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hepatocyte growth factor receptor isoform b p.. [gi:42741655] - Target BioActivity Data
Also known as: hepatocyte growth factor receptor isoform b precursor [Homo sapiens].
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BioActivity Outcomes:
Active(1289)
 
 
BioAssay Types:
Literature(1276)
 
 
BioActivity Types:
IC50(1032)
 
 
Kd(110)
 
 
Ki(101)
 
 
Substance Types:
Chemical(1289)
 
 
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Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 119    Data Row: 1289   Total Pages: 26   Display: Page     
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#StructureSubstanceCompoundActivityBioAssayLinks
OutcomeTypeValue [μM]
1
[SID104252247]
[CID24779724]
Kd 0.00019Binding constant for MET kinase domain [AID624794, Type: Literature]
View
2
[SID134448032]
[CID53310824]
IC50 0.0002Inhibition of human recombinant c-Met-catalyzed phosphorylation of N-biotinylated peptide (EQEDEPEGDYFEWLE-CONH2) by time-resolved fluorescence resonance energy transfer assay [AID605783, Type: Literature]
View
3
[SID103583760]
[CID10461815]
Kd 0.00027Binding constant for MET kinase domain [AID624794, Type: Literature]
View
4
[SID134434692]
[CID11851498]
IC50 0.0005Inhibition of human c-MET [AID614836, Type: Literature]
View
5
[SID103728028]
[CID11626560]
Kd 0.00055Binding constant for MET(M1250T) kinase domain [AID624795, Type: Literature]
View
6
[SID103583760]
[CID10461815]
Kd 0.00064Binding constant for MET(M1250T) kinase domain [AID624795, Type: Literature]
View
7
[SID134448165]
[CID16036535]
IC50 0.0007Inhibition of human recombinant c-Met-catalyzed phosphorylation of N-biotinylated peptide (EQEDEPEGDYFEWLE-CONH2) by time-resolved fluorescence resonance energy transfer assay [AID605783, Type: Literature]
View
8
[SID134450198]
[CID56672047]
IC50 0.0007Inhibition of human c-MET [AID614836, Type: Literature]
View
9
[SID134442369]
[CID11851497]
IC50 0.0007Inhibition of human c-MET [AID614836, Type: Literature]
View
10
[SID104252247]
[CID24779724]
Kd 0.00082Binding constant for MET(M1250T) kinase domain [AID624795, Type: Literature]
View
11
[SID136938397]
[CID57399640]
Kd 0.00082Binding constant for MET(Y1235D) kinase domain [AID624796, Type: Literature]
View
12
[SID103583760]
[CID10461815]
Kd 0.00083Binding constant for MET(Y1235D) kinase domain [AID624796, Type: Literature]
View
13
[SID103584803]
[CID24901691]
IC50 0.001Inhibition of human c-MET [AID614836, Type: Literature]
View
14
[SID103584804]
[CID11963059]
IC50 0.001Inhibition of human c-MET [AID614836, Type: Literature]
View
15
[SID103584892]
[CID24901693]
IC50 0.001Inhibition of human c-MET [AID614836, Type: Literature]
View
16
[SID103591621]
[CID25218742]
IC50 0.001Inhibition of human c-MET [AID614836, Type: Literature]
View
17
[SID103591623]
[CID25218744]
IC50 0.001Inhibition of human c-MET [AID614836, Type: Literature]
View
18
[SID103562944]
[CID9870238]
Ki 0.001Inhibition of human activated c-Met by PK/LDH coupled kinetic assay [AID363798, Type: Literature]
View
19
[SID103620917]
[CID44576886]
IC50 0.001Inhibition of human c-MET [AID614836, Type: Literature]
View
20
[SID103620969]
[CID44576916]
IC50 0.001Inhibition of human c-MET [AID614836, Type: Literature]
View
21
[SID136938397]
[CID57399640]
Kd 0.001Binding constant for MET(M1250T) kinase domain [AID624795, Type: Literature]
View
22
[SID134455445]
[CID11853013]
IC50 0.001Inhibition of human c-MET [AID614836, Type: Literature]
View
23
[SID134463355]
[CID53310690]
IC50 0.001Inhibition of human recombinant c-Met-catalyzed phosphorylation of N-biotinylated peptide (EQEDEPEGDYFEWLE-CONH2) by time-resolved fluorescence resonance energy transfer assay [AID605783, Type: Literature]
