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peroxisome proliferator-activated receptor ga.. [gi:20336229] - Target BioActivity Data
Also known as: peroxisome proliferator-activated receptor gamma isoform 2 [Homo sapiens].
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BioActivity Outcomes:
Probe(1)
 
 
Active(8104)
 
 
BioAssay Types:
Literature(3111)
 
 
Screening(3040)
 
 
Confirmatory(441)
 
 
BioActivity Types:
EC50(2069)
 
 
IC50(1002)
 
 
Ki(153)
 
 
Kd(15)
 
 
Substance Types:
Chemical(8105)
 
 
 
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Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 330    Data Row: 8105   Total Pages: 406   Display: Page     
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#StructureSubstanceCompoundActivityBioAssayLinks
OutcomeTypeValue [μM]
1
[SID124349301]
[CID53239856]
Late stage assay provider counterscreen results from the probe development effort to identify non-agonists of the peroxisome proliferator-activated receptor gamma (PPARg): chemiluminescence-based biochemical western blot assay for inhibitors of phosphorylation of PPARG protein levels [AID504938, Type: other]
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2
[SID134447814]
[CID56669690]
EC50 1e-07Transactivation of human PPARgamma expressed in human HepG2 cells co-transfected with PPRE3-TK-Luc by luciferase reporter gene assay [AID610311, Type: Literature]
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3
[SID134436215]
[CID56659348]
EC50 2e-07Transactivation of human PPARgamma expressed in human HepG2 cells co-transfected with PPRE3-TK-Luc by luciferase reporter gene assay [AID610311, Type: Literature]
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4
[SID134459372]
[CID56679849]
EC50 3e-07Transactivation of human PPARgamma expressed in human HepG2 cells co-transfected with PPRE3-TK-Luc by luciferase reporter gene assay [AID610311, Type: Literature]
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5
[SID134436214]
[CID56659347]
EC50 1.5e-06Transactivation of human PPARgamma expressed in human HepG2 cells co-transfected with PPRE3-TK-Luc by luciferase reporter gene assay [AID610311, Type: Literature]
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6
[SID134455510]
[CID53233135]
EC50 1.8e-05Transactivation of human PPARgamma expressed in human HepG2 cells co-transfected with PPRE3-TK-Luc by luciferase reporter gene assay [AID610311, Type: Literature]
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7
[SID134447813]
[CID56669689]
EC50 5e-05Transactivation of human PPARgamma expressed in human HepG2 cells co-transfected with PPRE3-TK-Luc by luciferase reporter gene assay [AID610311, Type: Literature]
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8
[SID103521630]
[CID25263407]
EC50 0.0001Agonist activity at human PPARgamma in HepG2 cells by PPAR-GAL4 transactivation assay [AID289933, Type: Literature]
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9
[SID103521626]
[CID25263404]
EC50 0.00019Agonist activity at human PPARgamma in HepG2 cells by PPAR-GAL4 transactivation assay [AID289933, Type: Literature]
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10
[SID103569797]
[CID446642]
EC50 0.0002Effective concentration against human peroxisome proliferator activated receptor gamma in Gal4 transactivation assay [AID240313, Type: Literature]
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11
[SID103569797]
[CID446642]
EC50 0.00028Agonist activity at human PPARgamma [AID330492, Type: Literature]
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12
[SID103521625]
[CID25263403]
EC50 0.0003Agonist activity at human PPARgamma in HepG2 cells by PPAR-GAL4 transactivation assay [AID289933, Type: Literature]
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13
[SID103521628]
[CID25263406]
EC50 0.00031Agonist activity at human PPARgamma in HepG2 cells by PPAR-GAL4 transactivation assay [AID289933, Type: Literature]
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14
[SID103324541]
[CID170364]
EC50 0.00034Agonist activity for Human PPAR gamma receptor in transcriptional activation assay [AID91246, Type: Literature]
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15
[SID103521627]
[CID25263405]
EC50 0.00036Agonist activity at human PPARgamma in HepG2 cells by PPAR-GAL4 transactivation assay [AID289933, Type: Literature]
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16
[SID124349300]
IC50 0.00037Late stage assay provider results from the probe development effort to identify non-agonists of the peroxisome proliferator-activated receptor gamma (PPARg): TR-FRET-based biochemical dose response competitive binding lanthascreen assay for non-agonists of the PPARg [AID504943, Type: confirmatory]
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17
[SID103261196]
[CID18944089]
Ki 0.0004inhibition of [125I]SB 236636 binding to human PPAR gamma receptor [AID156385, Type: confirmatory]
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18
[SID103316922]
[CID44331685]
EC50 0.0005Agonistic transcriptional activity in CV-1 cells expressing Gal4-PPAR gamma chimera [AID156798, Type: Literature]
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19
[SID104223102]
EC50 0.0005Late stage assay provider results from the probe development effort to identify non-agonists of the peroxisome proliferator-activated receptor gamma (PPARg): Luminescence-based cell-based dose response assay to identify transactivation inhibitor of PPRE (PPARG response element) [AID504939, Type: confirmatory]
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20
[SID134461452]
[CID44132175]
EC50 0.000501Partial agonist activity at human PPARgamma by luciferase reporter gene assay [AID617443, Type: Literature]
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