| 1 | [SID103594953] | Active | GI50 | 0.05 | Antiproliferative activity against human HCT116 cells [AID600789, Type: Literature] | |   View X | Row No. | 1 | | Structure | 
| | Substance | | | SID | 103594953 | | CID | 96851 | | Outcome | Active | | GI50 | 0.05 [uM] | | BioAssay | Antiproliferative activity against human HCT116 cells | | AID | 600789 | | BioAssay type | Literature | | Target | | | PubMed | 21526763 | | Data Table | |
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| 2 | [SID103594953] | Active | GI50 | 0.05 | Cytotoxicity against human HCT116 cells by SRB assay [AID393508, Type: Literature] | | View X | Row No. | 2 | | Structure |
| | Substance | | | SID | 103594953 | | CID | 96851 | | Outcome | Active | | GI50 | 0.05 [uM] | | BioAssay | Cytotoxicity against human HCT116 cells by SRB assay | | AID | 393508 | | BioAssay type | Literature | | Target | | | PubMed | 19256508 | | Data Table | |
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| 3 | [SID103594953] | Active | Ki | 4.46 | Inhibition of HSP70 by fluorescence polarization assay [AID600787, Type: Literature] | | View X | Row No. | 3 | | Structure |
| | Substance | | | SID | 103594953 | | CID | 96851 | | Outcome | Active | | Ki | 4.46 [uM] | | BioAssay | Inhibition of HSP70 by fluorescence polarization assay | | AID | 600787 | | BioAssay type | Literature | | Target | | | PubMed | 21526763 | | Data Table | |
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| 4 | [SID103594953] | Active | Kd | 6.8 | Binding affinity to histidine-tagged Grp78 by surface plasmon resonance analysis [AID600785, Type: Literature] | | View X | Row No. | 4 | | Structure |
| | Substance | | | SID | 103594953 | | CID | 96851 | | Outcome | Active | | Kd | 6.8 [uM] | | BioAssay | Binding affinity to histidine-tagged Grp78 by surface plasmon resonance analysis | | AID | 600785 | | BioAssay type | Literature | | Target | | | PubMed | 21526763 | | Data Table | |
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| 5 | [SID103594953] | Active | IC50 | 9.4 | Displacement of fluorescein labeled N6-(6-amino)hexyl-ATP-5-FAM from HSP70 by fluorescence polarization assay [AID393506, Type: Literature] | | View X | Row No. | 5 | | Structure |
| | Substance | | | SID | 103594953 | | CID | 96851 | | Outcome | Active | | IC50 | 9.4 [uM] | | BioAssay | Displacement of fluorescein labeled N6-(6-amino)hexyl-ATP-5-FAM from HSP70 by fluorescence polarization assay | | AID | 393506 | | BioAssay type | Literature | | Target | | | PubMed | 19256508 | | Data Table | |
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| 6 | [SID103594953] | Active | Kd | 11 | Binding affinity to HSP70 by Biocore direct binding assay [AID393507, Type: Literature] | | View X | Row No. | 6 | | Structure |
| | Substance | | | SID | 103594953 | | CID | 96851 | | Outcome | Active | | Kd | 11 [uM] | | BioAssay | Binding affinity to HSP70 by Biocore direct binding assay | | AID | 393507 | | BioAssay type | Literature | | Target | | | PubMed | 19256508 | | Data Table | |
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| 7 | [SID103594953] | Active | Kd | 11 | Binding affinity to HSP70 by surface plasmon resonance analysis [AID600786, Type: Literature] | | View X | Row No. | 7 | | Structure |
| | Substance | | | SID | 103594953 | | CID | 96851 | | Outcome | Active | | Kd | 11 [uM] | | BioAssay | Binding affinity to HSP70 by surface plasmon resonance analysis | | AID | 600786 | | BioAssay type | Literature | | Target | | | PubMed | 21526763 | | Data Table | |
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| 8 | [SID103594953] | Active | Kd | 14.14 | Binding affinity to Grp78 by isothermal titration calorimetric analysis [AID600788, Type: Literature] | | View X | Row No. | 8 | | Structure |
| | Substance | | | SID | 103594953 | | CID | 96851 | | Outcome | Active | | Kd | 14.14 [uM] | | BioAssay | Binding affinity to Grp78 by isothermal titration calorimetric analysis | | AID | 600788 | | BioAssay type | Literature | | Target | | | PubMed | 21526763 | | Data Table | |
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| 9 | [SID103594953] | Unspecified | Ki | 89.5 | Inhibition of calf placental adenosine deaminase by Lineweaver-Burk plot analysis [AID554262, Type: Literature] | Adenosine deaminase [gi:20141178] | View X | Row No. | 9 | | Structure |