View
24
[SID134464439]
[CID56683784]
IC50 0.001Inhibition of human c-MET [AID614836, Type: Literature]
View
25
[SID163321008]
[CID24851953]
Ki 0.001Competitive inhibition of N-terminal His6-tagged recombinant human c-MET (974 to 1390 amino acids) by spectrophotometry [AID702351, Type: Literature]
View
26
[SID163334860]
[CID24851730]
IC50 0.001Antagonist activity at c-MET receptor in human A549 cells assessed as inhibition of autophosphorylation after 1 hr by ELISA [AID702349, Type: Literature]
View
27
[SID164148324]
[CID25013686]
IC50 0.001Inhibition of c-MET (unknown origin)-catalyzed N-biotinylated EQEDEPEGDYFEWLECONH2 phosphorylation by TR-FRET assay [AID728080, Type: Literature]
View
28
[SID164148325]
[CID45142457]
IC50 0.001Inhibition of c-MET (unknown origin)-catalyzed N-biotinylated EQEDEPEGDYFEWLECONH2 phosphorylation by TR-FRET assay [AID728080, Type: Literature]
View
29
[SID164148328]
[CID71601483]
IC50 0.001Inhibition of c-MET (unknown origin)-catalyzed N-biotinylated EQEDEPEGDYFEWLECONH2 phosphorylation by TR-FRET assay [AID728080, Type: Literature]
View
30
[SID103584893]
[CID24901694]
IC50 0.0011Inhibition of human c-MET [AID614836, Type: Literature]
View
31
[SID103584974]
[CID24764449]
Ki 0.0012Inhibition of human c-Met by HTRF assay [AID343240, Type: Literature]
View
32
[SID103584972]
[CID24901695]
IC50 0.0013Inhibition of human c-MET [AID614836, Type: Literature]
View
33
[SID103586812]
[CID24901689]
IC50 0.0013Inhibition of human c-MET [AID614836, Type: Literature]
View
34
[SID163334885]
[CID53361985]
Ki 0.0013Competitive inhibition of N-terminal His6-tagged recombinant human c-MET (974 to 1390 amino acids) by spectrophotometry [AID702351, Type: Literature]
View
35
[SID136938397]
[CID57399640]
Kd 0.0014Binding constant for MET kinase domain [AID624794, Type: Literature]
View
36
[SID103728028]
[CID11626560]
Kd 0.0015Binding constant for MET(Y1235D) kinase domain [AID624796, Type: Literature]
View
37
[SID103561614]
[CID11504713]
IC50 0.0015Inhibition of human recombinant c-Met expressed in insect cell-baculovirus expression system [AID314689, Type: Literature]
View
38
[SID103561614]
[CID11504713]
IC50 0.0015Inhibition of human c-MET [AID614836, Type: Literature]
View
39
[SID134461628]
[CID11851595]
IC50 0.0016Inhibition of human c-MET [AID614836, Type: Literature]
View
40
[SID103586813]
[CID24901690]
IC50 0.0018Inhibition of human c-MET [AID614836, Type: Literature]
View
41
[SID103586518]
[CID21081761]
IC50 0.0018Inhibition of human c-MET [AID614836, Type: Literature]
View
42
[SID103586519]
[CID21081770]
IC50 0.0019Inhibition of human c-MET [AID614836, Type: Literature]
View
43
[SID103484200]
[CID11525727]
Ki 0.002Inhibition of human activated c-Met by PK/LDH coupled kinetic assay [AID363798, Type: Literature]
View
44
[SID103484200]
[CID11525727]
IC50 0.002Inhibition of human c-MET [AID614836, Type: Literature]
View
45
[SID103620970]
[CID44576917]
IC50 0.002Inhibition of HGF-mediated c-Met phosphorylation in serum-starved human PC2 cells [AID408231, Type: Literature]
View
46
[SID103620969]
[CID44576916]
IC50 0.002Inhibition of HGF-mediated c-Met phosphorylation in serum-starved human PC2 cells [AID408231, Type: Literature]
View
47
[SID103620918]
[CID16736063]
IC50 0.002Inhibition of human c-MET [AID614836, Type: Literature]
View
48
[SID103620917]
[CID44576886]
IC50 0.002Inhibition of HGF-mediated c-Met phosphorylation in serum-starved human PC2 cells [AID408231, Type: Literature]
View
49
[SID103642300]
[CID21081477]
IC50 0.002Inhibition of human c-MET [AID614836, Type: Literature]
View
50
[SID103642357]
[CID21081469]
IC50 0.002Inhibition of human c-MET [AID614836, Type: Literature]
View