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BioActivity Data for Targets
Filters: All Data » Active      
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BioActivity Outcomes:
Active(171)
 
 
BioAssay Types:
Literature(159)
 
 
BioActivity Types:
IC50(125)
 
 
Kd(12)
 
 
Ki(8)
 
 
Substance Types:
Chemical(171)
 
 
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Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 21    Data Row: 171   Total Pages: 4   Display: Page     
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#StructureSubstanceCompoundActivityBioAssayLinks
OutcomeTypeValue [μM]
1
[SID103583025]
[CID44560005]
IC50 0.0005Inhibition of tubulin polymerization [AID270819, Type: Literature]
View
2
[SID103168561]
[CID5351344]
Ki 0.003Displacement of [3H]colchicine from tubulin [AID256882, Type: Literature]
View
3
[SID103474446]
[CID44405621]
Ki 0.01Displacement of [3H]colchicine from tubulin [AID256882, Type: Literature]
View
4
[SID103480841]
[CID44408260]
IC50 0.01Displacement of [3H]colchicine from tubulin at 65 nM [AID261214, Type: Literature]
View
5
[SID103168561]
[CID5351344]
IC50 0.0129Displacement of [3H]colchicine from tubulin by scintillation proximity assay [AID265408, Type: Literature]
View
6
[SID103474497]
[CID11554148]
Ki 0.02Displacement of [3H]colchicine from tubulin [AID256882, Type: Literature]
View
7
[SID103730344]
[CID6445562]
Kd 0.021Binding constant for ERBB4 kinase domain [AID435797, Type: Literature]
View
8
[SID103202250]
[CID156414]
Kd 0.029Binding constant for ERBB4 kinase domain [AID435797, Type: Literature]
View
9
[SID103168561]
[CID5351344]
IC50 0.03Displacement of [3H]colchicine from tubulin at 65 nM [AID261214, Type: Literature]
View
10
[SID103480705]
[CID11668206]
IC50 0.03Displacement of [3H]colchicine from tubulin at 65 nM [AID261214, Type: Literature]
View
11
[SID103480706]
[CID44408198]
IC50 0.03Displacement of [3H]colchicine from tubulin at 65 nM [AID261214, Type: Literature]
View
12
[SID103480712]
[CID11258149]
IC50 0.03Displacement of [3H]colchicine from tubulin at 65 nM [AID261214, Type: Literature]
View
13
[SID103474440]
[CID44405616]
Ki 0.05Displacement of [3H]colchicine from tubulin [AID256882, Type: Literature]
View
14
[SID103177479]
[CID208908]
Kd 0.054Binding constant for ERBB4 kinase domain [AID435797, Type: Literature]
View
15
[SID103501621]
[CID3062316]
Kd 0.055Binding constant for ERBB4 kinase domain [AID435797, Type: Literature]
View
16
[SID103474430]
[CID11189667]
Ki 0.06Displacement of [3H]colchicine from tubulin [AID256882, Type: Literature]
View
17
[SID103480840]
[CID44408259]
IC50 0.075Displacement of [3H]colchicine from tubulin at 65 nM [AID261214, Type: Literature]
View
18
[SID103473889]
[CID11166006]
Ki 0.1Displacement of [3H]colchicine from tubulin [AID256882, Type: Literature]
View
19
[SID103474431]
[CID11247827]
Ki 0.16Displacement of [3H]colchicine from tubulin [AID256882, Type: Literature]
View
20
[SID103480698]
[CID44408195]
IC50 0.19Displacement of [3H]colchicine from tubulin at 65 nM [AID261214, Type: Literature]
View
21
[SID103177459]
[CID176870]
Kd 0.23Binding constant for ERBB4 kinase domain [AID435797, Type: Literature]
View
22
[SID103641275]
[CID9874913]
Kd 0.26Binding constant for ERBB4 kinase domain [AID435797, Type: Literature]
