
[SID174489504]
[CID73346641]
EC50 0.01905SUPPLEMENTARY: Inhibition of P-glycoprotein expressed in MDR CCRF vcr1000 cells by daunorubicin efflux assay. Same assay as CHEMBL914418 [AID781331, Type: confirmatory]
View
16
[SID174520266]
[CID73355754]
EC50 0.0257SUPPLEMENTARY: Inhibition of P-glycoprotein expressed in MDR CCRF vcr1000 cells by daunorubicin efflux assay. Same assay as CHEMBL914418 [AID781331, Type: confirmatory]
View
17
[SID103511384]
[CID44421054]
EC50 0.026Inhibition of P-glycoprotein expressed in MDR CCRF vcr1000 cells by daunorubicin efflux assay [AID281137, Type: Literature]
View
18
[SID174504907]
[CID73351213]
EC50 0.02692SUPPLEMENTARY: Inhibition of P-glycoprotein expressed in MDR CCRF vcr1000 cells by daunorubicin efflux assay. Same assay as CHEMBL914418 [AID781331, Type: confirmatory]
View
19
[SID103306217]
[CID10004336]
EC50 0.027Inhibition of P-glycoprotein expressed in MDR CCRF vcr1000 cells by daunorubicin efflux assay [AID281137, Type: Literature]
View
20
[SID174517086]
[CID71524818]
IC50 0.0291Inhibition of MDR1 (unknown origin) transfected in human SKOV3 cells assessed as growth inhibition after 48 hrs by SRB assay [AID751512, Type: Literature]
View