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BioActivity Data for Targets
Filters: All Data » Active      
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BioActivity Outcomes:
Active(154)
 
 
BioAssay Types:
Literature(148)
 
 
Confirmatory(6)
 
 
BioActivity Types:
IC50(129)
 
 
Ki(23)
 
 
Substance Types:
Chemical(154)
 
 
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Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 24    Data Row: 154   Total Pages: 8   Display: Page     
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#StructureSubstanceCompoundActivityBioAssayLinks
OutcomeTypeValue [μM]
1
[SID103501363]
[CID6918852]
Ki 0.001Inhibition of CDK4/Cyclin D1 [AID271733, Type: Literature]
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2
[SID103501396]
[CID10479319]
Ki 0.001Inhibition of CDK4/Cyclin D1 [AID271733, Type: Literature]
View
3
[SID103461562]
[CID5330279]
IC50 0.002Inhibition of [32P]ATP binding to Cyclin dependant kinase 4-cyclin D [AID241660, Type: Literature]
View
4
[SID103243222]
[CID44299148]
IC50 0.0029Inhibition of CDK6/Cyclin D1 (unknown origin)-mediated phosphorylation of peptide substrate incubated for 15 mins prior to substrate addition measured after 90 mins by P33-radiolabeled assay [AID745523, Type: Literature]
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5
[SID103501330]
[CID11743030]
Ki 0.003Inhibition of CDK4/Cyclin D1 [AID271733, Type: Literature]
View
6
[SID160692025]
[CID46937330]
IC50 0.003Inhibition of human CDK4/cyclin D1 expressed in baculovirus infected Sf9 cells assessed as inhibition of pRb Ser780 phosphorylation after 60 mins by TR-FRET assay [AID682622, Type: confirmatory]
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7
[SID174516437]
[CID66553053]
IC50 0.004Inhibition of CDK4/Cyclin D1 (unknown origin)-mediated phosphorylation of peptide substrate incubated for 15 mins prior to substrate addition measured after 90 mins by P33-radiolabeled assay [AID745525, Type: Literature]
View
8
[SID103461870]
[CID5330358]
IC50 0.004Inhibition of [32P]ATP binding to Cyclin dependant kinase 4-cyclin D [AID241660, Type: Literature]
View
9
[SID103461687]
[CID5330356]
IC50 0.005Inhibition of [32P]ATP binding to Cyclin dependant kinase 4-cyclin D [AID241660, Type: Literature]
View
10
[SID103461766]
[CID5330278]
IC50 0.005Inhibition of [32P]ATP binding to Cyclin dependant kinase 4-cyclin D [AID241660, Type: Literature]
View
11
[SID123083941]
[CID49840037]
IC50 0.005Inhibition of human CDK4/cyclin D1 expressed in baculovirus infected Sf21 cells after 60 mins by TR-FRET assay [AID528447, Type: Literature]
View
12
[SID103501386]
[CID11975206]
Ki 0.006Inhibition of CDK4/Cyclin D1 [AID271733, Type: Literature]
View
13
[SID103461732]
[CID5330280]
IC50 0.006Inhibition of [32P]ATP binding to Cyclin dependant kinase 4-cyclin D [AID241660, Type: Literature]
View
14
[SID103461620]
[CID5330333]
IC50 0.006Inhibition of [32P]ATP binding to Cyclin dependant kinase 4-cyclin D [AID241660, Type: Literature]
View
15
[SID160692024]
[CID49786055]
IC50 0.006Inhibition of human CDK4/cyclin D1 expressed in baculovirus infected Sf9 cells assessed as inhibition of pRb Ser780 phosphorylation after 60 mins by TR-FRET assay [AID682622, Type: confirmatory]
View
16
[SID174516437]
[CID66553053]
IC50 0.0066Inhibition of CDK6/Cyclin D1 (unknown origin)-mediated phosphorylation of peptide substrate incubated for 15 mins prior to substrate addition measured after 90 mins by P33-radiolabeled assay [AID745523, Type: Literature]
View
17
[SID103243222]
[CID44299148]
IC50 0.0066Inhibition of CDK4/Cyclin D1 (unknown origin)-mediated phosphorylation of peptide substrate incubated for 15 mins prior to substrate addition measured after 90 mins by P33-radiolabeled assay [AID745525, Type: Literature]
View
18
[SID103382397]
[CID5330254]
IC50 0.007Inhibition of [32P]ATP binding to Cyclin dependant kinase 4-cyclin D [AID241660, Type: Literature]
View
19
[SID103501306]
[CID9979700]
Ki 0.007Inhibition of CDK4/Cyclin D1 [AID271733, Type: Literature]
View
20
[SID123085735]
[CID49840176]
IC50 0.009Inhibition of human CDK4/cyclin D1 expressed in baculovirus infected Sf21 cells after 60 mins by TR-FRET assay [AID528447, Type: Literature]
View