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RAC-gamma serine/threonine-protein kinase; Pr.. [gi:12643943] - Target BioActivity Data
Also known as: RAC-gamma serine/threonine-protein kinase; Protein kinase Akt-3; Protein kinase B gamma; PKB gamma; RAC-PK-gamma; STK-2.
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BioActivity Outcomes:
Active(149)
 
 
BioAssay Types:
Literature(149)
 
 
BioActivity Types:
IC50(131)
 
 
Kd(10)
 
 
Ki(3)
 
 
EC50(3)
 
 
Substance Types:
Chemical(149)
 
 
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Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 21    Data Row: 149   Total Pages: 3   Display: Page     
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#StructureSubstanceCompoundActivityBioAssayLinks
OutcomeTypeValue [μM]
1
[SID103718372]
[CID46226079]
IC50 0.001Inhibition of human AKT3 [AID455026, Type: Literature]
View
2
[SID103718442]
[CID46226137]
IC50 0.001Inhibition of human AKT3 [AID455026, Type: Literature]
View
3
[SID103718472]
[CID46226156]
IC50 0.001Inhibition of human AKT3 [AID455026, Type: Literature]
View
4
[SID163331672]
[CID58458278]
IC50 0.001Competitive inhibition of wild-type full-length amino-terminal polyhistidine-tagged human Akt3 expressed in recombinant baculovirus system using fluorescence labeled Crosstide as substrate after 60 mins by fluorescence polarization assay in presence of ATP [AID708171, Type: Literature]
View
5
[SID163321303]
[CID59671151]
IC50 0.002Competitive inhibition of wild-type full-length amino-terminal polyhistidine-tagged human Akt3 expressed in recombinant baculovirus system using fluorescence labeled Crosstide as substrate after 60 mins by fluorescence polarization assay in presence of ATP [AID708171, Type: Literature]
View
6
[SID103718441]
[CID46226136]
IC50 0.002Inhibition of human AKT3 [AID455026, Type: Literature]
View
7
[SID103718373]
[CID46226080]
IC50 0.002Inhibition of human AKT3 [AID455026, Type: Literature]
View
8
[SID103718374]
[CID25190977]
IC50 0.002Inhibition of human AKT3 [AID455026, Type: Literature]
View
9
[SID163335288]
[CID58191081]
IC50 0.002Competitive inhibition of wild-type full-length amino-terminal polyhistidine-tagged human Akt3 expressed in recombinant baculovirus system using fluorescence labeled Crosstide as substrate after 60 mins by fluorescence polarization assay in presence of ATP [AID708171, Type: Literature]
View
10
[SID103495052]
[CID16043304]
IC50 0.0026Inhibition of AKT3 in presence of 0.2 uM ATP [AID269858, Type: Literature]
View
11
[SID103495052]
[CID16043304]
IC50 0.003Inhibition of AKT3 [AID269861, Type: Literature]
View
12
[SID103604655]
[CID16725726]
Kd 0.003Binding constant for AKT3 kinase domain [AID625019, Type: Literature]
View
13
[SID163338532]
[CID58191080]
IC50 0.003Competitive inhibition of wild-type full-length amino-terminal polyhistidine-tagged human Akt3 expressed in recombinant baculovirus system using fluorescence labeled Crosstide as substrate after 60 mins by fluorescence polarization assay in presence of ATP [AID708171, Type: Literature]
View
14
[SID163338659]
[CID70676464]
IC50 0.003Competitive inhibition of wild-type full-length amino-terminal polyhistidine-tagged human Akt3 expressed in recombinant baculovirus system using fluorescence labeled Crosstide as substrate after 60 mins by fluorescence polarization assay in presence of ATP [AID708171, Type: Literature]
View
15
[SID103718397]
[CID25222706]
IC50 0.003Inhibition of human AKT3 [AID455026, Type: Literature]
View
16
[SID163314381]
[CID70676312]
IC50 0.004Competitive inhibition of wild-type full-length amino-terminal polyhistidine-tagged human Akt3 expressed in recombinant baculovirus system using fluorescence labeled Crosstide as substrate after 60 mins by fluorescence polarization assay in presence of ATP [AID708171, Type: Literature]
View
17
[SID163317839]
[CID59671148]
