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BioActivity Data for Targets
Filters: All Data » Active      
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BioActivity Outcomes:
Active(228)
 
 
BioAssay Types:
Literature(228)
 
 
BioActivity Types:
IC50(225)
 
 
Ki(3)
 
 
Substance Types:
Chemical(228)
 
 
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Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 13    Data Row: 228   Total Pages: 5   Display: Page     
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#StructureSubstanceCompoundActivityBioAssayLinks
OutcomeTypeValue [μM]
1
[SID103456957]
[CID11327430]
IC50 0.01Inhibitory activity against DNA-dependent protein kinase (DNA-PK) [AID241618, Type: Literature]
View
2
[SID103456957]
[CID11327430]
IC50 0.02Inhibitory activity against DNA-dependent protein kinase (DNA-PK) at 0.5 uM [AID241922, Type: Literature]
View
3
[SID103456957]
[CID11327430]
IC50 0.02Inhibitory activity against DNA-dependent protein kinase receptor [AID257403, Type: Literature]
View
4
[SID103474349]
[CID11567907]
IC50 0.023Inhibitory activity against DNA-dependent protein kinase receptor [AID257403, Type: Literature]
View
5
[SID103456957]
[CID11327430]
IC50 0.03Inhibition of DNA-PK autophosphorylation at Ser2056 residue in human CLL cells by Western blot method [AID705441, Type: Literature]
View
6
[SID103456718]
[CID11668417]
IC50 0.04Inhibitory activity against DNA-dependent protein kinase (DNA-PK) at 0.5 uM [AID241922, Type: Literature]
View
7
[SID103456718]
[CID11668417]
IC50 0.04Inhibitory activity against DNA-dependent protein kinase receptor [AID257403, Type: Literature]
View
8
[SID103174804]
[CID312145]
Ki 0.12Binding affinity for DNA dependent protein kinase isolated from HeLa cells; Range is 20-120 [AID239094, Type: Literature]
View
9
[SID103174804]
[CID312145]
Ki 0.12Inhibition of DNA-PK isolated from human HeLa cell extract [AID705450, Type: Literature]
View
10
[SID103322751]
[CID9843885]
IC50 0.16Inhibition of DNA-PK in HeLa cell nuclear extracts [AID281337, Type: Literature]
View
11
[SID103322931]
[CID16203245]
IC50 0.16Inhibition of DNA-PK in HeLa cell nuclear extracts [AID281337, Type: Literature]
View
12
[SID103323311]
[CID10062895]
IC50 0.18Inhibition of DNA-PK in HeLa cell nuclear extracts [AID281337, Type: Literature]
View
13
[SID103440799]
[CID10017389]
IC50 0.19Inhibition of DNA dependent protein kinase isolated from HeLa cells [AID241691, Type: Literature]
View
14
[SID103440799]
[CID10017389]
IC50 0.19Inhibitory activity against DNA-dependent protein kinase (DNA-PK) at 0.5 uM [AID241922, Type: Literature]
View
15
[SID103322433]
[CID16745325]
IC50 0.22Inhibition of DNA-PK in HeLa cell nuclear extracts [AID281337, Type: Literature]
View
16
[SID103322569]
[CID9860529]
IC50 0.23Inhibitory activity against DNA-dependent protein kinase (DNA-PK) [AID241618, Type: Literature]
View
17
[SID103322569]
[CID9860529]
IC50 0.23Inhibition of DNA dependent protein kinase isolated from HeLa cells [AID241691, Type: Literature]
View
18
[SID103322569]
[CID9860529]
IC50 0.23Inhibitory activity against DNA-dependent protein kinase receptor [AID257403, Type: Literature]
View
19
[SID103474152]
[CID25817490]
IC50 0.25Inhibitory activity against DNA-dependent protein kinase receptor [AID257403, Type: Literature]
View
20
[SID103322458]
[CID16203247]
IC50 0.26Inhibition of DNA-PK in HeLa cell nuclear extracts [AID281337, Type: Literature]
View
21
[SID103440761]
[CID11426483]
IC50 0.26Inhibition of DNA dependent protein kinase isolated from HeLa cells [AID241691, Type: Literature]
View
22
[SID103440754]
[CID10039361]
IC50 0.28Inhibition of DNA dependent protein kinase isolated from HeLa cells [AID241691, Type: Literature]
View
23
[SID103323038]
[CID9817915]
