Bookmark and Share

BioActivity Data for Compound CID 9875011 (CID 9875011)

BioActivity Outcomes:
Active(9)
 
 
Unspecified(1)
 
 
BioAssay Types:
Literature(7)
 
 
 
Confirmatory(3)
 
 
BioAssay Categories:
In vitro(6)
 
 
Biochemical(3)
 
 
ADME(1)
 
 
Cell-based(9)
 
 
BioActivity Types:
EC50(9)
 
 
Data download

Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 10    Data Row: 10   Total Pages: 1   
Sort: [Click the result table header to sort]
#SubstanceActivityBioAssayTargetLinks
OutcomeTypeValue [μM]
1
[SID103547743]
EC50 0.27Agonist activity at human recombinant P2Y6 receptor expressed in human 1321N1 cells using [3H]inositol as substrate assessed as [3H]inositol phosphate formation after 30 mins by liquid scintillation counting analysis [AID1121982, Type: confirmatory]P2Y purinoceptor 6 [gi:2495018]
View
2
[SID103547743]
EC50 0.27Agonist activity at human recombinant P2Y6 receptor expressed in human 1321N1 cells assessed as [3H]inositol phosphate production by scintillation proximity assay [AID484784, Type: Literature]P2Y purinoceptor 6 [gi:2495018]
View
3
[SID103547743]
EC50 0.27Agonist activity at human P2Y6 receptor expressed in human 1321N1 cells assessed as [3H]inositol phosphate accumulation by scintillation proximity assay [AID404830, Type: Literature]P2Y purinoceptor 6 [gi:2495018]
View
4
[SID103547743]
EC50 0.87Agonist activity at human recombinant P2Y4 receptor expressed in human 1321N1 cells using [3H]inositol as substrate assessed as [3H]inositol phosphate formation after 30 mins by liquid scintillation counting analysis [AID1121979, Type: confirmatory]P2Y purinoceptor 4 [gi:1709524]
View
5
[SID103547743]
EC50 0.87Agonist activity at human recombinant P2Y4 receptor expressed in human 1321N1 cells assessed as [3H]inositol phosphate production by scintillation proximity assay [AID484777, Type: Literature]P2Y purinoceptor 4 [gi:1709524]
View
6
[SID103547743]
EC50 0.87Agonist activity at human P2Y4 receptor expressed in human 1321N1 cells assessed as [3H]inositol phosphate accumulation by scintillation proximity assay [AID404834, Type: Literature]P2Y purinoceptor 4 [gi:1709524]
View
7
[SID103547743]
EC50 1.31Agonist activity at human P2Y2 receptor expressed in human 1321N1 cells assessed as [3H]inositol phosphate accumulation by scintillation proximity assay [AID404832, Type: Literature]P2Y purinoceptor 2 [gi:311033490]
View
8
[SID103547743]
EC50 1.31Agonist activity at human recombinant P2Y2 receptor expressed in human 1321N1 cells assessed as [3H]inositol phosphate production by scintillation proximity assay [AID484783, Type: Literature]P2Y purinoceptor 2 [gi:311033490]
View
9
[SID103547743]
EC50 1.31Agonist activity at human recombinant P2Y2 receptor expressed in human 1321N1 cells using [3H]inositol as substrate assessed as [3H]inositol phosphate formation after 30 mins by liquid scintillation counting analysis [AID1121981, Type: confirmatory]P2Y purinoceptor 2 [gi:311033490]
View
10
[SID103547743]
Stability of the compound assessed as human e-NPP1-mediated hydrolysis at pH 8.5 after 20 mins by HPLC analysis [AID644880, Type: Literature]
View