| | Substance | | | SID | 103594953 | | CID | 96851 | | Outcome | Unspecified | | Ki | 89.5 [uM] | | BioAssay | Inhibition of calf placental adenosine deaminase by Lineweaver-Burk plot analysis | | AID | 554262 | | BioAssay type | Literature | | Target | Adenosine deaminase [gi:20141178] | | PubMed | 21138280 | | Data Table | |
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| 10 | [SID103594953] | Unspecified | IC50 | 400 | Binding affinity to HSP90 by fluorescence polarization assay [AID393511, Type: Literature] | | View X | Row No. | 10 | | Structure |
| | Substance | | | SID | 103594953 | | CID | 96851 | | Outcome | Unspecified | | IC50 | 400 [uM] | | BioAssay | Binding affinity to HSP90 by fluorescence polarization assay | | AID | 393511 | | BioAssay type | Literature | | Target | | | PubMed | 19256508 | | Data Table | |
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| 11 | [SID103594953] | Unspecified | | | Cytotoxicity against mouse J774A1 cells [AID584550, Type: Literature] | | View X | Row No. | 11 | | Structure |
| | Substance | | | SID | 103594953 | | CID | 96851 | | Outcome | Unspecified | | BioAssay | Cytotoxicity against mouse J774A1 cells | | AID | 584550 | | BioAssay type | Literature | | Target | | | PubMed | 20921305 | | Data Table | |
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| 12 | [SID103594953] | Inactive | | | Inhibition of HSP70 in human HCT116 cells assessed as reduction of He2 protein levels after 24 hrs by western blot [AID393509, Type: Literature] | | View X | Row No. | 12 | | Structure |
| | Substance | | | SID | 103594953 | | CID | 96851 | | Outcome | Inactive | | BioAssay | Inhibition of HSP70 in human HCT116 cells assessed as reduction of He2 protein levels after 24 hrs by western blot | | AID | 393509 | | BioAssay type | Literature | | Target | | | PubMed | 19256508 | | Data Table | |
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| 13 | [SID103594953] | Inactive | | | Inhibition of HSP70 in human HCT116 cells assessed as reduction of Raf1 protein levels after 24 hrs by western blot [AID393510, Type: Literature] | | View X | Row No. | 13 | | Structure |
| | Substance | | | SID | 103594953 | | CID | 96851 | | Outcome | Inactive | | BioAssay | Inhibition of HSP70 in human HCT116 cells assessed as reduction of Raf1 protein levels after 24 hrs by western blot | | AID | 393510 | | BioAssay type | Literature | | Target | | | PubMed | 19256508 | | Data Table | |
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| 14 | [SID103594953] | Inactive | IC50 | | Inhibition of inosine/L-alanine-induced Bacillus anthracis Sterne 34F2 spore germination pretreated for 15 mins before inosine/L-alanine challenge [AID584546, Type: Literature] | | View X | Row No. | 14 | | Structure |
| | Substance | | | SID | 103594953 | | CID | 96851 | | Outcome | Inactive | | IC50 | [uM] | | BioAssay | Inhibition of inosine/L-alanine-induced Bacillus anthracis Sterne 34F2 spore germination pretreated for 15 mins before inosine/L-alanine challenge | | AID | 584546 | | BioAssay type | Literature | | Target | | | PubMed | 20921305 | | Data Table | |
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| 15 | [SID103594953] | Inactive | IC50 | | Antibacterial activity against Bacillus anthracis Sterne 34F2 infected in mouse J774A.1 cells assessed as protection against bacteria-induced cytotoxicity using propidium iodide staining after 3 hrs measured every hours for up to 7 hrs [AID584547, Type: Literature] | | View X | Row No. | 15 | | Structure |
| | Substance | | | SID | 103594953 | | CID | 96851 | | Outcome | Inactive | | IC50 | [uM] | | BioAssay | Antibacterial activity against Bacillus anthracis Sterne 34F2 infected in mouse J774A.1 cells assessed as protection against bacteria-induced cytotoxicity using propidium iodide staining after 3 hrs measured every hours for up to 7 hrs | | AID | 584547 | | BioAssay type | Literature | | Target | | | PubMed | 20921305 | | Data Table | |
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| 16 | [SID103594953] | Inactive | | | Activation of Bacillus anthracis Sterne 34F2 spore germination after 1 hr [AID584549, Type: Literature] | | View X | Row No. | 16 | | Structure |
| | Substance | | | SID | 103594953 | | CID | 96851 | | Outcome | Inactive | | BioAssay | Activation of Bacillus anthracis Sterne 34F2 spore germination after 1 hr | | AID | 584549 | | BioAssay type | Literature | | Target | | | PubMed | 20921305 | | Data Table | |
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Chemical Probe 
Active 
Inactive 
Inconclusive 
Unspecified 
