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serine/threonine-protein kinase B-raf [Homo s.. [gi:33188459] - Target BioActivity Data
Also known as: serine/threonine-protein kinase B-raf [Homo sapiens].
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BioActivity Outcomes:
Active(408)
 
 
BioAssay Types:
Literature(403)
 
 
Confirmatory(1)
 
 
BioActivity Types:
IC50(306)
 
 
Kd(87)
 
 
EC50(3)
 
 
Ki(1)
 
 
Substance Types:
Chemical(408)
 
 
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Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 44    Data Row: 408   Total Pages: 21   Display: Page     
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#StructureSubstanceCompoundActivityBioAssayLinks
OutcomeTypeValue [μM]
1
[SID103642962]
[CID11616462]
IC50 2e-05Inhibition of human recombinant B-Raf by fluorescence anisotropy [AID362268, Type: Literature]
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2
[SID103643282]
[CID11653652]
IC50 3e-05Inhibition of human recombinant B-Raf by fluorescence anisotropy [AID362268, Type: Literature]
View
3
[SID103643051]
[CID44587047]
IC50 4e-05Inhibition of human recombinant B-Raf by fluorescence anisotropy [AID362268, Type: Literature]
View
4
[SID103643223]
[CID44587190]
IC50 5e-05Inhibition of human recombinant B-Raf by fluorescence anisotropy [AID362268, Type: Literature]
View
5
[SID103643052]
[CID44587048]
IC50 9e-05Inhibition of human recombinant B-Raf by fluorescence anisotropy [AID362268, Type: Literature]
View
6
[SID103643222]
[CID11717001]
IC50 0.00013Inhibition of human recombinant B-Raf by fluorescence anisotropy [AID362268, Type: Literature]
View
7
[SID103642961]
[CID11522118]
IC50 0.00015Inhibition of human recombinant B-Raf by fluorescence anisotropy [AID362268, Type: Literature]
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8
[SID103623690]
[CID11316960]
Ki 0.00016Inhibition of N-terminus His-6 tagged human B-Raf expressed in baculovirus infected insect Sf9 cells [AID644002, Type: Literature]
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9
[SID103476069]
[CID11316960]
Kd 0.00016Binding affinity to human N-His6-tagged B-Raf expressed in Sf9 cells [AID632312, Type: Literature]
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10
[SID103643222]
[CID11717001]
Kd 0.00018Binding constant for BRAF(V600E) kinase domain [AID624947, Type: Literature]
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11
[SID103643222]
[CID11717001]
Kd 0.00019Binding constant for BRAF kinase domain [AID624946, Type: Literature]
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12
[SID103643341]
[CID11624965]
IC50 0.00022Inhibition of human recombinant B-Raf by fluorescence anisotropy [AID362268, Type: Literature]
View
13
[SID103643343]
[CID44587235]
IC50 0.00023Inhibition of human recombinant B-Raf by fluorescence anisotropy [AID362268, Type: Literature]
View
14
[SID103623690]
[CID11316960]
Kd 0.0003Binding affinity at bRaf kinase in fluorescent ligand displacement assay [AID258282, Type: Literature]
View
15
[SID103737886]
[CID44226449]
IC50 0.00032Inhibition of human recombinant B-Raf expressed in Sf9 cells assessed as inhibition of Mek1 phosphorylation [AID469343, Type: Literature]
View
16
[SID103738109]
[CID46880076]
IC50 0.00032Inhibition of human recombinant B-Raf expressed in Sf9 cells assessed as inhibition of Mek1 phosphorylation [AID469343, Type: Literature]
View
17
[SID103738155]
[CID46880102]
IC50 0.00032Inhibition of human recombinant B-Raf expressed in Sf9 cells assessed as inhibition of Mek1 phosphorylation [AID469343, Type: Literature]
View
18
[SID103738156]
[CID46880103]
IC50 0.00032Inhibition of human recombinant B-Raf expressed in Sf9 cells assessed as inhibition of Mek1 phosphorylation [AID469343, Type: Literature]
View
19
[SID103738157]
[CID46880104]
IC50 0.00032Inhibition of human recombinant B-Raf expressed in Sf9 cells assessed as inhibition of Mek1 phosphorylation [AID469343, Type: Literature]
View
20
[SID103738216]
[CID46880137]
IC50 0.00032Inhibition of human recombinant B-Raf expressed in Sf9 cells assessed as inhibition of Mek1 phosphorylation [AID469343, Type: Literature]
View