IC50 0.004Competitive inhibition of wild-type full-length amino-terminal polyhistidine-tagged human Akt3 expressed in recombinant baculovirus system using fluorescence labeled Crosstide as substrate after 60 mins by fluorescence polarization assay in presence of ATP [AID708171, Type: Literature]
View
18
[SID164128907]
[CID42602264]
IC50 0.004Inhibition of recombinant Akt3 (unknown origin) using 5-FAM-labeled peptide as substrate after 1 hr by caliper off-chip incubation mobility shift assay [AID728521, Type: Literature]
View
19
[SID103495241]
[CID44414579]
IC50 0.0048Inhibition of AKT3 in presence of 0.2 uM ATP [AID269858, Type: Literature]
View
20
[SID103243222]
[CID44299148]
IC50 0.005Inhibition of AKT3 [AID269861, Type: Literature]
View
21
[SID163335125]
[CID70675988]
IC50 0.005Competitive inhibition of wild-type full-length amino-terminal polyhistidine-tagged human Akt3 expressed in recombinant baculovirus system using fluorescence labeled Crosstide as substrate after 60 mins by fluorescence polarization assay in presence of ATP [AID708171, Type: Literature]
View
22
[SID163314383]
[CID25170562]
IC50 0.005Competitive inhibition of wild-type full-length amino-terminal polyhistidine-tagged human Akt3 expressed in recombinant baculovirus system using fluorescence labeled Crosstide as substrate after 60 mins by fluorescence polarization assay in presence of ATP [AID708171, Type: Literature]
View
23
[SID163321306]
[CID24788432]
IC50 0.005Competitive inhibition of wild-type full-length amino-terminal polyhistidine-tagged human Akt3 expressed in recombinant baculovirus system using fluorescence labeled Crosstide as substrate after 60 mins by fluorescence polarization assay in presence of ATP [AID708171, Type: Literature]
View
24
[SID163324660]
[CID24788739]
IC50 0.005Competitive inhibition of wild-type full-length amino-terminal polyhistidine-tagged human Akt3 expressed in recombinant baculovirus system using fluorescence labeled Crosstide as substrate after 60 mins by fluorescence polarization assay in presence of ATP [AID708171, Type: Literature]
View
25
[SID163324661]
[CID24786152]
IC50 0.005Competitive inhibition of wild-type full-length amino-terminal polyhistidine-tagged human Akt3 expressed in recombinant baculovirus system using fluorescence labeled Crosstide as substrate after 60 mins by fluorescence polarization assay in presence of ATP [AID708171, Type: Literature]
View
26
[SID103718400]
[CID25221040]
IC50 0.006Inhibition of human AKT3 [AID455026, Type: Literature]
View
27
[SID164142961]
[CID57750407]
IC50 0.006Inhibition of recombinant Akt3 (unknown origin) using 5-FAM-labeled peptide as substrate after 1 hr by caliper off-chip incubation mobility shift assay [AID728521, Type: Literature]
View
28
[SID163338530]
[CID59671179]
IC50 0.007Competitive inhibition of wild-type full-length amino-terminal polyhistidine-tagged human Akt3 expressed in recombinant baculovirus system using fluorescence labeled Crosstide as substrate after 60 mins by fluorescence polarization assay in presence of ATP [AID708171, Type: Literature]
View
29
[SID163331669]
[CID59671180]
IC50 0.007Competitive inhibition of wild-type full-length amino-terminal polyhistidine-tagged human Akt3 expressed in recombinant baculovirus system using fluorescence labeled Crosstide as substrate after 60 mins by fluorescence polarization assay in presence of ATP [AID708171, Type: Literature]
View
30
[SID164145791]
[CID42602178]
IC50 0.007Inhibition of recombinant Akt3 (unknown origin) using 5-FAM-labeled peptide as substrate after 1 hr by caliper off-chip incubation mobility shift assay [AID728521, Type: Literature]
View
31
[SID163321308]
[CID24788740]
IC50 0.008Competitive inhibition of wild-type full-length amino-terminal polyhistidine-tagged human Akt3 expressed in recombinant baculovirus system using fluorescence labeled Crosstide as substrate after 60 mins by fluorescence polarization assay in presence of ATP [AID708171, Type: Literature]
View
32
[SID164134558]
[CID25227436]
