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thyroid hormone receptor beta [Homo sapiens] [gi:40806162] - Target BioActivity Data
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BioActivity Outcomes:
Probe(1)
 
 
Active(1700)
 
 
BioAssay Types:
Confirmatory(1180)
 
 
Literature(508)
 
 
Summary(6)
 
 
 
Screening(3)
 
 
BioActivity Types:
Potency(1186)
 
 
 
IC50(361)
 
 
Ki(64)
 
 
EC50(41)
 
 
Kd(25)
 
 
Substance Types:
Chemical(1701)
 
 
 
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Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 57    Data Row: 1701   Total Pages: 86   Display: Page     
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#StructureSubstanceCompoundActivityBioAssayLinks
OutcomeTypeValue [μM]
1
[SID87550851]
[CID5184800]
Tx-SRC2-2 Potency (uM) 1.4qHTS Assay for Inhibitors of the Interaction of Thyroid Hormone Receptor and Steroid Receptor Coregulator 2: Probe Summary [AID2512, Type: summary]
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2
[SID103219193]
[CID5804]
IC50 1.91e-05Inhibition of human thyroid hormone receptor beta 1 [AID299948, Type: Literature]
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3
[SID103219195]
[CID10456830]
IC50 2.51e-05Inhibition of human thyroid hormone receptor beta 1 [AID299948, Type: Literature]
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4
[SID103219116]
[CID5803]
IC50 4.79e-05Inhibition of human thyroid hormone receptor beta 1 [AID299948, Type: Literature]
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5
[SID103356078]
[CID22339645]
IC50 5.62e-05Inhibition of human thyroid hormone receptor beta 1 [AID299948, Type: Literature]
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6
[SID24275635]
[CID15991372]
Potency 5.623e-05Total Fluorescence Counterscreen for Inhibitors of the Interaction of Thyroid Hormone Receptor and Steroid Receptor Coregulator 2 [AID1479, Type: confirmatory]
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7
[SID103481478]
[CID9951790]
IC50 6e-05Inhibition of human TR-beta-1 by radioligand binding assay [AID261713, Type: Literature]
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8
[SID103570000]
[CID5920]
Kd 8.1e-05Displacement of [125I]T3 from human TRbeta receptor [AID323175, Type: Literature]
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9
[SID103218344]
[CID9933119]
IC50 9.5e-05Binding affinity at human thyroid hormone receptor beta-1 expressed in CHOK1 cells [AID299561, Type: Literature]
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10
[SID103218344]
[CID9933119]
IC50 9.55e-05Inhibition of human thyroid hormone receptor beta 1 [AID299948, Type: Literature]
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11
[SID103327605]
[CID9862248]
Kd 0.0001Binding affinity against human Thyroid hormone receptor beta 1 (hTRbeta1) using radiolabeled T3 [AID213183, Type: Literature]
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12
[SID103570000]
[CID5920]
Kd 0.0001Binding affinity against human Thyroid hormone receptor beta 1 (hTRbeta1) using radiolabeled T3 [AID213183, Type: Literature]
View
13
[SID103538695]
[CID6431911]
IC50 0.00011Inhibition of human thyroid hormone receptor beta 1 [AID299948, Type: Literature]
View
14
[SID103356191]
[CID22339458]
IC50 0.000112Inhibition of human thyroid hormone receptor beta 1 [AID299948, Type: Literature]
View
15
[SID103570000]
[CID5920]
Kd 0.00014Binding affinity towards thyroid hormone receptor (hTR beta 1) [AID213176, Type: Literature]
View
16
[SID103219085]
[CID10904700]
IC50 0.000151Inhibition of human thyroid hormone receptor beta 1 [AID299948, Type: Literature]
View
17
[SID103355713]
[CID10390904]
IC50 0.000195Inhibition of human thyroid hormone receptor beta 1 [AID299948, Type: Literature]
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18
[SID24407537]
[CID7522100]
Potency 0.0002Total Fluorescence Counterscreen for Inhibitors of the Interaction of Thyroid Hormone Receptor and Steroid Receptor Coregulator 2 [AID1479, Type: confirmatory]
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19
[SID103327605]
[CID9862248]
Kd 0.0002Binding affinity to human TRbeta1 [AID715452, Type: Literature]
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20
[SID103218312]
[CID9863447]
Ki 0.00024Displacement of [125I]3,5,3'-triiodo-L-thyronine His-tagged human recombinant TRbeta1 by scintillation proximity assay [AID345696, Type: Literature]
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