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CHEMBL318351 (CID 9825046) - Compound BioActivity Data
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BioActivity Outcomes:
Active(6)
 
 
Unspecified(2)
 
 
Top Targets:
NR LBD PPAR(8)
 
 
 
BioAssay Types:
Literature(8)
 
 
 
BioActivity Types:
EC50(6)
 
 
Data download

Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 8    Data Row: 8   Total Pages: 1   
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#SubstanceActivityBioAssayTargetLinks
OutcomeTypeValue [μM]
1
[SID103326409]
EC50 0.000615Transcriptional activation activity on human Peroxisome proliferator activated receptor alpha expressed in CHO-K1 cells [AID156124, Type: Literature]Peroxisome proliferator-activated receptor alpha [gi:3041727]
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2
[SID103326409]
EC50 0.013Transactivation of human PPARalpha expressed in CHO-K1 cells [AID638935, Type: Literature]Peroxisome proliferator-activated receptor alpha [gi:3041727]
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3
[SID103326409]
EC50 0.014Transcriptional activation activity on human T279M-mutant Peroxisome proliferator activated receptor alpha expressed in CHO-K1 cells [AID156126, Type: Literature]Peroxisome proliferator-activated receptor alpha [gi:3041727]
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4
[SID103326409]
EC50 0.667Transcriptional activation activity on human I272F-mutant Peroxisome proliferator activated receptor alpha expressed in CHO-K1 cells [AID156125, Type: Literature]Peroxisome proliferator-activated receptor alpha [gi:3041727]
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5
[SID103326409]
EC50 1.92Transactivation of human PPARdelta expressed in CHO-K1 cells [AID638937, Type: Literature]Peroxisome proliferator-activated receptor delta [gi:417522]
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6
[SID103326409]
EC50 2.5Transactivation of human PPARgamma expressed in CHO-K1 cells [AID638936, Type: Literature]Peroxisome proliferator-activated receptor gamma [gi:13432234]
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7
[SID103326409]
Ratio of transcriptional activation of I272F mutant compared to wild type PPAR-GAL4 chimeric receptors in CHO-K1 cells [AID156303, Type: Literature]Peroxisome proliferator-activated receptor alpha [gi:3041727]
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8
[SID103326409]
Ratio of transcriptional activation of T279M mutant compared to wild type PPAR-GAL4 chimeric receptors in CHO-K1 cells [AID156306, Type: Literature]Peroxisome proliferator-activated receptor alpha [gi:3041727]
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