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epidermal growth factor receptor isoform a pr.. [gi:29725609] - Target BioActivity Data
Also known as: epidermal growth factor receptor isoform a precursor [Homo sapiens].
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BioActivity Outcomes:
Probe(1)
 
 
Active(2978)
 
 
BioAssay Types:
Literature(2792)
 
 
Confirmatory(166)
 
 
Summary(10)
 
 
 
BioActivity Types:
IC50(2143)
 
 
 
Kd(558)
 
 
Ki(40)
 
 
Potency(23)
 
 
EC50(8)
 
 
Substance Types:
Chemical(2979)
 
 
 
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Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 322    Data Row: 2979   Total Pages: 149   Display: Page     
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#StructureSubstanceCompoundActivityBioAssayLinks
OutcomeTypeValue [μM]
1
[SID22409543]
[CID2303746]
EGFR IC50 0.7079Quantitative High-Throughput Screen for Inhibitors of the ERK Signaling Pathway using a Homogeneous Screening Assay: Summary [AID1742, Type: summary]
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2
[SID103257428]
[CID5328245]
IC50 3e-06Inhibition of tyrosine kinase activity of Epidermal growth factor receptor from human A431 carcinoma cells [AID69415, Type: Literature]
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3
[SID103257455]
[CID2428]
IC50 8e-06Inhibition of tyrosine kinase activity of Epidermal growth factor receptor from human A431 carcinoma cells [AID69415, Type: Literature]
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4
[SID103433753]
[CID5328234]
IC50 1e-05Inhibition of tyrosine kinase activity of Epidermal growth factor receptor from human A431 carcinoma cells [AID69415, Type: Literature]
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5
[SID103432958]
[CID2427]
IC50 2.5e-05Inhibition of tyrosine kinase activity of Epidermal growth factor receptor from human A431 carcinoma cells [AID69415, Type: Literature]
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6
[SID103200288]
[CID4705]
IC50 2.5e-05Inhibition of tyrosine kinase activity of Epidermal growth factor receptor from human A431 cells [AID69402, Type: Literature]
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7
[SID103200288]
[CID4705]
IC50 2.9e-05Inhibition of Epidermal growth factor receptor from human A431 cell membranes [AID66446, Type: Literature]
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8
[SID103460666]
[CID10362209]
IC50 3.7e-05Inhibition of EGF Receptor autophosphorylation in A431 cell lysate [AID241077, Type: Literature]
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9
[SID103460717]
[CID9952784]
IC50 7e-05Inhibition of EGF Receptor autophosphorylation in A431 cell lysate [AID241077, Type: Literature]
View
10
[SID103441767]
[CID9915743]
IC50 8e-05Inhibition of human EGFR in presence of 1 uM ATP [AID295762, Type: Literature]
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11
[SID103238923]
[CID5328253]
IC50 8.91e-05Inhibition of human recombinant EGFR [AID345876, Type: Literature]
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12
[SID103244983]
[CID123631]
IC50 0.0001Inhibition of wild type EGFR (unknown origin) after 1.5 hrs by FRET-based Z'Lyte assay [AID748091, Type: Literature]
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13
[SID103244983]
[CID123631]
IC50 0.0001Inhibition of wild type EGFR (unknown origin) using Tyr 4 peptide as substrate after 1.5 hrs by FRET based Z'-lyte assay [AID761603, Type: Literature]
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14
[SID103202250]
[CID156414]
Kd 0.0001Binding constant for EGFR(T790M) kinase domain [AID625007, Type: Literature]
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15
[SID103304089]
[CID5328045]
IC50 0.0001Inhibition of Epidermal growth factor receptor from A431 cells [AID66603, Type: Literature]
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16
[SID103768626]
[CID10184653]
Kd 0.0001Binding constant for EGFR(G719C) kinase domain [AID624998, Type: Literature]
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17
[SID103768626]
[CID10184653]
Kd 0.00011Binding constant for EGFR(E746-A750del) kinase domain [AID624997, Type: Literature]
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18
[SID103460812]
[CID21080010]
IC50 0.00011Inhibition of EGF Receptor autophosphorylation in A431 cell lysate [AID241077, Type: Literature]
View
19
[SID103460534]
[CID10320940]
IC50 0.00012Inhibition of EGF Receptor autophosphorylation in A431 cell lysate [AID241077, Type: Literature]
View
20
[SID103304190]
[CID2426]
IC50 0.00012Inhibition of tyrosine kinase activity of Epidermal growth factor receptor from human A431 carcinoma cells [AID69415, Type: Literature]
View