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serine/threonine-protein kinase PLK1 [Homo sa.. [gi:21359873] - Target BioActivity Data
Also known as: serine/threonine-protein kinase PLK1 [Homo sapiens].
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BioActivity Outcomes:
Active(11190)
 
 
BioAssay Types:
Confirmatory(10304)
 
 
Screening(689)
 
 
Literature(195)
 
 
BioActivity Types:
Potency(10204)
 
 
IC50(200)
 
 
EC50(30)
 
 
Kd(15)
 
 
Ki(3)
 
 
Substance Types:
Chemical(11190)
 
 
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Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 44    Data Row: 11190   Total Pages: 560   Display: Page     
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#StructureSubstanceCompoundActivityBioAssayLinks
OutcomeTypeValue [μM]
1
[SID136925373]
[CID15983966]
Kd 9.4e-05Binding constant for PLK1 kinase domain [AID624975, Type: Literature]
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2
[SID103624610]
[CID11364421]
Kd 0.00019Binding constant for PLK1 kinase domain [AID624975, Type: Literature]
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3
[SID103508344]
[CID11957417]
IC50 0.0008Inhibition of human PLK1 kinase domain expressed in baculovirus-infected Trichoplusia ni cells by scintillation proximity assay [AID418643, Type: Literature]
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4
[SID103624610]
[CID11364421]
IC50 0.00083Competitive inhibition of human PLK1 in presence of ATP [AID718976, Type: Literature]
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5
[SID104249696]
[CID10461508]
IC50 0.00087Competitive inhibition of human PLK1 in presence of ATP [AID718976, Type: Literature]
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6
[SID134453399]
[CID25263120]
IC50 0.001Inhibition of human PLK1 kinase domain expressed in baculovirus-infected Trichoplusia ni cells by scintillation proximity assay [AID418643, Type: Literature]
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7
[SID174491504]
[CID25253525]
IC50 0.001Inhibition of PLK1 (unknown origin) using biotin-AGAGTVPESIHSFIGDGLV as substrate by TR-FRET assay [AID753523, Type: Literature]
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8
[SID174491506]
[CID57970023]
IC50 0.001Inhibition of PLK1 (unknown origin) using biotin-AGAGTVPESIHSFIGDGLV as substrate by TR-FRET assay [AID753523, Type: Literature]
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9
[SID103612637]
[CID25263118]
IC50 0.001Inhibition of human PLK1 kinase domain expressed in baculovirus-infected Trichoplusia ni cells by scintillation proximity assay [AID418643, Type: Literature]
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10
[SID174512134]
[CID71654873]
IC50 0.001Inhibition of PLK1 (unknown origin) using biotin-AGAGTVPESIHSFIGDGLV as substrate by TR-FRET assay [AID753523, Type: Literature]
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11
[SID174517180]
[CID53357478]
IC50 0.002Inhibition of PLK1 (unknown origin) using biotin-AGAGTVPESIHSFIGDGLV as substrate by TR-FRET assay [AID753523, Type: Literature]
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12
[SID174517181]
[CID25252909]
IC50 0.002Inhibition of PLK1 (unknown origin) using biotin-AGAGTVPESIHSFIGDGLV as substrate by TR-FRET assay [AID753523, Type: Literature]
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13
[SID103610848]
[CID9826308]
IC50 0.002Inhibition of human PLK1 kinase domain expressed in baculovirus-infected Trichoplusia ni cells by scintillation proximity assay [AID418643, Type: Literature]
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14
[SID103610915]
[CID25263092]
IC50 0.002Inhibition of human PLK1 kinase domain expressed in baculovirus-infected Trichoplusia ni cells by scintillation proximity assay [AID418643, Type: Literature]
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15
[SID134437919]
[CID16051023]
IC50 0.002Inhibition of human PLK1 kinase domain expressed in baculovirus-infected Trichoplusia ni cells by scintillation proximity assay [AID418643, Type: Literature]
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16
[SID123089933]
[CID16050925]
IC50 0.002Inhibition of human PLK1 kinase domain expressed in baculovirus-infected Trichoplusia ni cells by scintillation proximity assay [AID418643, Type: Literature]
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17
[SID136922934]
[CID57391401]
IC50 0.003Inhibition of human PLK1 kinase domain expressed in baculovirus-infected Trichoplusia ni cells by scintillation proximity assay [AID418643, Type: Literature]
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18
[SID136932653]
[CID25263125]
IC50 0.003Inhibition of human PLK1 kinase domain expressed in baculovirus-infected Trichoplusia ni cells by scintillation proximity assay [AID418643, Type: Literature]
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19
[SID136936063]
[CID16050921]
IC50 0.003Inhibition of human PLK1 kinase domain expressed in baculovirus-infected Trichoplusia ni cells by scintillation proximity assay [AID418643, Type: Literature]
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20
[SID103612791]
[CID25263119]
IC50 0.003Inhibition of human PLK1 kinase domain expressed in baculovirus-infected Trichoplusia ni cells by scintillation proximity assay [AID418643, Type: Literature]
View