IC50 0.008Inhibition of recombinant Akt3 (unknown origin) using 5-FAM-labeled peptide as substrate after 1 hr by caliper off-chip incubation mobility shift assay [AID728521, Type: Literature]
View
33
[SID103604655]
[CID16725726]
IC50 0.009Inhibition of human AKT3 [AID391376, Type: Literature]
View
34
[SID103243222]
[CID44299148]
IC50 0.01Inhibition of Akt3 using 10 uM ATP [AID262363, Type: Literature]
View
35
[SID103243222]
[CID44299148]
IC50 0.01Inhibition of Akt3 at 10 uM ATP [AID262971, Type: Literature]
View
36
[SID164142997]
[CID57750342]
IC50 0.01Inhibition of recombinant Akt3 (unknown origin) using 5-FAM-labeled peptide as substrate after 1 hr by caliper off-chip incubation mobility shift assay [AID728521, Type: Literature]
View
37
[SID163321305]
[CID24788164]
IC50 0.01Competitive inhibition of wild-type full-length amino-terminal polyhistidine-tagged human Akt3 expressed in recombinant baculovirus system using fluorescence labeled Crosstide as substrate after 60 mins by fluorescence polarization assay in presence of ATP [AID708171, Type: Literature]
View
38
[SID163314384]
[CID24783593]
IC50 0.01Competitive inhibition of wild-type full-length amino-terminal polyhistidine-tagged human Akt3 expressed in recombinant baculovirus system using fluorescence labeled Crosstide as substrate after 60 mins by fluorescence polarization assay in presence of ATP [AID708171, Type: Literature]
View
39
[SID103718399]
[CID46226096]
IC50 0.01Inhibition of human AKT3 [AID455026, Type: Literature]
View
40
[SID103495053]
[CID44414447]
IC50 0.011Inhibition of AKT3 in presence of 0.2 uM ATP [AID269858, Type: Literature]
View
41
[SID163321304]
[CID59670989]
IC50 0.012Competitive inhibition of wild-type full-length amino-terminal polyhistidine-tagged human Akt3 expressed in recombinant baculovirus system using fluorescence labeled Crosstide as substrate after 60 mins by fluorescence polarization assay in presence of ATP [AID708171, Type: Literature]
View
42
[SID163328105]
[CID25170563]
IC50 0.012Competitive inhibition of wild-type full-length amino-terminal polyhistidine-tagged human Akt3 expressed in recombinant baculovirus system using fluorescence labeled Crosstide as substrate after 60 mins by fluorescence polarization assay in presence of ATP [AID708171, Type: Literature]
View
43
[SID163335123]
[CID24788623]
IC50 0.013Competitive inhibition of wild-type full-length amino-terminal polyhistidine-tagged human Akt3 expressed in recombinant baculovirus system using fluorescence labeled Crosstide as substrate after 60 mins by fluorescence polarization assay in presence of ATP [AID708171, Type: Literature]
View
44
[SID103604655]
[CID16725726]
Ki 0.013Binding affinity to human AKT3 [AID391400, Type: Literature]
View
45
[SID164128908]
[CID57750369]
IC50 0.015Inhibition of recombinant Akt3 (unknown origin) using 5-FAM-labeled peptide as substrate after 1 hr by caliper off-chip incubation mobility shift assay [AID728521, Type: Literature]
View
46
[SID164140232]
[CID42602096]
IC50 0.015Inhibition of recombinant Akt3 (unknown origin) using 5-FAM-labeled peptide as substrate after 1 hr by caliper off-chip incubation mobility shift assay [AID728521, Type: Literature]
View
47
[SID164148586]
[CID42602260]
IC50 0.015Inhibition of recombinant Akt3 (unknown origin) using 5-FAM-labeled peptide as substrate after 1 hr by caliper off-chip incubation mobility shift assay [AID728521, Type: Literature]
View
48
[SID164148587]
[CID57750408]
IC50 0.016Inhibition of recombinant Akt3 (unknown origin) using 5-FAM-labeled peptide as substrate after 1 hr by caliper off-chip incubation mobility shift assay [AID728521, Type: Literature]
View
49
[SID103604720]
[CID25023736]
IC50 0.016Inhibition of human AKT3 [AID391376, Type: Literature]
View
50
[SID164137412]
[CID57750290]
IC50 0.018Inhibition of recombinant Akt3 (unknown origin) using 5-FAM-labeled peptide as substrate after 1 hr by caliper off-chip incubation mobility shift assay [AID728521, Type: Literature]
View