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Inhibitor of nuclear factor kappa-B kinase su.. [gi:317373368] - Target BioActivity Data
Also known as: Inhibitor of nuclear factor kappa-B kinase subunit alpha; I-kappa-B kinase alpha; IKK-A; IKK-alpha; IkBKA; IkappaB kinase; Conserved helix-loop-helix ubiquitous kinase; I-kappa-B kinase 1; IKK1; Nuclear factor NF-kappa-B inhibitor kinase alpha; NFKBIKA; Transcription factor 16; TCF-16.
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BioActivity Outcomes:
Active(178)
 
 
BioAssay Types:
Literature(178)
 
 
BioActivity Types:
IC50(145)
 
 
Kd(17)
 
 
Ki(1)
 
 
Substance Types:
Chemical(178)
 
 
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Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 33    Data Row: 178   Total Pages: 9   Display: Page     
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#StructureSubstanceCompoundActivityBioAssayLinks
OutcomeTypeValue [μM]
1
[SID103243222]
[CID44299148]
Kd 0.0058Binding constant for IKK-alpha kinase domain [AID624832, Type: Literature]
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2
[SID123092436]
[CID44259]
Kd 0.0058Binding constant for IKK-alpha kinase domain [AID624832, Type: Literature]
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3
[SID164133368]
[CID71717270]
Kd 0.009Binding constant for IKK-alpha kinase domain [AID624832, Type: Literature]
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4
[SID103722924]
[CID126565]
Kd 0.009Binding constant for IKK-alpha kinase domain [AID624832, Type: Literature]
View
5
[SID103652167]
[CID44591575]
IC50 0.01259Inhibition of human recombinant IKK1 [AID354255, Type: Literature]
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6
[SID103476101]
[CID44406565]
IC50 0.03Inhibitory activity against IKK1 [AID258073, Type: Literature]
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7
[SID103476152]
[CID44406586]
IC50 0.03Inhibitory activity against IKK1 [AID258073, Type: Literature]
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8
[SID103476152]
[CID44406586]
IC50 0.03Inhibitory activity against IKK complex isolated from HeLa cells [AID258074, Type: Literature]
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9
[SID103652012]
[CID44591532]
IC50 0.03162Inhibition of human recombinant IKK1 [AID354255, Type: Literature]
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10
[SID103243222]
[CID44299148]
IC50 0.039Inhibition of human recombinant IKK-alpha expressed in insect Sf21 cells using phospho-Ulight-IkappaB-alpha as substrate at 30 uM [AID590191, Type: Literature]
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11
[SID123092436]
[CID44259]
IC50 0.039Inhibition of human recombinant IKK-alpha expressed in insect Sf21 cells using phospho-Ulight-IkappaB-alpha as substrate at 30 uM [AID590191, Type: Literature]
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12
[SID103476101]
[CID44406565]
IC50 0.04Inhibitory activity against IKK complex isolated from HeLa cells [AID258074, Type: Literature]
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13
[SID103476285]
[CID44406635]
IC50 0.04Inhibitory activity against IKK complex isolated from HeLa cells [AID258074, Type: Literature]
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14
[SID103694306]
[CID11409972]
Kd 0.041Binding constant for IKK-alpha kinase domain [AID624832, Type: Literature]
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15
[SID103476214]
[CID44406614]
IC50 0.05Inhibitory activity against IKK complex isolated from HeLa cells [AID258074, Type: Literature]
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16
[SID103652088]
[CID23648953]
IC50 0.05012Inhibition of human recombinant IKK1 [AID354255, Type: Literature]
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17
[SID103476099]
[CID9549298]
IC50 0.07Inhibitory activity against IKK complex isolated from HeLa cells [AID258074, Type: Literature]
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18
[SID103522292]
[CID16047968]
IC50 0.07943Inhibition of human recombinant GST-IKKalpha by TR-FRET assay [AID290819, Type: Literature]
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19
[SID103475883]
[CID44406419]
IC50 0.08Inhibitory activity against IKK complex isolated from HeLa cells [AID258074, Type: Literature]
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20
[SID103476289]
[CID44406636]
IC50 0.1Inhibitory activity against IKK complex isolated from HeLa cells [AID258074, Type: Literature]
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