View
23
[SID103480874]
[CID44408278]
IC50 0.39Displacement of [3H]colchicine from tubulin at 65 nM [AID261214, Type: Literature]
View
24
[SID103481086]
[CID44408383]
IC50 0.39Displacement of [3H]colchicine from tubulin at 65 nM [AID261214, Type: Literature]
View
25
[SID103244983]
[CID123631]
Kd 0.41Binding constant for ERBB4 kinase domain [AID435797, Type: Literature]
View
26
[SID103502389]
[CID16007391]
Kd 0.47Binding constant for ERBB4 kinase domain [AID435797, Type: Literature]
View
27
[SID103194628]
[CID3081361]
Kd 0.48Binding constant for ERBB4 kinase domain [AID435797, Type: Literature]
View
28
[SID103177124]
[CID6167]
IC50 0.5Inhibition of [3H]colchicine binding to beta tubulin [AID270966, Type: Literature]
View
29
[SID103480689]
[CID44408191]
IC50 0.5Inhibition of tubulin polymerization [AID261211, Type: Literature]
View
30
[SID103500654]
[CID16090892]
IC50 0.64Inhibition of tubulin polymerization [AID273280, Type: Literature]
View
31
[SID103481067]
[CID44408372]
IC50 0.7Inhibition of tubulin polymerization [AID261211, Type: Literature]
View
32
[SID103480712]
[CID11258149]
IC50 0.7Inhibition of tubulin polymerization [AID261211, Type: Literature]
View
33
[SID103498776]
[CID16086295]
IC50 0.75Inhibition of [3H]colchicine binding to beta tubulin [AID270966, Type: Literature]
View
34
[SID103498780]
[CID16086305]
IC50 0.75Inhibition of [3H]colchicine binding to beta tubulin [AID270966, Type: Literature]
View
35
[SID103243222]
[CID44299148]
Kd 0.77Binding constant for ERBB4 kinase domain [AID435797, Type: Literature]
View
36
[SID103492159]
[CID11552708]
IC50 0.8Inhibition of tubulin polymerization [AID273280, Type: Literature]
View
37
[SID103492158]
[CID11610751]
IC50 0.86Inhibition of tubulin polymerization [AID273280, Type: Literature]
View
38
[SID103500614]
[CID16090898]
IC50 0.97Inhibition of tubulin polymerization [AID273280, Type: Literature]
View
39
[SID103499003]
[CID1068397]
IC50 1Inhibition of [3H]colchicine binding to beta tubulin [AID270966, Type: Literature]
View
40
[SID103480705]
[CID11668206]
IC50 1Inhibition of tubulin polymerization [AID261211, Type: Literature]
View
41
[SID103498701]
[CID164454]
IC50 1.1Inhibition of tubulin polymerization [AID270819, Type: Literature]
View
42
[SID103500621]
[CID16090890]
IC50 1.1Inhibition of tubulin polymerization [AID273280, Type: Literature]
View
43
[SID103500632]
[CID16090891]
IC50 1.1Inhibition of tubulin polymerization [AID273280, Type: Literature]
View
44
[SID103500680]
[CID16090893]
IC50 1.1Inhibition of tubulin polymerization [AID273280, Type: Literature]
View
45
[SID103492190]
[CID11516867]
IC50 1.1Inhibition of tubulin polymerization [AID273280, Type: Literature]
View
46
[SID103501257]
[CID16215971]
IC50 1.1Inhibition of tubulin polymerization [AID271658, Type: Literature]
View
47
[SID103489398]
[CID44412095]
IC50 1.16Displacement of [3H]colchicine from tubulin by scintillation proximity assay [AID265408, Type: Literature]
View
48
[SID103480874]
[CID44408278]
IC50 1.2Inhibition of tubulin polymerization [AID261211, Type: Literature]
View
49
[SID103491713]
[CID11509549]
IC50 1.2Inhibition of tubulin polymerization [AID273280, Type: Literature]
View
50
[SID103500703]
[CID16090886]
IC50 1.2Inhibition of tubulin polymerization [AID273280, Type: Literature]
View