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N-desmethyl loperamide (CID 9805944) - Compound BioActivity Data
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BioActivity Outcomes:
Active(12)
 
 
Unspecified(33)
 
 
Top Targets:
7tm 4(12)
 
 
SLC6sbd SERT(2)
 
 
 
ERG2 Sigma1R(2)
 
 
 
SLC6sbd NET(1)
 
 
DUF3353(1)
 
 
BioAssay Types:
Literature(45)
 
 
 
BioActivity Types:
Ki(12)
 
 
Data download

Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 45    Data Row: 45   Total Pages: 3   Display: Page     
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#SubstanceActivityBioAssayTargetLinks
OutcomeTypeValue [μM]
1
[SID103606134]
Ki 0.0006Displacement of [3H]DAMGO from mu opioid receptor [AID391603, Type: Literature]
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2
[SID103606134]
Ki 0.0008Displacement of [3H]Pentazocine from rat sigma 1 receptor in rat PC12 cells [AID391604, Type: Literature]Sigma non-opioid intracellular receptor 1 [gi:81882051]
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3
[SID103606134]
Ki 0.001Displacement of [125I]HEAT from adrenergic alpha2A receptor [AID391596, Type: Literature]
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4
[SID103606134]
Ki 0.0011Displacement of [3H]N-methylspiperone from dopamine D4 receptor [AID391599, Type: Literature]
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5
[SID103606134]
Ki 0.0017Displacement of [3H]tiotidine from human histamine H2 receptor [AID391601, Type: Literature]Histamine H2 receptor [gi:123120]
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6
[SID103606134]
Ki 0.0019Displacement of [3H]DTG from rat sigma 2 receptor in rat PC12 cells [AID391605, Type: Literature]
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7
[SID103606134]
Ki 0.0024Displacement of [125I]HEAT from adrenergic Alpha-2C receptor [AID391597, Type: Literature]
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8
[SID103606134]
Ki 0.0042Displacement of [3H]pyrilamine from human histamine H1 receptor [AID391600, Type: Literature]Histamine H1 receptor [gi:547645]
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9
[SID103606134]
Ki 0.0062Displacement of [3H]citalopram from human SERT [AID391606, Type: Literature]Sodium-dependent serotonin transporter [gi:400630]
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10
[SID103606134]
Ki 0.007Displacement of [125I]HEAT from adrenergic alpha2B receptor [AID391598, Type: Literature]
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11
[SID103606134]
Ki 0.0093Displacement of [3H]alpha-methylhistamine from human histamine H3 receptor [AID391602, Type: Literature]Histamine H3 receptor [gi:17367264]
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12
[SID103606134]
Ki 0.0099Displacement of [125I]HEAT from adrenergic alpha1A receptor [AID391595, Type: Literature]
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13
[SID103606134]
Displacement of [3H]DADLE from human delta opioid receptor at 10 uM [AID391305, Type: Literature]Delta-type opioid receptor [gi:311033488]
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14
[SID103606134]
Displacement of [3H]QNB from human muscarinic M4 receptor at 10 uM [AID391303, Type: Literature]Muscarinic acetylcholine receptor M4 [gi:23503039]
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15
[SID103606134]
Displacement of [3H]pentazocine from rat sigma 1 receptor in rat PC12 cells at 10 uM [AID391317, Type: Literature]Sigma non-opioid intracellular receptor 1 [gi:81882051]
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16
[SID103606134]
Displacement of [3H]LSD from human 5HT2B receptor at 10 uM [AID391293, Type: Literature]5-hydroxytryptamine receptor 2B [gi:1168220]
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17
[SID103606134]
Displacement of [3H]alpha-methylhistamine from human histamine H3 receptor at 10 uM [AID391315, Type: Literature]Histamine H3 receptor [gi:17367264]
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18
[SID103606134]
Displacement of [3H]U69593 from rat kappa opioid receptor at 10 uM [AID391304, Type: Literature]Kappa-type opioid receptor [gi:464313]
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19
[SID103606134]
Displacement of [3H]ketanserin from human 5HT2A receptor at 10 uM [AID391292, Type: Literature]5-hydroxytryptamine receptor 2A [gi:543727]
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20
[SID103606134]
Displacement of [3H]pyrilamine from human histamine H1 receptor at 10 uM [AID391313, Type: Literature]Histamine H1 receptor [gi:547645]
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