IC50 0.28Inhibition of DNA-PK in HeLa cell nuclear extracts [AID281337, Type: Literature]
View
24
[SID103456878]
[CID11623802]
IC50 0.3Inhibitory activity against DNA-dependent protein kinase (DNA-PK) at 0.5 uM [AID241922, Type: Literature]
View
25
[SID103456878]
[CID11623802]
IC50 0.3Inhibitory activity against DNA-dependent protein kinase receptor [AID257403, Type: Literature]
View
26
[SID103322549]
[CID21106400]
IC50 0.31Inhibition of DNA-PK in HeLa cell nuclear extracts [AID281337, Type: Literature]
View
27
[SID103323310]
[CID10912743]
IC50 0.35Inhibition of DNA-PK in HeLa cell nuclear extracts [AID281337, Type: Literature]
View
28
[SID103474041]
[CID11676414]
IC50 0.35Inhibitory activity against DNA-dependent protein kinase receptor [AID257403, Type: Literature]
View
29
[SID103440790]
[CID11737711]
IC50 0.36Inhibition of DNA dependent protein kinase isolated from HeLa cells [AID241691, Type: Literature]
View
30
[SID103310559]
[CID11522900]
IC50 0.38Inhibitory activity against DNA-dependent protein kinase receptor [AID257403, Type: Literature]
View
31
[SID103440798]
[CID11437483]
IC50 0.39Inhibition of DNA dependent protein kinase isolated from HeLa cells [AID241691, Type: Literature]
View
32
[SID103511166]
[CID21106429]
IC50 0.39Inhibition of DNA-PK in HeLa cell nuclear extracts [AID281337, Type: Literature]
View
33
[SID103511221]
[CID16203946]
IC50 0.4Inhibition of DNA-PK in HeLa cell nuclear extracts [AID281337, Type: Literature]
View
34
[SID163318299]
[CID9815659]
IC50 0.4Inhibition of DNA-PK isolated from human HeLa cell extract assessed as inhibition of p53 peptide fragment phosphorylation after 10 mins [AID705444, Type: Literature]
View
35
[SID103440798]
[CID11437483]
IC50 0.4Inhibitory activity against DNA-dependent protein kinase receptor [AID257403, Type: Literature]
View
36
[SID103473925]
[CID11631748]
IC50 0.44Inhibitory activity against DNA-dependent protein kinase receptor [AID257403, Type: Literature]
View
37
[SID103474050]
[CID11589142]
IC50 0.44Inhibitory activity against DNA-dependent protein kinase receptor [AID257403, Type: Literature]
View
38
[SID103474101]
[CID11715743]
IC50 0.45Inhibitory activity against DNA-dependent protein kinase receptor [AID257403, Type: Literature]
View
39
[SID103511197]
[CID21106425]
IC50 0.47Inhibition of DNA-PK in HeLa cell nuclear extracts [AID281337, Type: Literature]
View
40
[SID103473452]
[CID11553441]
IC50 0.47Inhibitory activity against DNA-dependent protein kinase receptor [AID257403, Type: Literature]
View
41
[SID103322432]
[CID21955998]
IC50 0.48Inhibition of DNA-PK in HeLa cell nuclear extracts [AID281337, Type: Literature]
View
42
[SID103474026]
[CID11595862]
IC50 0.49Inhibitory activity against DNA-dependent protein kinase receptor [AID257403, Type: Literature]
View
43
[SID103511318]
[CID16203940]
IC50 0.5Inhibition of DNA-PK in HeLa cell nuclear extracts [AID281337, Type: Literature]
View
44
[SID103473900]
[CID11581520]
IC50 0.5Inhibitory activity against DNA-dependent protein kinase receptor [AID257403, Type: Literature]
View
45
[SID103323039]
[CID11580379]
IC50 0.53Inhibition of DNA-PK in HeLa cell nuclear extracts [AID281337, Type: Literature]
View
46
[SID103511196]
[CID21106426]
IC50 0.53Inhibition of DNA-PK in HeLa cell nuclear extracts [AID281337, Type: Literature]
View
47
[SID103323308]
[CID21106405]
IC50 0.54Inhibition of DNA-PK in HeLa cell nuclear extracts [AID281337, Type: Literature]
View
48
[SID103456572]
[CID11660078]
IC50 0.6Inhibitory activity against DNA-dependent protein kinase (DNA-PK) at 0.5 uM [AID241922, Type: Literature]
View
49
[SID103456572]
[CID11660078]
IC50 0.6Inhibitory activity against DNA-dependent protein kinase receptor [AID257403, Type: Literature]
View
50
[SID103511228]
[CID16203948]
IC50 0.6Inhibition of DNA-PK in HeLa cell nuclear extracts [AID281337, Type: Literature]
View