CHEMBL212965 (CID 9937660) - BioAssay Data Summary for Compound
.
BioActivity Outcomes:
Active(5)
 
 
Inactive(1)
 
 
Inconclusive(2)
 
 
Top Targets:
Firefly Luc l..(1)
 
 
PTKc EGFR(1)
 
 
PTKc HER2(1)
 
 
BioAssay Types:
Literature(5)
 
 
Confirmatory(3)
 
 
 
BioActivity Types:
IC50(5)
 
 
Potency(3)
 
 
 
SAR
Target summary
Data download

Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 8    Data Row: 8   Total Pages: 1   
Sort: [Click the result table header to sort]
#SubstanceActivityBioAssayTargetLinks
OutcomeTypeValue [μM]
1
[SID103498679]
IC50 0.012Inhibition of ErbB1 [AID270617, Type: Literature]Epidermal growth factor receptor [gi:2811086]
View
2
[SID103498679]
IC50 0.012Inhibition of ErbB1 [AID270617, Type: Literature]Epidermal growth factor receptor [gi:2811086]
View
3
[SID103498679]
IC50 0.012Inhibition of ErbB1 [AID270617, Type: Literature]Epidermal growth factor receptor [gi:2811086]
View
4
[SID103498679]
IC50 0.023Inhibition of ErbB2 [AID270616, Type: Literature]Receptor tyrosine-protein kinase erbB-2 [gi:119533]
View
5
[SID103498679]
IC50 0.023Inhibition of ErbB2 [AID270616, Type: Literature]Receptor tyrosine-protein kinase erbB-2 [gi:119533]
View
6
[SID103498679]
IC50 0.32Inhibition of HN5 cell growth after 72 hrs [AID270618, Type: Literature]
View
7
[SID103498679]
IC50 0.42Inhibition of BT474 cell growth after 72 hrs [AID270619, Type: Literature]
View
8
[SID103498679]
IC50 0.46Inhibition of N87 cell growth after 72 hrs [AID270620, Type: Literature]
View
9
[SID124350082]
Potency 0.0005qHTS Assay for Inhibitors of Sea Pansy Luciferase from the GSK Published Protein Kinase Inhibitor Set [AID652015, Type: confirmatory]Renilla-luciferin 2-monooxygenase (EC 1.13.12.5) - sea pansy (Renilla reniformis) (fragment) [gi:84399]
View
10
[SID124350082]
Potency 1.9872qHTS for Inhibitors of binding or entry into cells for Lassa Virus [AID540256, Type: confirmatory]
View
11
[SID124350082]
Potency 14.5659qHTS Assay for Inhibitors of Firefly Luciferase from the GSK Published Protein Kinase Inhibitor Set [AID652016, Type: confirmatory]Luciferase [Photinus pyralis] [gi:160794]
View