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MLS000724462 (CID 9653891) - Compound BioActivity Data
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BioActivity Outcomes:
Active(2)
 
 
Inactive(687)
 
 
Inconclusive(7)
 
 
Unspecified(6)
 
 
Top Targets:
7TM GPCR Srx(23)
 
 
7TM GPCR Srsx(17)
 
 
Bcl-2 like(11)
 
 
alkPPc(10)
 
 
G-alpha(8)
 
 
 
BioAssay Types:
Screening(478)
 
 
 
 
Confirmatory(195)
 
 
 
 
Literature(16)
 
 
 
BioActivity Types:
Potency(142)
 
 
 
 
IC50(40)
 
 
 
EC50(8)
 
 
Data download

Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 636    Data Row: 702   Total Pages: 36   Display: Page     
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#SubstanceActivityBioAssayTargetLinks
OutcomeTypeValue [μM]
1
[SID24810136]
Aqueous Solubility from MLSMR Stock Solutions [AID1996, Type: other]
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2
[SID24810136]
HTS to identify compounds that promote myeloid differentiation with MLPCN compound set [AID624256, Type: screening] [geneid:3205]
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3
[SID174496118]
IC50 58.3Inhibition of Escherichia coli N-terminal His-tagged full length FabH expressed in Escherichia coli BL21 (DE3) using [3H]acetyl-CoA as substrate assessed as incorporation of [3H] signal into product after 25 mins by liquid scintillation counting analysis [AID749374, Type: Literature]
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4
[SID174496118]
Antimicrobial activity against Staphylococcus aureus ATCC 6538 after 24 hrs by two fold serial dilution method [AID749375, Type: Literature]
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5
[SID174496118]
Antimicrobial activity against Bacillus subtilis ATCC 530 after 24 hrs by two fold serial dilution method [AID749376, Type: Literature]
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6
[SID174496118]
Antimicrobial activity against Pseudomonas aeruginosa ATCC 27853 after 24 hrs by two fold serial dilution method [AID749377, Type: Literature]
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7
[SID174496118]
Antimicrobial activity against Escherichia coli ATCC 25922 after 24 hrs by two fold serial dilution method [AID749378, Type: Literature]
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8
[SID24810136]
Potency qHTS for Inhibitors of Human Acid Sphingomyelinase Assay: Native Substrate [AID624178, Type: confirmatory]acid sphingomyelinase [Homo sapiens] [gi:179095]
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9
[SID24810136]
Potency Inhibitors of Secretory Acid Sphingomyelinase (S-ASM): qHTS [AID504937, Type: confirmatory]acid sphingomyelinase [Homo sapiens] [gi:179095]
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10
[SID24810136]
Development of CDK5 inhibitors Measured in Biochemical System Using Plate Reader - 2083-01_Inhibitor_SinglePoint_HTS_Activity [AID488839, Type: screening]Cyclin-dependent kinase 5, regulatory subunit 1 (p35) [Homo sapiens] [gi:20072248]
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11
[SID24810136]
High-Throughput Screening for Modulators of Cytosolic Chaperonin Activity [AID651819, Type: screening]TRIC [Homo sapiens] [gi:83758679]
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12
[SID24810136]
Development of Small Molecule Probes of the Histone Methyltransferase, NSD2 Measured in Biochemical System Using Plate Reader - 7053-01_Inhibitor_SinglePoint_HTS_Activity_Set2 [AID743445, Type: screening]histone-lysine N-methyltransferase NSD2 isoform 1 [Homo sapiens] [gi:109633019]
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13
[SID24810136]
Fluorescence polarization-based cell-based primary high throughput screening assay to identify activators of insulin-degrading enzyme (IDE) [AID493087, Type: screening]insulin-degrading enzyme isoform 1 [Homo sapiens] [gi:155969707]
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14
[SID24810136]
Fluorescence polarization-based cell-based primary high throughput screening assay to identify inhibitors of insulin-degrading enzyme (IDE) [AID434962, Type: screening]insulin-degrading enzyme isoform 1 [Homo sapiens] [gi:155969707]
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15
[SID24810136]
uHTS identification of modulators of interaction between CendR and NRP-1 using Fluorescence Polarization assay [AID602438, Type: screening]Chain A, Crystal Structure Of The B1b2 Domains From Human Neuropilin-1 [gi:160877737]
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16
[SID24810136]
Fluorescence-based biochemical high throughput primary assay to identify inhibitors of Trypanosoma brucei RNA editing ligase 1 (TbREL1) [AID1117264, Type: screening]RNA-editing ligase 1, mitochondrial [gi:342179211]
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17
[SID24810136]
qHTS Assay for Inhibitors of the Six1/Eya2 Interaction [AID651725, Type: screening]six1 [Homo sapiens] [gi:1246761]
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18
[SID24810136]
Potency qHTS of GLP-1 Receptor Inverse Agonists (Inhibition Mode) [AID624417, Type: confirmatory]glp-1 receptor, partial [Homo sapiens] [gi:1724069]
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19
[SID24810136]
Potency qHTS of GLP-1 Receptor Agonists [AID624172, Type: confirmatory]glp-1 receptor, partial [Homo sapiens] [gi:1724069]
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20
[SID24810136]
Potency qHTS Assay for Inhibitors of RanGTP induced Rango (Ran-regulated importin-beta cargo) - Importin beta complex dissociation [AID540253, Type: confirmatory]snurportin-1 [Homo sapiens] [gi:5031833]
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