SureCN4265257 (CID 9850395) - BioAssay Data Summary for Compound
.
BioActivity Outcomes:
Active(3)
 
 
Unspecified(1)
 
 
Top Targets:
NR LBD PPAR(2)
 
 
BioAssay Types:
Literature(4)
 
 
 
BioActivity Types:
EC50(3)
 
 
SAR
Target summary
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Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 4    Data Row: 4   Total Pages: 1   
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#SubstanceActivityBioAssayTargetLinks
OutcomeTypeValue [μM]
1
[SID103187549]
EC50 0.008In vitro transcriptional activation in CV-1 cells expressing human Gal4-PPAR alpha ligand binding domain [AID156137, Type: Literature]
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2
[SID103187549]
EC50 2.4In vitro transcriptional activation in CV-1 cells expressing human Gal4-PPAR gamma ligand binding domain [AID156937, Type: Literature]Peroxisome proliferator-activated receptor gamma [gi:13432234]
View
3
[SID103187549]
EC50 2.4In vitro transcriptional activation in CV-1 cells expressing human Gal4-PPAR gamma ligand binding domain [AID156937, Type: Literature]Peroxisome proliferator-activated receptor gamma [gi:13432234]
View
4
[SID103187549]
EC50 2.4In vitro transcriptional activation in CV-1 cells expressing human Gal4-PPAR gamma ligand binding domain [AID156937, Type: Literature]Peroxisome proliferator-activated receptor gamma [gi:13432234]
View
5
[SID103187549]
EC50 2.4In vitro transcriptional activation in CV-1 cells expressing human Gal4-PPAR gamma ligand binding domain [AID156937, Type: Literature]Peroxisome proliferator-activated receptor gamma [gi:13432234]
View
6
[SID103187549]
EC50 5In vitro transcriptional activation in CV-1 cells expressing human Gal4-PPAR delta ligand binding domain [AID156359, Type: Literature]Peroxisome proliferator-activated receptor delta [gi:417522]
View
7
[SID103187549]
EC50 5In vitro transcriptional activation in CV-1 cells expressing human Gal4-PPAR delta ligand binding domain [AID156359, Type: Literature]Peroxisome proliferator-activated receptor delta [gi:417522]
View
8
[SID103187549]
EC50 5In vitro transcriptional activation in CV-1 cells expressing human Gal4-PPAR delta ligand binding domain [AID156359, Type: Literature]Peroxisome proliferator-activated receptor delta [gi:417522]
View
9
[SID103187549]
 In vivo triglyceride lowering activity in fat-fed hamsters at a dose of 3 mg/kg, po for 7 days [AID84143, Type: Literature]
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